Whole-Cell Screen of Fragment Library Identifies Gut Microbiota Metabolite Indole Propionic Acid as Antitubercular
Negatu, Dereje A, Liu, Joe J J, Zimmerman, Matthew, Kaya, Firat, Dartois, Véronique, Aldrich, Courtney C, Gengenbacher, Martin, Dick, Thomas
Published in Antimicrobial agents and chemotherapy (01.03.2018)
Published in Antimicrobial agents and chemotherapy (01.03.2018)
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Journal Article
Matrix metalloproteinase inhibitors enhance the efficacy of frontline drugs against Mycobacterium tuberculosis
Xu, Yitian, Wang, Lihua, Zimmerman, Matthew D, Chen, Kai-Yuan, Huang, Lu, Fu, Dah-Jiun, Kaya, Firat, Rakhilin, Nikolai, Nazarova, Evgeniya V, Bu, Pengcheng, Dartois, Veronique, Russell, David G, Shen, Xiling
Published in PLoS pathogens (01.04.2018)
Published in PLoS pathogens (01.04.2018)
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Journal Article
Pyrazinamide Resistance Is Caused by Two Distinct Mechanisms: Prevention of Coenzyme A Depletion and Loss of Virulence Factor Synthesis
Gopal, Pooja, Yee, Michelle, Sarathy, Jickky, Low, Jian Liang, Sarathy, Jansy P, Kaya, Firat, Dartois, Véronique, Gengenbacher, Martin, Dick, Thomas
Published in ACS infectious diseases (09.09.2016)
Published in ACS infectious diseases (09.09.2016)
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Journal Article
A Multimodal Desorption Electrospray Ionisation Workflow Enabling Visualisation of Lipids and Biologically Relevant Elements in a Single Tissue Section
Costa, Catia, De Jesus, Janella, Nikula, Chelsea, Murta, Teresa, Grime, Geoffrey W, Palitsin, Vladimir, Dartois, Véronique, Firat, Kaya, Webb, Roger, Bunch, Josephine, Bailey, Melanie J
Published in Metabolites (01.02.2023)
Published in Metabolites (01.02.2023)
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Journal Article
Obesity and Loss of Kidney Function: Two Complications to Face for Older Living Kidney Donors
Firat Kaya, Demet, Sayin, Burak, Saglam, Hatice, Gurlek Demirci, Bahar, Colak, Turan
Published in Experimental and clinical transplantation : official journal of the Middle East Society for Organ Transplantation (01.02.2017)
Published in Experimental and clinical transplantation : official journal of the Middle East Society for Organ Transplantation (01.02.2017)
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Journal Article
The association between sterilizing activity and drug distribution into tuberculosis lesions
Prideaux, Brendan, Via, Laura E, Zimmerman, Matthew D, Eum, Seokyong, Sarathy, Jansy, O'Brien, Paul, Chen, Chao, Kaya, Firat, Weiner, Danielle M, Chen, Pei-Yu, Song, Taeksun, Lee, Myungsun, Shim, Tae Sun, Cho, Jeong Su, Kim, Wooshik, Cho, Sang Nae, Olivier, Kenneth N, Barry, Clifton E, Dartois, Véronique
Published in Nature medicine (01.10.2015)
Published in Nature medicine (01.10.2015)
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Journal Article
Selective Inactivity of Pyrazinamide against Tuberculosis in C3HeB/FeJ Mice Is Best Explained by Neutral pH of Caseum
Lanoix, Jean-Philippe, Ioerger, Thomas, Ormond, Aimee, Kaya, Firat, Sacchettini, James, Dartois, Véronique, Nuermberger, Eric
Published in Antimicrobial agents and chemotherapy (01.02.2016)
Published in Antimicrobial agents and chemotherapy (01.02.2016)
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Journal Article
Rifabutin central nervous system concentrations in a rabbit model of tuberculous meningitis
Wasserman, Sean, Antilus-Sainte, Rosleine, Abdelgawad, Noha, Odjourian, Narineh M, Cristaldo, Melissa, Dougher, Maureen, Kaya, Firat, Zimmerman, Matthew, Denti, Paolo, Gengenbacher, Martin
Published in Antimicrobial agents and chemotherapy (07.08.2024)
Published in Antimicrobial agents and chemotherapy (07.08.2024)
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Journal Article
Ethambutol Partitioning in Tuberculous Pulmonary Lesions Explains Its Clinical Efficacy
Zimmerman, Matthew, Lestner, Jodi, Prideaux, Brendan, O'Brien, Paul, Dias-Freedman, Isabela, Chen, Chao, Dietzold, Jillian, Daudelin, Isaac, Kaya, Firat, Blanc, Landry, Chen, Pei-Yu, Park, Steven, Salgame, Padmini, Sarathy, Jansy, Dartois, Véronique
Published in Antimicrobial agents and chemotherapy (01.09.2017)
Published in Antimicrobial agents and chemotherapy (01.09.2017)
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Journal Article
A preclinical model of TB meningitis to determine drug penetration and activity at the sites of disease
Lanni, Faye, Antilus Sainte, Rosleine, Hansen, Jr, Mark, Parigi, Paul, Kaya, Firat, LoMauro, Katherine, Siow, Bernard, Wilkinson, Robert J, Wasserman, Sean, Podell, Brendan K, Gengenbacher, Martin, Dartois, Véronique
Published in Antimicrobial agents and chemotherapy (14.12.2023)
Published in Antimicrobial agents and chemotherapy (14.12.2023)
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Journal Article
Spatial quantitation of antibiotics in bone tissue compartments by laser-capture microdissection coupled with UHPLC-tandem mass spectrometry
Kaya, Firat, Zimmerman, Matthew D., Antilus-Sainte, Rosleine, Gengenbacher, Martin, Carter, Claire L., Dartois, Véronique
Published in Analytical and bioanalytical chemistry (01.09.2022)
Published in Analytical and bioanalytical chemistry (01.09.2022)
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Journal Article
Tissue Distribution of Doxycycline in Animal Models of Tuberculosis
Gengenbacher, Martin, Zimmerman, Matthew D, Sarathy, Jansy P, Kaya, Firat, Wang, Han, Mina, Marizel, Carter, Claire, Hossen, Md Amir, Su, Hongwei, Trujillo, Carolina, Ehrt, Sabine, Schnappinger, Dirk, Dartois, Véronique
Published in Antimicrobial agents and chemotherapy (21.04.2020)
Published in Antimicrobial agents and chemotherapy (21.04.2020)
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Journal Article
Fluoroquinolone Efficacy against Tuberculosis Is Driven by Penetration into Lesions and Activity against Resident Bacterial Populations
Sarathy, Jansy, Blanc, Landry, Alvarez-Cabrera, Nadine, O'Brien, Paul, Dias-Freedman, Isabela, Mina, Marizel, Zimmerman, Matthew, Kaya, Firat, Ho Liang, Hsin-Pin, Prideaux, Brendan, Dietzold, Jillian, Salgame, Padmini, Savic, Radojka M, Linderman, Jennifer, Kirschner, Denise, Pienaar, Elsje, Dartois, Véronique
Published in Antimicrobial agents and chemotherapy (01.05.2019)
Published in Antimicrobial agents and chemotherapy (01.05.2019)
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Journal Article
On-Slide Heat Sterilization Enables Mass Spectrometry Imaging of Tissue Infected with High-Threat Pathogens Outside of Biocontainment: A Study Directed at Mycobacterium tuberculosis
Wang, Ning, Sarathy, Jansy P, Zimmerman, Matthew, Kaya, Firat, Wang, Han, Dartois, Véronique, Carter, Claire L
Published in Journal of the American Society for Mass Spectrometry (03.11.2021)
Published in Journal of the American Society for Mass Spectrometry (03.11.2021)
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Journal Article
Colocation of Lipids, Drugs, and Metal Biomarkers Using Spatially Resolved Lipidomics with Elemental Mapping
Lewis, Holly-May, Costa, Catia, Dartois, Véronique, Kaya, Firat, Chambers, Mark, de Jesus, Janella, Palitsin, Vladimir, Webb, Roger, Bailey, Melanie J.
Published in Analytical chemistry (Washington) (30.08.2022)
Published in Analytical chemistry (Washington) (30.08.2022)
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Journal Article
Comparative Analysis of Pharmacodynamics in the C3HeB/FeJ Mouse Tuberculosis Model for DprE1 Inhibitors TBA-7371, PBTZ169, and OPC-167832
Robertson, Gregory T, Ramey, Michelle E, Massoudi, Lisa M, Carter, Claire L, Zimmerman, Matt, Kaya, Firat, Graham, Barbara G, Gruppo, Veronica, Hastings, Courtney, Woolhiser, Lisa K, Scott, Dashick W L, Asay, Bryce C, Eshun-Wilson, Franceen, Maidj, Ekaterina, Podell, Brendan K, Vásquez, Joshua J, Lyons, Mike A, Dartois, Véronique, Lenaerts, Anne J
Published in Antimicrobial agents and chemotherapy (18.10.2021)
Published in Antimicrobial agents and chemotherapy (18.10.2021)
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Journal Article
Lesion Penetration and Activity Limit the Utility of Second-Line Injectable Agents in Pulmonary Tuberculosis
Ernest, Jacqueline P, Sarathy, Jansy, Wang, Ning, Kaya, Firat, Zimmerman, Matthew D, Strydom, Natasha, Wang, Han, Xie, Min, Gengenbacher, Martin, Via, Laura E, Barry, 3rd, Clifton E, Carter, Claire L, Savic, Radojka M, Dartois, Véronique
Published in Antimicrobial agents and chemotherapy (17.09.2021)
Published in Antimicrobial agents and chemotherapy (17.09.2021)
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Journal Article
Evolutionary dynamics in gut-colonizing Candida glabrata during caspofungin therapy: Emergence of clinically important mutations in sphingolipid biosynthesis
Hassoun, Yasmine, Aptekmann, Ariel A, Keniya, Mikhail V, Gomez, Rosa Y, Alayo, Nicole, Novi, Giovanna, Quinteros, Christopher, Kaya, Firat, Zimmerman, Matthew, Caceres, Diego H, Chow, Nancy A, Perlin, David S, Shor, Erika
Published in PLoS pathogens (09.09.2024)
Published in PLoS pathogens (09.09.2024)
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Journal Article
A Rabbit Model to Study Antibiotic Penetration at the Site of Infection for Nontuberculous Mycobacterial Lung Disease: Macrolide Case Study
Kaya, Firat, Ernest, Jacqueline P, LoMauro, Katherine, Gengenbacher, Martin, Madani, Abdeldjalil, Aragaw, Wassihun Wedajo, Zimmerman, Matthew D, Sarathy, Jansy P, Alvarez, Nadine, Daudelin, Isaac, Wang, Han, Lanni, Faye, Weiner, Danielle M, Via, Laura E, Barry, 3rd, Clifton E, Olivier, Kenneth N, Dick, Thomas, Podell, Brendan K, Savic, Radojka M, Dartois, Véronique
Published in Antimicrobial agents and chemotherapy (15.03.2022)
Published in Antimicrobial agents and chemotherapy (15.03.2022)
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Journal Article
Pharmacokinetics and Target Attainment of SQ109 in Plasma and Human-Like Tuberculosis Lesions in Rabbits
Egbelowo, Oluwaseun, Sarathy, Jansy P, Gausi, Kamunkhwala, Zimmerman, Matthew D, Wang, Han, Wijnant, Gert-Jan, Kaya, Firat, Gengenbacher, Martin, Van, Nhi, Degefu, Yonatan, Nacy, Carol, Aldridge, Bree B, Carter, Claire L, Denti, Paolo, Dartois, Véronique
Published in Antimicrobial agents and chemotherapy (17.08.2021)
Published in Antimicrobial agents and chemotherapy (17.08.2021)
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Journal Article