Improving Nonspecific Binding and Solubility: Bicycloalkyl Groups and Cubanes as para‐Phenyl Bioisosteres
Auberson, Yves P., Brocklehurst, Cara, Furegati, Markus, Fessard, Thomas C., Koch, Guido, Decker, Andrea, La Vecchia, Luigi, Briard, Emmanuelle
Published in ChemMedChem (20.04.2017)
Published in ChemMedChem (20.04.2017)
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[2]-Ladderanes as isosteres for meta-substituted aromatic rings and rigidified cyclohexanes
Epplin, Rachel C., Paul, Shashwati, Herter, Loïc, Salome, Christophe, Hancock, Erin N., Larrow, Jay F., Baum, Erich W., Dunstan, David R., Ginsburg-Moraff, Carol, Fessard, Thomas C., Brown, M. Kevin
Published in Nature communications (13.10.2022)
Published in Nature communications (13.10.2022)
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Strain-Release [2π + 2σ] Cycloadditions for the Synthesis of Bicyclo[2.1.1]hexanes Initiated by Energy Transfer
Guo, Renyu, Chang, Yu-Che, Herter, Loic, Salome, Christophe, Braley, Sarah E., Fessard, Thomas C., Brown, M. Kevin
Published in Journal of the American Chemical Society (11.05.2022)
Published in Journal of the American Chemical Society (11.05.2022)
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Oxetanyl Peptides: Novel Peptidomimetic Modules for Medicinal Chemistry
McLaughlin, Martin, Yazaki, Ryo, Fessard, Thomas C, Carreira, Erick M
Published in Organic letters (15.08.2014)
Published in Organic letters (15.08.2014)
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Nickel‐Photoredox‐Catalyzed Synthesis of sp2−sp3 Fragments and the Impact of Bicycloalkane Isosteric Replacement on Their Physical‐Chemical Properties
Lefebvre, Quentin, Bocu, Mina, Giorgiutti, Christophe, Fessard, Thomas C.
Published in Helvetica chimica acta (01.04.2023)
Published in Helvetica chimica acta (01.04.2023)
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Diversification of Simple Arenes into Complex (Amino)cyclitols
Angelini, Elisa, Martinelli, Matteo, Roà, Eugenio, Ungarean, Chad N., Salome, Christophe, Lefebvre, Quentin, Bournez, Colin, Fessard, Thomas C., Sarlah, David
Published in Chemistry : a European journal (26.01.2024)
Published in Chemistry : a European journal (26.01.2024)
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Synthesis of Borylated Carbocycles by [2 + 2]-Cycloadditions and Photo-Ene Reactions
Posz, Jarett M., Sharma, Neetu, Royalty, Paige A., Liu, Yanyao, Salome, Christophe, Fessard, Thomas C., Brown, M. Kevin
Published in Journal of the American Chemical Society (10.04.2024)
Published in Journal of the American Chemical Society (10.04.2024)
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Reactivity and Selectivity of Azaspirocycles in Radical C–H Functionalization
Ungarean, Chad N., Larin, Egor M., Egger, Dominic T., Ziegler, Philipp, Lefebvre, Quentin, Fessard, Thomas C., Morandi, Bill
Published in Organic letters (12.04.2024)
Published in Organic letters (12.04.2024)
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3,3-Dinitratooxetane - an important leap towards energetic oxygen-rich monomers and polymers
Born, Max, Fessard, Thomas C, Göttemann, Lucas, Klapötke, Thomas M, Stierstorfer, Jörg, Voggenreiter, Michael
Published in Chemical communications (Cambridge, England) (16.03.2021)
Published in Chemical communications (Cambridge, England) (16.03.2021)
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Nickel-Photoredox-Catalyzed Synthesis of sp(2)-sp(3) Fragments and the Impact of Bicycloalkane Isosteric Replacement on Their Physical-Chemical Properties
Lefebvre, Quentin, Bocu, Mina, Giorgiutti, Christophe, Fessard, Thomas C.
Published in Helvetica chimica acta (01.04.2023)
Published in Helvetica chimica acta (01.04.2023)
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