Synaptic Therapy in Alzheimer’s Disease: A CREB-centric Approach
Teich, Andrew F., Nicholls, Russell E., Puzzo, Daniela, Fiorito, Jole, Purgatorio, Rosa, Fa’, Mauro, Arancio, Ottavio
Published in Neurotherapeutics (2015)
Published in Neurotherapeutics (2015)
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Journal Article
Synaptic and memory dysfunction induced by tau oligomers is rescued by up-regulation of the nitric oxide cascade
Acquarone, Erica, Argyrousi, Elentina K, van den Berg, Manon, Gulisano, Walter, Fà, Mauro, Staniszewski, Agnieszka, Calcagno, Elisa, Zuccarello, Elisa, D'Adamio, Luciano, Deng, Shi-Xian, Puzzo, Daniela, Arancio, Ottavio, Fiorito, Jole
Published in Molecular neurodegeneration (27.06.2019)
Published in Molecular neurodegeneration (27.06.2019)
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Journal Article
Antiangiogenic Effect of (±)-Haloperidol Metabolite II Valproate Ester [(±)-MRJF22] in Human Microvascular Retinal Endothelial Cells
Olivieri, Melania, Amata, Emanuele, Vinciguerra, Shila, Fiorito, Jole, Giurdanella, Giovanni, Drago, Filippo, Caporarello, Nunzia, Prezzavento, Orazio, Arena, Emanuela, Salerno, Loredana, Rescifina, Antonio, Lupo, Gabriella, Anfuso, Carmelina Daniela, Marrazzo, Agostino
Published in Journal of medicinal chemistry (10.11.2016)
Published in Journal of medicinal chemistry (10.11.2016)
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Journal Article
Correction: Synaptic and memory dysfunction induced by tau oligomers is rescued by up-regulation of the nitric oxide cascade
Acquarone, Erica, Argyrousi, Elentina K, van den Berg, Manon, Gulisano, Walter, Fà, Mauro, Staniszewski, Agnieszka, Calcagno, Elisa, Zuccarello, Elisa, D'Adamio, Luciano, Deng, Shi-Xian, Puzzo, Daniela, Arancio, Ottavio, Fiorito, Jole
Published in Molecular neurodegeneration (29.04.2024)
Published in Molecular neurodegeneration (29.04.2024)
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Journal Article
Development of novel phosphodiesterase 5 inhibitors for the therapy of Alzheimer’s disease
Zuccarello, Elisa, Acquarone, Erica, Calcagno, Elisa, Argyrousi, Elentina K., Deng, Shi-Xian, Landry, Donald W., Arancio, Ottavio, Fiorito, Jole
Published in Biochemical pharmacology (01.06.2020)
Published in Biochemical pharmacology (01.06.2020)
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Journal Article
Identification of a Novel 1,2,3,4-Tetrahydrobenzo[b][1,6]naphthyridine Analogue as a Potent Phosphodiesterase 5 Inhibitor with Improved Aqueous Solubility for the Treatment of Alzheimer’s Disease
Fiorito, Jole, Vendome, Jeremie, Saeed, Faisal, Staniszewski, Agnieszka, Zhang, Hong, Yan, Shijun, Deng, Shi-Xian, Arancio, Ottavio, Landry, Donald W
Published in Journal of medicinal chemistry (09.11.2017)
Published in Journal of medicinal chemistry (09.11.2017)
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Journal Article
Optimizing metabolic stability of phosphodiesterase 5 inhibitors: Discovery of a potent N-(pyridin-3-ylmethyl)quinoline derivative targeting synaptic plasticity
Zuccarello, Elisa, Zhang, Hong, Acquarone, Erica, Pham, Dang, Staniszewski, Anna, Deng, Shi-Xian, Landry, Donald W., Arancio, Ottavio, Fiorito, Jole
Published in Bioorganic & medicinal chemistry letters (15.08.2023)
Published in Bioorganic & medicinal chemistry letters (15.08.2023)
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Journal Article
Histone Acetyltransferase (HAT) Activator, YF2, Modulates the p53:BCL6 Axis and Antigen Presentation in Diffuse Large B-Cell Lymphomas
Estrella, Brian, Liu, Yuxuan, Ricker, Edd C, Pazos, Manuel A, Fiorito, Jole, Zuccarello, Elisa, Calcagno, Elisa, Honig, Barry, Arancio, Ottavio, Amengual, Jennifer E.
Published in Blood (23.11.2021)
Published in Blood (23.11.2021)
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Journal Article
PDE5 inhibitors against synaptic and cognitive impairment in Alzheimer’s disease and related dementia
Arancio, Ottavio, Zuccarello, Elisa, Fiorito, Jole, Acquarone, Erica, Argyrousi, Elentina, Staniszewski, Agnieszka, Calcagno, Elisa, Puzzo, Daniela, Deng, Shi‐Xian, Landry, Donald
Published in Alzheimer's & dementia (01.12.2022)
Published in Alzheimer's & dementia (01.12.2022)
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Journal Article
Synthesis of quinoline derivatives: Discovery of a potent and selective phosphodiesterase 5 inhibitor for the treatment of Alzheimer's disease
Fiorito, Jole, Saeed, Faisal, Zhang, Hong, Staniszewski, Agnieszka, Feng, Yan, Francis, Yitshak I., Rao, Sudha, Thakkar, Devarshi M., Deng, Shi-Xian, Landry, Donald W., Arancio, Ottavio
Published in European journal of medicinal chemistry (01.02.2013)
Published in European journal of medicinal chemistry (01.02.2013)
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Journal Article
Strategy for Overcoming Crebbp and EP300 Mutations in Lymphoma: Development of First-in-Class HAT Activators
Liu, Yuxuan, Fiorito, Jole, Gonzalez, Yulissa, Estrella, Brian, Calcagno, Elisa, Zuccarello, Elisa, Hwang, Howook, Honig, Barry, Deng, Shixian, Landry, Donald, O'Connor, Owen A., Arancio, Ottavio, Amengual, Jennifer E
Published in Blood (13.11.2019)
Published in Blood (13.11.2019)
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Journal Article
Haloperidol metabolite II prodrug: Asymmetric synthesis and biological evaluation on rat C6 glioma cells
Sozio, Piera, Fiorito, Jole, Di Giacomo, Viviana, Di Stefano, Antonio, Marinelli, Lisa, Cacciatore, Ivana, Cataldi, Amelia, Pacella, Stephanie, Turkez, Hasan, Parenti, Carmela, Rescifina, Antonio, Marrazzo, Agostino
Published in European journal of medicinal chemistry (27.01.2015)
Published in European journal of medicinal chemistry (27.01.2015)
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Journal Article
Development of First-in-Class Histone Acetyltransferase (HAT) Activators for Precision Targeting of Epigenetic Derangements in Lymphoma
Liu, Yuxuan, Fiorito, Jole, Gonzalez, Yulissa, Zuccarello, Elisa, Calcagno, Elisa, Mazzeo, Adolfo, Abshiru, Nebiyu Ali, Camarillo, Jeannie, Kelleher, Neil L, Qiao, Changhong, Nandakumar, Renu, Serge, Cremers, Deng, Shixian, Landry, Donald, O'Connor, Owen A., Arancio, Ottavio, Amengual, Jennifer E
Published in Blood (29.11.2018)
Published in Blood (29.11.2018)
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Journal Article
Antiproliferative activity of phenylbutyrate ester of haloperidol metabolite II [(±)-MRJF4] in prostate cancer cells
Marrazzo, Agostino, Fiorito, Jole, Zappalà, Laura, Prezzavento, Orazio, Ronsisvalle, Simone, Pasquinucci, Lorella, Scoto, Giovanna M., Bernardini, Renato, Ronsisvalle, Giuseppe
Published in European journal of medicinal chemistry (01.01.2011)
Published in European journal of medicinal chemistry (01.01.2011)
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히스톤 아세틸트랜스퍼라제 활성화제 및 이의 조성물 및 용도
PURGATORIO ROSA, SCOTTO LUIGI, ARANCIO OTTAVIO, DENG SHI XIAN, AMENGUAL JENNIFER EFFIE, LANDRY DONALD W, O'CONNOR OWEN ANTHONY, FIORITO JOLE
Year of Publication 22.03.2019
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Year of Publication 22.03.2019
Patent
Phosphodiesterase inhibitors and uses thereof
Fiorito, Jole, Arancio, Ottavio, Wasmuth, Andrew, Landry, Donald W, Deng, Shixian
Year of Publication 26.12.2023
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Year of Publication 26.12.2023
Patent
NOVEL PHOSPHODIESTERASE INHIBITORS AND USES THEREOF
DENG, Shixian, FIORITO, Jole, WASMUTH, Andrew, LANDRY, Donald W, ARANCIO, Ottavio
Year of Publication 06.05.2021
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Year of Publication 06.05.2021
Patent