Investigational drugs in early phase clinical trials targeting thermotransient receptor potential (thermoTRP) channels
Fernández-Carvajal, Asia, González-Muñiz, Rosario, Fernández-Ballester, Gregorio, Ferrer-Montiel, Antonio
Published in Expert opinion on investigational drugs (01.11.2020)
Published in Expert opinion on investigational drugs (01.11.2020)
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Journal Article
β-Lactam TRPM8 Antagonists Derived from Phe-Phenylalaninol Conjugates: Structure–Activity Relationships and Antiallodynic Activity
Martín-Escura, Cristina, Bonache, M. Ángeles, Medina, Jessy A., Medina-Peris, Alicia, De Andrés-López, Jorge, González-Rodríguez, Sara, Kerselaers, Sara, Fernández-Ballester, Gregorio, Voets, Thomas, Ferrer-Montiel, Antonio, Fernández-Carvajal, Asia, González-Muñiz, Rosario
Published in International journal of molecular sciences (01.10.2023)
Published in International journal of molecular sciences (01.10.2023)
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Journal Article
Estrogen destabilizes microtubules through an ion‐conductivity‐independent TRPV1 pathway
Goswami, Chandan, Kuhn, Julia, Dina, Olayinka A., Fernández‐Ballester, Gregorio, Levine, Jon D., Ferrer‐Montiel, Antonio, Hucho, Tim
Published in Journal of neurochemistry (01.06.2011)
Published in Journal of neurochemistry (01.06.2011)
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Journal Article
β-Lactam TRPM8 Antagonist RGM8-51 Displays Antinociceptive Activity in Different Animal Models
Martín-Escura, Cristina, Medina-Peris, Alicia, Spear, Luke A, de la Torre Martínez, Roberto, Olivos-Oré, Luis A, Barahona, María Victoria, González-Rodríguez, Sara, Fernández-Ballester, Gregorio, Fernández-Carvajal, Asia, Artalejo, Antonio R, Ferrer-Montiel, Antonio, González-Muñiz, Rosario
Published in International journal of molecular sciences (28.02.2022)
Published in International journal of molecular sciences (28.02.2022)
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Journal Article
Highly functionalized β-lactams and 2-ketopiperazines as TRPM8 antagonists with antiallodynic activity
Bonache, M Ángeles, Martín-Escura, Cristina, de la Torre Martínez, Roberto, Medina, Alicia, González-Rodríguez, Sara, Francesch, Andrés, Cuevas, Carmen, Roa, Ana María, Fernández-Ballester, Gregorio, Ferrer-Montiel, Antonio, Fernández-Carvajal, Asia, González-Muñiz, Rosario
Published in Scientific reports (25.08.2020)
Published in Scientific reports (25.08.2020)
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Journal Article
Identification of molecular determinants of channel gating in the transient receptor potential box of vanilloid receptor I
Valente, Pierluigi, García-Sanz, Nuria, Gomis, Ana, Fernández-Carvajal, Asia, Fernández-Ballester, Gregorio, Viana, Félix, Belmonte, Carlos, Ferrer-Montiel, Antonio
Published in The FASEB journal (01.09.2008)
Published in The FASEB journal (01.09.2008)
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Journal Article
Phenylalanine-Derived β-Lactam TRPM8 Modulators. Configuration Effect on the Antagonist Activity
Bonache, María Ángeles, Llabrés, Pedro Juan, Martín-Escura, Cristina, De la Torre-Martínez, Roberto, Medina-Peris, Alicia, Butrón, Laura, Gómez-Monterrey, Isabel, Roa, Ana María, Fernández-Ballester, Gregorio, Ferrer-Montiel, Antonio, Fernández-Carvajal, Asia, González-Muñiz, Rosario
Published in International journal of molecular sciences (27.02.2021)
Published in International journal of molecular sciences (27.02.2021)
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Journal Article
Structure-Based Design of Novel Biphenyl Amide Antagonists of Human Transient Receptor Potential Cation Channel Subfamily M Member 8 Channels with Potential Implications in the Treatment of Sensory Neuropathies
Journigan, V. Blair, Feng, Zhiwei, Rahman, Saifur, Wang, Yuanqiang, Amin, A. R. M. Ruhul, Heffner, Colleen E, Bachtel, Nicholas, Wang, Siyi, Gonzalez-Rodriguez, Sara, Fernández-Carvajal, Asia, Fernández-Ballester, Gregorio, Hilton, Jacob K, Van Horn, Wade D, Ferrer-Montiel, Antonio, Xie, Xiang-Qun, Rahman, Taufiq
Published in ACS chemical neuroscience (05.02.2020)
Published in ACS chemical neuroscience (05.02.2020)
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Journal Article
Competing Lipid-Protein and Protein-Protein Interactions Determine Clustering and Gating Patterns in the Potassium Channel from Streptomyces lividans (KcsA)
Molina, M. Luisa, Giudici, A. Marcela, Poveda, José A., Fernández-Ballester, Gregorio, Montoya, Estefanía, Renart, M. Lourdes, Fernández, Asia M., Encinar, José A., Riquelme, Gloria, Morales, Andrés, González-Ros, José M.
Published in The Journal of biological chemistry (16.10.2015)
Published in The Journal of biological chemistry (16.10.2015)
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Journal Article
Mutation of Ser-50 and Cys-66 in Snapin Modulates Protein Structure and Stability
Navarro, Aaron, Encinar, José A., López-Méndez, Blanca, Aguado-Llera, David, Prieto, Jesús, Gómez, Javier, Martínez-Cruz, Luís Alfonso, Millet, Oscar, González-Ros, José Manuel, Fernández-Ballester, Gregorio, Neira, José L., Ferrer-Montiel, Antonio
Published in Biochemistry (Easton) (24.04.2012)
Published in Biochemistry (Easton) (24.04.2012)
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Journal Article
TRPM8 contributes to sex dimorphism by promoting recovery of normal sensitivity in a mouse model of chronic migraine
Alarcón-Alarcón, David, Cabañero, David, de Andrés-López, Jorge, Nikolaeva-Koleva, Magdalena, Giorgi, Simona, Fernández-Ballester, Gregorio, Fernández-Carvajal, Asia, Ferrer-Montiel, Antonio
Published in Nature communications (22.10.2022)
Published in Nature communications (22.10.2022)
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Journal Article
Comprehensive Survey of Consensus Docking for High-Throughput Virtual Screening
Blanes-Mira, Clara, Fernández-Aguado, Pilar, de Andrés-López, Jorge, Fernández-Carvajal, Asia, Ferrer-Montiel, Antonio, Fernández-Ballester, Gregorio
Published in Molecules (Basel, Switzerland) (25.12.2022)
Published in Molecules (Basel, Switzerland) (25.12.2022)
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Journal Article
Small peptides patterned after the N‐terminus domain of SNAP25 inhibit SNARE complex assembly and regulated exocytosis
Blanes‐Mira, Clara, Merino, Jaime M., Valera, Elvira, Fernández‐Ballester, Gregorio, Gutiérrez, Luis M., Viniegra, Salvador, Pérez‐Payá, Enrique, Ferrer‐Montiel, Antonio
Published in Journal of neurochemistry (01.01.2004)
Published in Journal of neurochemistry (01.01.2004)
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Journal Article
A capsaicinoid-based soft drug, AG1529, for attenuating TRPV1-mediated histaminergic and inflammatory sensory neuron excitability
Nikolaeva-Koleva, Magdalena, Butron, Laura, González-Rodríguez, Sara, Devesa, Isabel, Valente, Pierluigi, Serafini, Marta, Genazzani, Armando A, Pirali, Tracey, Ballester, Gregorio Fernández, Fernández-Carvajal, Asia, Ferrer-Montiel, Antonio
Published in Scientific reports (08.01.2021)
Published in Scientific reports (08.01.2021)
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Journal Article
Design and validation of neuronal exocytosis blocking peptides as potential novel antiperspirants
Butron, Laura, Nikolaeva‐Koleva, Magdalena, Sempere, Ana, Rivero, Verónica, Fernandez‐Ballester, Gregorio, Espinosa, Ana, Vergassola, Matteo, Mastrocola, Elena, Zucchi, Sara, Ragni, Lorella, Fernández‐Carvajal, Asia, Mangano, Giorgina, Ferrer‐Montiel, Antonio, Devesa, Isabel
Published in Experimental dermatology (01.07.2023)
Published in Experimental dermatology (01.07.2023)
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Journal Article
Peimine, an Anti-Inflammatory Compound from Chinese Herbal Extracts, Modulates Muscle-Type Nicotinic Receptors
Alberola-Die, Armando, Encinar, José Antonio, Cobo, Raúl, Fernández-Ballester, Gregorio, González-Ros, José Manuel, Ivorra, Isabel, Morales, Andrés
Published in International journal of molecular sciences (19.10.2021)
Published in International journal of molecular sciences (19.10.2021)
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