Discovery of Clinical Candidate BMS-906024: A Potent Pan-Notch Inhibitor for the Treatment of Leukemia and Solid Tumors
Gavai, Ashvinikumar V, Quesnelle, Claude, Norris, Derek, Han, Wen-Ching, Gill, Patrice, Shan, Weifang, Balog, Aaron, Chen, Ke, Tebben, Andrew, Rampulla, Richard, Wu, Dauh-Rurng, Zhang, Yingru, Mathur, Arvind, White, Ronald, Rose, Anne, Wang, Haiqing, Yang, Zheng, Ranasinghe, Asoka, D’Arienzo, Celia, Guarino, Victor, Xiao, Lan, Su, Ching, Everlof, Gerry, Arora, Vinod, Shen, Ding Ren, Cvijic, Mary Ellen, Menard, Krista, Wen, Mei-Li, Meredith, Jere, Trainor, George, Lombardo, Louis J, Olson, Richard, Baran, Phil S, Hunt, John T, Vite, Gregory D, Fischer, Bruce S, Westhouse, Richard A, Lee, Francis Y
Published in ACS medicinal chemistry letters (14.05.2015)
Published in ACS medicinal chemistry letters (14.05.2015)
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Nivolumab Alone and With Ipilimumab in Previously Treated Metastatic Urothelial Carcinoma: CheckMate 032 Nivolumab 1 mg/kg Plus Ipilimumab 3 mg/kg Expansion Cohort Results
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Adjuvant Nivolumab versus Placebo in Muscle-Invasive Urothelial Carcinoma
Bajorin, Dean F, Witjes, J. Alfred, Gschwend, Jürgen E, Schenker, Michael, Valderrama, Begoña P, Tomita, Yoshihiko, Bamias, Aristotelis, Lebret, Thierry, Shariat, Shahrokh F, Park, Se Hoon, Ye, Dingwei, Agerbaek, Mads, Enting, Deborah, McDermott, Ray, Gajate, Pablo, Peer, Avivit, Milowsky, Matthew I, Nosov, Alexander, Neif Antonio, João, Tupikowski, Krzysztof, Toms, Laurence, Fischer, Bruce S, Qureshi, Anila, Collette, Sandra, Unsal-Kacmaz, Keziban, Broughton, Edward, Zardavas, Dimitrios, Koon, Henry B, Galsky, Matthew D
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Published in The New England journal of medicine (03.06.2021)
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Fibroblast Growth Factor Receptor 3 Alterations and Response to PD-1/PD-L1 Blockade in Patients with Metastatic Urothelial Cancer
Wang, Li, Gong, Yixuan, Saci, Abdel, Szabo, Peter M., Martini, Alberto, Necchi, Andrea, Siefker-Radtke, Arlene, Pal, Sumanta, Plimack, Elizabeth R., Sfakianos, John P., Bhardwaj, Nina, Horowitz, Amir, Farkas, Adam M., Mulholland, David, Fischer, Bruce S., Oh, William K., Sharma, Padmanee, Zhu, Jun, Galsky, Matthew D.
Published in European urology (01.11.2019)
Published in European urology (01.11.2019)
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Gamma Secretase Inhibition by BMS-906024 Enhances Efficacy of Paclitaxel in Lung Adenocarcinoma
Morgan, Katherine M, Fischer, Bruce S, Lee, Francis Y, Shah, Jamie J, Bertino, Joseph R, Rosenfeld, Jeffrey, Singh, Amartya, Khiabanian, Hossein, Pine, Sharon R
Published in Molecular cancer therapeutics (01.12.2017)
Published in Molecular cancer therapeutics (01.12.2017)
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A multi-arm phase I dose escalating study of an oral NOTCH inhibitor BMS-986115 in patients with advanced solid tumours
Aung, Kyaw L., El-Khoueiry, Anthony B., Gelmon, Karen, Tran, Ben, Bajaj, Gaurav, He, Bing, Chen, Tian, Zhu, Lili, Poojary, Sharath, Basak, Shashwati, Qi, Zhenhao, Spreafico, Anna, Fischer, Bruce S., Desai, Jayesh
Published in Investigational new drugs (01.12.2018)
Published in Investigational new drugs (01.12.2018)
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Treatment of muscle-invasive urothelial cancer with nivolumab (CheckMate 274 study): a plain language summary
Bajorin, Dean F, Witjes, J Alfred, Gschwend, Jürgen E, Schenker, Michael, Valderrama, Begoña P, Tomita, Yoshihiko, Bamias, Aristotelis, Lebret, Thierry, Shariat, Shahrokh F, Park, Se Hoon, Ye, Dingwei, Agerbaek, Mads, Enting, Deborah, McDermott, Ray, Gajate, Pablo, Peer, Avivit, Milowsky, Matthew I, Nosov, Alexander, Antonio, Jr, João Neif, Tupikowski, Krzysztof, Toms, Laurence, Fischer, Bruce S, Qureshi, Anila, Collette, Sandra, Unsal-Kacmaz, Keziban, Broughton, Edward, Zardavas, Dimitrios, Koon, Henry B, Galsky, Matthew D
Published in Future oncology (London, England) (01.02.2023)
Published in Future oncology (London, England) (01.02.2023)
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Metabolism, Excretion, and Pharmacokinetics of Oral Brivanib in Patients with Advanced or Metastatic Solid Tumors
MEKHAIL, Tarek, MASSON, Eric, FISCHER, Bruce S, JIACHANG GONG, LYER, Ramaswamy, JINPING GAN, PURSLEY, Janice, PATRICIA, Daniel, WILLIAMS, Daphne, GANAPATHI, Ram
Published in Drug metabolism and disposition (01.11.2010)
Published in Drug metabolism and disposition (01.11.2010)
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The effects of liver impairment on the pharmacokinetics of brivanib, a dual inhibitor of fibroblast growth factor receptor and vascular endothelial growth factor receptor tyrosine kinases
El-Khoueiry, Anthony, Posey, James A., Castillo Ferrando, Juan Ramón, Krishnamurthi, Smitha S., Syed, Shariq, Kollia, Georgia, Walters, Ian, Fischer, Bruce S., Masson, Eric
Published in Cancer chemotherapy and pharmacology (01.07.2013)
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JAK2 V617F patients with essential thrombocythemia present with clinical features of polycythemia vera
Zhang, Sujiang, Qiu, Hongxia, Fischer, Bruce S., Li, Weida, Duan, Limin, Sun, Xuemei, Xu, Wei, Li, Jianyong
Published in Leukemia & lymphoma (01.04.2008)
Published in Leukemia & lymphoma (01.04.2008)
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암 요법을 위한 복합 바이오마커
SANTUCCI PEREIRA DEL BUONO JULIA, KANDOUSSI ENZO YACOBI, GREENAWALT DANIELLE MARIE, WIND ROTOLO MEGAN M, ISHII YUKO, NELSON DAVID MARTIN, FISCHER BRUCE S
Year of Publication 24.05.2022
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Year of Publication 24.05.2022
Patent
Abstract 4834: Preclinical analysis of the Notch gamma secretase inhibitor BMS-906024 in combination with chemotherapy in the treatment of lung adenocarcinoma
Morgan, Katherine M., Lee, Francis, Michaud, Erin, Fischer, Bruce S., Pine, Sharon R.
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Adjuvant Nivolumab versus Placebo in Muscle-Invasive Urothelial Carcinoma
Published in The New England journal of medicine
(26.08.2021)
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Fibroblast growth factor receptor 3 (FGFR3), peroxisome proliferator-activated receptor gamma (PPARg), and outcomes with nivolumab (nivo) in metastatic urothelial cancer (UC)
Galsky, Matt D., Saci, Abdel, Szabo, Peter, Wang, Li, Zhu, Jun, Azrilevich, Alex, Fischer, Bruce S., Necchi, Andrea, Siefker-Radtke, Arlene O., Sharma, Padmanee
Published in Journal of clinical oncology (20.02.2018)
Published in Journal of clinical oncology (20.02.2018)
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A phase II, randomized study of nivolumab (NIVO), NIVO plus linrodostat mesylate, or NIVO plus intravesical bacillus Calmette-Guerin (BCG) in BCG-unresponsive, high-risk, nonmuscle invasive bladder cancer (NMIBC): CheckMate 9UT
Hahn, Noah M., Chang, Sam, Meng, Maxwell, Shore, Neal D., Konety, Badrinath R., Steinberg, Gary D., Gschwend, Juergen, Nishiyama, Hiroyuki, Palou, Joan, Taylor, John A, Lambert, Alexandre, Zhu, Li, Maeda, Toshiki, Raybold, Bradley, Fischer, Bruce S., Jeyamohan, Chandrika, Zardavas, Dimitrios, Witjes, Fred
Published in Journal of clinical oncology (20.05.2020)
Published in Journal of clinical oncology (20.05.2020)
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Abstract 2535: Synergistic anti-tumor activity of the Notch gamma secretase inhibitor BMS-906024 and paclitaxel in the treatment of lung adenocarcinoma
Morgan, Katherine M., Lee, Francis, Michaud, Erin, Bertino, Joseph R., Fischer, Bruce S., Pine, Sharon R.
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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A phase I study of AL101, a pan-NOTCH inhibitor, in patients (pts) with locally advanced or metastatic solid tumors
El-Khoueiry, Anthony B., Desai, Jayesh, Iyer, Swaminathan Padmanabhan, Gadgeel, Shirish M., Ramalingam, Suresh S., Horn, Leora, LoRusso, Patricia, Bajaj, Gaurav, Kollia, Georgia, Qi, Zhenhao, Basak, Shashwati, Fischer, Bruce S., Davis, Matti, Bedard, Philippe L.
Published in Journal of clinical oncology (20.05.2018)
Published in Journal of clinical oncology (20.05.2018)
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