Highly effective combination of LSD1 (KDM1A) antagonist and pan-histone deacetylase inhibitor against human AML cells
Fiskus, W, Sharma, S, Shah, B, Portier, B P, Devaraj, S G T, Liu, K, Iyer, S P, Bearss, D, Bhalla, K N
Published in Leukemia (01.11.2014)
Published in Leukemia (01.11.2014)
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Journal Article
BET protein proteolysis targeting chimera (PROTAC) exerts potent lethal activity against mantle cell lymphoma cells
Sun, B, Fiskus, W, Qian, Y, Rajapakshe, K, Raina, K, Coleman, K G, Crew, A P, Shen, A, Saenz, D T, Mill, C P, Nowak, A J, Jain, N, Zhang, L, Wang, M, Khoury, J D, Coarfa, C, Crews, C M, Bhalla, K N
Published in Leukemia (01.02.2018)
Published in Leukemia (01.02.2018)
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Novel BET protein proteolysis-targeting chimera exerts superior lethal activity than bromodomain inhibitor (BETi) against post-myeloproliferative neoplasm secondary (s) AML cells
Saenz, D T, Fiskus, W, Qian, Y, Manshouri, T, Rajapakshe, K, Raina, K, Coleman, K G, Crew, A P, Shen, A, Mill, C P, Sun, B, Qiu, P, Kadia, T M, Pemmaraju, N, DiNardo, C, Kim, M-S, Nowak, A J, Coarfa, C, Crews, C M, Verstovsek, S, Bhalla, K N
Published in Leukemia (01.09.2017)
Published in Leukemia (01.09.2017)
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Journal Article
SPOP regulates prostate epithelial cell proliferation and promotes ubiquitination and turnover of c-MYC oncoprotein
Geng, C, Kaochar, S, Li, M, Rajapakshe, K, Fiskus, W, Dong, J, Foley, C, Dong, B, Zhang, L, Kwon, O-J, Shah, S S, Bolaki, M, Xin, L, Ittmann, M, O'Malley, B W, Coarfa, C, Mitsiades, N
Published in Oncogene (17.08.2017)
Published in Oncogene (17.08.2017)
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Comprehensive proteomic profiling identifies the androgen receptor axis and other signaling pathways as targets of microRNAs suppressed in metastatic prostate cancer
Coarfa, C, Fiskus, W, Eedunuri, V K, Rajapakshe, K, Foley, C, Chew, S A, Shah, S S, Geng, C, Shou, J, Mohamed, J S, O'Malley, B W, Mitsiades, N
Published in Oncogene (05.05.2016)
Published in Oncogene (05.05.2016)
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Journal Article
BET protein bromodomain inhibitor-based combinations are highly active against post-myeloproliferative neoplasm secondary AML cells
Saenz, Dyana T, Fiskus, Warren, Manshouri, Taghi, Rajapakshe, Kimal, Krieger, Stephanie, Sun, Baohua, Mill, Christopher P, DiNardo, Courtney, Pemmaraju, Naveen, Kadia, Tapan, Parmar, Simrit, Sharma, Sunil, Coarfa, Cristian, Qiu, Peng, Verstovsek, Srdan, Bhalla, Kapil N
Published in Leukemia (01.03.2017)
Published in Leukemia (01.03.2017)
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Journal Article
Pre-clinical efficacy of combined therapy with novel β-catenin antagonist BC2059 and histone deacetylase inhibitor against AML cells
Fiskus, W, Sharma, S, Saha, S, Shah, B, Devaraj, S G T, Sun, B, Horrigan, S, Leveque, C, Zu, Y, Iyer, S, Bhalla, K N
Published in Leukemia (01.06.2015)
Published in Leukemia (01.06.2015)
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Phase I–II study of vorinostat plus paclitaxel and bevacizumab in metastatic breast cancer: evidence for vorinostat-induced tubulin acetylation and Hsp90 inhibition in vivo
Ramaswamy, B., Fiskus, W., Cohen, B., Pellegrino, C., Hershman, D. L., Chuang, E., Luu, Thehang, Somlo, G., Goetz, M., Swaby, R., Shapiro, C. L., Stearns, V., Christos, P., Espinoza-Delgado, I., Bhalla, K., Sparano, J. A.
Published in Breast cancer research and treatment (01.04.2012)
Published in Breast cancer research and treatment (01.04.2012)
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Journal Article
HEXIM1 induction is mechanistically involved in mediating anti-AML activity of BET protein bromodomain antagonist
Devaraj, S G T, Fiskus, W, Shah, B, Qi, J, Sun, B, Iyer, S P, Sharma, S, Bradner, J E, Bhalla, K N
Published in Leukemia (01.02.2016)
Published in Leukemia (01.02.2016)
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Journal Article
Highly effective combination of LSD1 (KDM1A) antagonist and pan-histone deacetylase inhibitor against human AML cells
Fiskus, W, Sharma, S, Shah, B, Portier, B P, Devaraj, S G T, Liu, K, Iyer, S P, Bearss, D, Bhalla, K N
Published in Leukemia (01.07.2017)
Published in Leukemia (01.07.2017)
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Journal Article
515 Superior Efficacy of Co-treatment with NPM1 Antagonist and FLT3 Inhibitor or Pan-histone Deacetylase Inhibitor Against Cultured and Primary Human AML Cells Co-expressing Mutant NPM1 and FLT3-ITD
Balusu, R, Huffman, N, Fiskus, W, Smith, J, Peth, K, Hembruff, S, Rao, R, Ganguly, S, McGuirk, J, Bhalla, K.N
Published in European journal of cancer (1990) (01.11.2012)
Published in European journal of cancer (1990) (01.11.2012)
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51 Deacetylation and inactivation of peroxiredoxin by SIRT2 increases sensitivity of breast cancer cells to oxidative stress
Kandaswamy, V. Coothan, Chen, J, Fiskus, W, Rao, R, Nalluri, S, Buckley, K, Balusu, R, Bhalla, K
Published in European journal of cancer supplements (2010)
Published in European journal of cancer supplements (2010)
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Journal Article
Inhibition of histone deacetylase 6 acetylates and disrupts the chaperone function of heat shock protein 90: a novel basis for antileukemia activity of histone deacetylase inhibitors
Bali, Purva, Pranpat, Michael, Bradner, James, Balasis, Maria, Fiskus, Warren, Guo, Fei, Rocha, Kathy, Kumaraswamy, Sandhya, Boyapalle, Sandhya, Atadja, Peter, Seto, Edward, Bhalla, Kapil
Published in The Journal of biological chemistry (22.07.2005)
Published in The Journal of biological chemistry (22.07.2005)
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Targetable genetic alterations of TCF4 ( E2-2 ) drive immunoglobulin expression in diffuse large B cell lymphoma
Jain, Neeraj, Hartert, Keenan, Tadros, Saber, Fiskus, Warren, Havranek, Ondrej, Ma, Man Chun John, Bouska, Alyssa, Heavican, Tayla, Kumar, Dhiraj, Deng, Qing, Moore, Dalia, Pak, Christine, Liu, Chih Long, Gentles, Andrew J, Hartmann, Elena, Kridel, Robert, Smedby, Karin Ekstrom, Juliusson, Gunnar, Rosenquist, Richard, Gascoyne, Randy D, Rosenwald, Andreas, Giancotti, Filippo, Neelapu, Sattva S, Westin, Jason, Vose, Julie M, Lunning, Matthew A, Greiner, Timothy, Rodig, Scott, Iqbal, Javeed, Alizadeh, Ash A, Davis, R Eric, Bhalla, Kapil, Green, Michael R
Published in Science translational medicine (19.06.2019)
Published in Science translational medicine (19.06.2019)
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Journal Article
Combination of the histone deacetylase inhibitor LBH589 and the hsp90 inhibitor 17-AAG is highly active against human CML-BC cells and AML cells with activating mutation of FLT-3
George, Prince, Bali, Purva, Annavarapu, Srinivas, Scuto, Anna, Fiskus, Warren, Guo, Fei, Sigua, Celia, Sondarva, Gautam, Moscinski, Lynn, Atadja, Peter, Bhalla, Kapil
Published in Blood (15.02.2005)
Published in Blood (15.02.2005)
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Journal Article
Highly effective combination of LSD1
Devaraj, S G T, Portier, B P, Shah, B, Fiskus, W, Sharma, S, Bearss, D, Bhalla, K N, Liu, K, Iyer, S P
Published in Leukemia (01.07.2017)
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Published in Leukemia (01.07.2017)
Journal Article
Erratum: Highly effective combination of LSD1 (KDM1A) antagonist and pan-histone deacetylase inhibitor against human AML cells
Fiskus, W, Sharma, S, Shah, B, Portier, B P, Devaraj, S G T, Liu, K, Iyer, S P, Bearss, D, Bhalla, K N
Published in Leukemia (01.07.2017)
Published in Leukemia (01.07.2017)
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Journal Article
Activity of Suberoylanilide Hydroxamic Acid Against Human Breast Cancer Cells with Amplification of Her-2
BALI, Purva, PRANPAT, Michael, SWABY, Ramona, FISKUS, Warren, YAMAGUCHI, Hirohito, BALASIS, Maria, ROCHA, Kathy, WANG, Hong-Gang, RICHON, Victoria, BHALLA, Kapil
Published in Clinical cancer research (01.09.2005)
Published in Clinical cancer research (01.09.2005)
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Journal Article
Abrogation of heat shock protein 70 induction as a strategy to increase antileukemia activity of heat shock protein 90 inhibitor 17-allylamino-demethoxy geldanamycin
FEI GUO, ROCHA, Kathy, LAWRENCE, Nicholas, BHALLA, Kapil, BALI, Purva, PRANPAT, Michael, FISKUS, Warren, BOYAPALLE, Sandhya, KUMARASWAMY, Sandhya, BALASIS, Maria, GREEDY, Benjamin, ARMITAGE, E. Simon M
Published in Cancer research (Chicago, Ill.) (15.11.2005)
Published in Cancer research (Chicago, Ill.) (15.11.2005)
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Journal Article
BET protein proteolysis targeting chimera
Jain, N, Zhang, L, Coarfa, C, Saenz, D T, Mill, C P, Crews, C M, Qian, Y, Raina, K, Nowak, A J, Rajapakshe, K, Coleman, K G, Wang, M, Shen, A, Fiskus, W, Khoury, J D, Sun, B, Crew, A P, Bhalla, K N
Published in Leukemia (01.02.2018)
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Published in Leukemia (01.02.2018)
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