Thalidomide promotes degradation of SALL4, a transcription factor implicated in Duane Radial Ray syndrome
Donovan, Katherine A, An, Jian, Nowak, Radosław P, Yuan, Jingting C, Fink, Emma C, Berry, Bethany C, Ebert, Benjamin L, Fischer, Eric S
Published in eLife (01.08.2018)
Published in eLife (01.08.2018)
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Patterns of substrate affinity, competition, and degradation kinetics underlie biological activity of thalidomide analogs
Sperling, Adam S., Burgess, Michael, Keshishian, Hasmik, Gasser, Jessica A., Bhatt, Shruti, Jan, Max, Słabicki, Mikołaj, Sellar, Rob S., Fink, Emma C., Miller, Peter G., Liddicoat, Brian J., Sievers, Quinlan L., Sharma, Rohan, Adams, Dylan N., Olesinski, Elyse A., Fulciniti, Mariateresa, Udeshi, Namrata D., Kuhn, Eric, Letai, Anthony, Munshi, Nikhil C., Carr, Steven A., Ebert, Benjamin L.
Published in Blood (11.07.2019)
Published in Blood (11.07.2019)
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Androgen receptor monomers and dimers regulate opposing biological processes in prostate cancer cells
Safi, Rachid, Wardell, Suzanne E, Watkinson, Paige, Qin, Xiaodi, Lee, Marissa, Park, Sunghee, Krebs, Taylor, Dolan, Emma L, Blattler, Adam, Tsuji, Toshiya, Nayak, Surendra, Khater, Marwa, Fontanillo, Celia, Newlin, Madeline A, Kirkland, Megan L, Xie, Yingtian, Long, Henry, Fink, Emma C, Fanning, Sean W, Runyon, Scott, Brown, Myles, Xu, Shuichan, Owzar, Kouros, Norris, John D, McDonnell, Donald P
Published in Nature communications (03.09.2024)
Published in Nature communications (03.09.2024)
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Csnk1a1 inhibition has p53-dependent therapeutic efficacy in acute myeloid leukemia
Järås, Marcus, Miller, Peter G, Chu, Lisa P, Puram, Rishi V, Fink, Emma C, Schneider, Rebekka K, Al-Shahrour, Fatima, Peña, Pablo, Breyfogle, L Jordan, Hartwell, Kimberly A, McConkey, Marie E, Cowley, Glenn S, Root, David E, Kharas, Michael G, Mullally, Ann, Ebert, Benjamin L
Published in The Journal of experimental medicine (07.04.2014)
Published in The Journal of experimental medicine (07.04.2014)
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The CDK inhibitor CR8 acts as a molecular glue degrader that depletes cyclin K
Słabicki, Mikołaj, Kozicka, Zuzanna, Petzold, Georg, Li, Yen-Der, Manojkumar, Manisha, Bunker, Richard D, Donovan, Katherine A, Sievers, Quinlan L, Koeppel, Jonas, Suchyta, Dakota, Sperling, Adam S, Fink, Emma C, Gasser, Jessica A, Wang, Li R, Corsello, Steven M, Sellar, Rob S, Jan, Max, Gillingham, Dennis, Scholl, Claudia, Fröhling, Stefan, Golub, Todd R, Fischer, Eric S, Thomä, Nicolas H, Ebert, Benjamin L
Published in Nature (London) (10.09.2020)
Published in Nature (London) (10.09.2020)
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Lenalidomide induces ubiquitination and degradation of CK1α in del(5q) MDS
Krönke, Jan, Fink, Emma C, Hollenbach, Paul W, MacBeth, Kyle J, Hurst, Slater N, Udeshi, Namrata D, Chamberlain, Philip P, Mani, D R, Man, Hon Wah, Gandhi, Anita K, Svinkina, Tanya, Schneider, Rebekka K, McConkey, Marie, Järås, Marcus, Griffiths, Elizabeth, Wetzler, Meir, Bullinger, Lars, Cathers, Brian E, Carr, Steven A, Chopra, Rajesh, Ebert, Benjamin L
Published in Nature (London) (09.07.2015)
Published in Nature (London) (09.07.2015)
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Journal Article
Notch signaling without the APH-2/nicastrin subunit of gamma secretase in Caenorhabditis elegans germline stem cells
Brinkley, David M, Smith, Karen C, Fink, Emma C, Kwen, Woohyun, Yoo, Nina H, West, Zachary, Sullivan, Nora L, Farthing, Alex S, Hale, Valerie A, Goutte, Caroline
Published in Genetics (Austin) (08.07.2024)
Published in Genetics (Austin) (08.07.2024)
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Sequence similarity network analysis of drug- and dye-modifying azoreductase enzymes found in the human gut microbiome
Long, Audrey R., Mortara, Emma L., Mendoza, Brisa N., Fink, Emma C., Sacco, Francis X., Ciesla, Matthew J., Stack, Tyler M.M.
Published in Archives of biochemistry and biophysics (01.07.2024)
Published in Archives of biochemistry and biophysics (01.07.2024)
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Development of NR0B2 as a therapeutic target for the re-education of tumor associated myeloid cells
Vidana Gamage, Hashni Epa, Albright, Samuel T., Smith, Amanda J., Farmer, Rachel, Shahoei, Sayyed Hamed, Wang, Yu, Fink, Emma C., Jacquin, Elise, Weisser, Erin, Bautista, Rafael O., Henn, Madeline A., Schane, Claire P., Nelczyk, Adam T., Ma, Liqian, Das Gupta, Anasuya, Bendre, Shruti V., Nguyen, Tiffany, Tiwari, Srishti, Krawczynska, Natalia, He, Sisi, Tjoanda, Evelyn, Chen, Hong, Sverdlov, Maria, Gann, Peter H., Boidot, Romain, Vegran, Frederique, Fanning, Sean W., Apetoh, Lionel, Hergenrother, Paul J., Nelson, Erik R.
Published in Cancer letters (10.08.2024)
Published in Cancer letters (10.08.2024)
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NR0B2 re-educates myeloid immune cells to reduce regulatory T cell expansion and progression of breast and other solid tumors
Vidana Gamage, Hashni Epa, Shahoei, Sayyed Hamed, Wang, Yu, Jacquin, Elise, Weisser, Erin, Bautista, Rafael O., Henn, Madeline A., Schane, Claire P., Nelczyk, Adam T., Ma, Liqian, Das Gupta, Anasuya, Bendre, Shruti V., Nguyen, Tiffany, Tiwari, Srishti, Tjoanda, Evelyn, Krawczynska, Natalia, He, Sisi, Albright, Samuel T., Farmer, Rachel, Smith, Amanda J., Fink, Emma C., Chen, Hong, Sverdlov, Maria, Gann, Peter H., Boidot, Romain, Vegran, Frederique, Fanning, Sean W., Hergenrother, Paul J., Apetoh, Lionel, Nelson, Erik R.
Published in Cancer letters (10.08.2024)
Published in Cancer letters (10.08.2024)
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Crbn I391V is sufficient to confer in vivo sensitivity to thalidomide and its derivatives in mice
Fink, Emma C, McConkey, Marie, Adams, Dylan N, Haldar, Saurav D, Kennedy, James A, Guirguis, Andrew A, Udeshi, Namrata D, Mani, D R, Chen, Michelle, Liddicoat, Brian, Svinkina, Tanya, Nguyen, Andrew T, Carr, Steven A, Ebert, Benjamin L
Published in Blood (04.10.2018)
Published in Blood (04.10.2018)
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Journal Article
CrbnI391V is sufficient to confer in vivo sensitivity to thalidomide and its derivatives in mice
Fink, Emma C., McConkey, Marie, Adams, Dylan N., Haldar, Saurav D., Kennedy, James A., Guirguis, Andrew A., Udeshi, Namrata D., Mani, D.R., Chen, Michelle, Liddicoat, Brian, Svinkina, Tanya, Nguyen, Andrew T., Carr, Steven A., Ebert, Benjamin L.
Published in Blood (04.10.2018)
Published in Blood (04.10.2018)
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Journal Article
Degradation of GSPT1 causes TP53-independent cell death in leukemia while sparing normal hematopoietic stem cells
Sellar, Rob S, Sperling, Adam S, Słabicki, Mikołaj, Gasser, Jessica A, McConkey, Marie E, Donovan, Katherine A, Mageed, Nada, Adams, Dylan N, Zou, Charles, Miller, Peter G, Dutta, Ravi K, Boettcher, Steffen, Lin, Amy E, Sandoval, Brittany, Quevedo Barrios, Vanessa A, Kovalcik, Veronica, Koeppel, Jonas, Henderson, Elizabeth K, Fink, Emma C, Yang, Lu, Chan, Anthony, Pokharel, Sheela Pangeni, Bergstrom, Erik J, Burt, Rajan, Udeshi, Namrata D, Carr, Steven A, Fischer, Eric S, Chen, Chun-Wei, Ebert, Benjamin L
Published in The Journal of clinical investigation (15.08.2022)
Published in The Journal of clinical investigation (15.08.2022)
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Journal Article
Notch signaling without the APH-2/Nicastrin subunit of Gamma Secretase in C. elegans germline stem cells
Brinkley, David M, Smith, Karen C, Fink, Emma C, Kwen, Woohyun, Yoo, Nina H, West, Zachary, Sullivan, Nora L, Farthing, Alex S, Hale, Valerie A, Goutte, Caroline
Published in Genetics (Austin) (08.05.2024)
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Published in Genetics (Austin) (08.05.2024)
Journal Article
Lenalidomide Induces Ubiquitination and Degradation of CSNK1A1 in MDS with Del(5q)
Fink, Emma C., Krönke, Jan, Hurst, Slater N., Udeshi, Namrata D., Svinkina, Tanya, Schneider, Rebekka K., McConkey, Marie E., Järås, Marcus, Bullinger, Lars, Carr, Steven A., Ebert, Benjamin L.
Published in Blood (06.12.2014)
Published in Blood (06.12.2014)
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Journal Article
Lenalidomide induces ubiquitination and degradation of CK1[alpha] in del(5q) MDS
Krönke, Jan, Fink, Emma C, Hollenbach, Paul W, MacBeth, Kyle J, Hurst, Slater N, Udeshi, Namrata D, Chamberlain, Philip P, Mani, D R, Man, Hon Wah, Gandhi, Anita K, Svinkina, Tanya, Schneider, Rebekka K, McConkey, Marie, Järås, Marcus, Griffiths, Elizabeth, Wetzler, Meir, Bullinger, Lars, Cathers, Brian E, Carr, Steven A, Chopra, Rajesh, Ebert, Benjamin L
Published in Nature (London) (09.07.2015)
Published in Nature (London) (09.07.2015)
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