Structural basis of metallo-β-lactamase, serine-β-lactamase and penicillin-binding protein inhibition by cyclic boronates
Brem, Jürgen, Cain, Ricky, Cahill, Samuel, McDonough, Michael A, Clifton, Ian J, Jiménez-Castellanos, Juan-Carlos, Avison, Matthew B, Spencer, James, Fishwick, Colin W G, Schofield, Christopher J
Published in Nature communications (08.08.2016)
Published in Nature communications (08.08.2016)
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Structure-based discovery of antibacterial drugs
Fishwick, Colin W. G, Simmons, Katie J, Chopra, Ian
Published in Nature reviews. Microbiology (01.07.2010)
Published in Nature reviews. Microbiology (01.07.2010)
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Journal Article
Cyclic Boronates Inhibit All Classes of β-Lactamases
Cahill, Samuel T, Cain, Ricky, Wang, David Y, Lohans, Christopher T, Wareham, David W, Oswin, Henry P, Mohammed, Jabril, Spencer, James, Fishwick, Colin W G, McDonough, Michael A, Schofield, Christopher J, Brem, Jürgen
Published in Antimicrobial agents and chemotherapy (01.04.2017)
Published in Antimicrobial agents and chemotherapy (01.04.2017)
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Inhibition of D-Ala:D-Ala ligase through a phosphorylated form of the antibiotic D-cycloserine
Batson, Sarah, de Chiara, Cesira, Majce, Vita, Lloyd, Adrian J, Gobec, Stanislav, Rea, Dean, Fülöp, Vilmos, Thoroughgood, Christopher W, Simmons, Katie J, Dowson, Christopher G, Fishwick, Colin W G, de Carvalho, Luiz Pedro S, Roper, David I
Published in Nature communications (05.12.2017)
Published in Nature communications (05.12.2017)
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Journal Article
Mutations in 15-hydroxyprostaglandin dehydrogenase cause primary hypertrophic osteoarthropathy
Bonthron, David T, Uppal, Sandeep, Diggle, Christine P, Carr, Ian M, Fishwick, Colin W G, Ahmed, Mushtaq, Ibrahim, Gamal H, Helliwell, Philip S, Latos-Biele ska, Anna, Phillips, Simon E V, Markham, Alexander F, Bennett, Christopher P
Published in Nature genetics (01.06.2008)
Published in Nature genetics (01.06.2008)
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Natural and synthetic flavonoid modulation of TRPC5 channels
Naylor, Jacqueline, Minard, Aisling, Gaunt, Hannah J, Amer, Mohamed S, Wilson, Lesley A, Migliore, Marco, Cheung, Sin Y, Rubaiy, Hussein N, Blythe, Nicola M, Musialowski, Katie E, Ludlow, Melanie J, Evans, William D, Green, Ben L, Yang, Hongjun, You, Yun, Li, Jing, Fishwick, Colin W G, Muraki, Katsuhiko, Beech, David J, Bon, Robin S
Published in British journal of pharmacology (01.02.2016)
Published in British journal of pharmacology (01.02.2016)
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Journal Article
Determinants of Hepatitis C Virus p7 Ion Channel Function and Drug Sensitivity Identified In Vitro
STGELAIS, Corine, FOSTER, Toshana L, VEROW, Mark, ATKINS, Elizabeth, FISHWICK, Colin W. G, ROWLANDS, David, HARRIS, Mark, GRIFFIN, Stephen
Published in Journal of Virology (01.08.2009)
Published in Journal of Virology (01.08.2009)
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Journal Article
Buttock Claudication and Erectile Dysfunction After Internal Iliac Artery Embolization in Patients Prior to Endovascular Aortic Aneurysm Repair
Rayt, H. S., Bown, M. J., Lambert, K. V., Fishwick, N. G., McCarthy, M. J., London, N. J. M., Sayers, R. D.
Published in Cardiovascular and interventional radiology (01.07.2008)
Published in Cardiovascular and interventional radiology (01.07.2008)
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Journal Article
Affimer proteins inhibit immune complex binding to FcγRIIIa with high specificity through competitive and allosteric modes of action
Robinson, James I., Baxter, Euan W., Owen, Robin L., Thomsen, Maren, Tomlinson, Darren C., Waterhouse, Mark P., Win, Stephanie J., Nettleship, Joanne E., Tiede, Christian, Foster, Richard J., Owens, Raymond J., Fishwick, Colin W. G., Harris, Sarah A., Goldman, Adrian, McPherson, Michael J., Morgan, Ann W.
Published in Proceedings of the National Academy of Sciences - PNAS (02.01.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (02.01.2018)
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Molecular mechanism of ligand recognition by membrane transport protein, Mhp1
Simmons, Katie J, Jackson, Scott M, Brueckner, Florian, Patching, Simon G, Beckstein, Oliver, Ivanova, Ekaterina, Geng, Tian, Weyand, Simone, Drew, David, Lanigan, Joseph, Sharples, David J, Sansom, Mark SP, Iwata, So, Fishwick, Colin WG, Johnson, A Peter, Cameron, Alexander D, Henderson, Peter JF
Published in The EMBO journal (18.08.2014)
Published in The EMBO journal (18.08.2014)
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Journal Article
Structure-Based Design, Synthesis, and Characterization of Inhibitors of Human and Plasmodium falciparum Dihydroorotate Dehydrogenases
Davies, Matthew, Heikkilä, Timo, McConkey, Glenn A, Fishwick, Colin W. G, Parsons, Mark R, Johnson, A. Peter
Published in Journal of medicinal chemistry (14.05.2009)
Published in Journal of medicinal chemistry (14.05.2009)
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Journal Article
Cyclic dinucleotides bind the C-linker of HCN4 to control channel cAMP responsiveness
Lolicato, Marco, Bucchi, Annalisa, Arrigoni, Cristina, Zucca, Stefano, Nardini, Marco, Schroeder, Indra, Simmons, Katie, Aquila, Marco, DiFrancesco, Dario, Bolognesi, Martino, Schwede, Frank, Kashin, Dmitry, Fishwick, Colin W G, Johnson, A Peter, Thiel, Gerhard, Moroni, Anna
Published in Nature chemical biology (01.06.2014)
Published in Nature chemical biology (01.06.2014)
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Factors Influencing the Specificity of Inhibitor Binding to the Human and Malaria Parasite Dihydroorotate Dehydrogenases
Bedingfield, Paul T. P, Cowen, Deborah, Acklam, Paul, Cunningham, Fraser, Parsons, Mark R, McConkey, Glenn A, Fishwick, Colin W. G, Johnson, A. Peter
Published in Journal of medicinal chemistry (28.06.2012)
Published in Journal of medicinal chemistry (28.06.2012)
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Journal Article
Furanyl-Rhodanines Are Unattractive Drug Candidates for Development as Inhibitors of Bacterial RNA Polymerase
MARINER, Katherine R, TROWBRIDGE, Rachel, AGARWAL, Anil K, MILLER, Keith, O'NEILL, Alex J, FISHWICK, Colin W. G, CHOPRA, Ian
Published in Antimicrobial Agents and Chemotherapy (01.10.2010)
Published in Antimicrobial Agents and Chemotherapy (01.10.2010)
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Molecular Genetic and Structural Modeling Studies of Staphylococcus aureus RNA Polymerase and the Fitness of Rifampin Resistance Genotypes in Relation to Clinical Prevalence
O'Neill, A J, Huovinen, T, Fishwick, C W G, Chopra, I
Published in Antimicrobial Agents and Chemotherapy (01.01.2006)
Published in Antimicrobial Agents and Chemotherapy (01.01.2006)
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Structure-based design of anti-infectives
Agarwal, Anil K, Fishwick, Colin W. G.
Published in Annals of the New York Academy of Sciences (01.12.2010)
Published in Annals of the New York Academy of Sciences (01.12.2010)
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Journal Article
Selective Phosphonylation of 5′-Adenosine Monophosphate (5′-AMP) via Pyrophosphite [PPi(III)]
Kaye, Karl, Bryant, David E., Marriott, Katie E. R., Ohara, Shohei, Fishwick, Colin W. G., Kee, Terence P.
Published in Origins of life and evolution of biospheres (01.11.2016)
Published in Origins of life and evolution of biospheres (01.11.2016)
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