Structural complementarity facilitates E7820-mediated degradation of RBM39 by DCAF15
Faust, Tyler B, Yoon, Hojong, Nowak, Radosław P, Donovan, Katherine A, Li, Zhengnian, Cai, Quan, Eleuteri, Nicholas A, Zhang, Tinghu, Gray, Nathanael S, Fischer, Eric S
Published in Nature chemical biology (01.01.2020)
Published in Nature chemical biology (01.01.2020)
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Journal Article
Bruton tyrosine kinase degradation as a therapeutic strategy for cancer
Dobrovolsky, Dennis, Wang, Eric S., Morrow, Sara, Leahy, Catharine, Faust, Tyler, Nowak, Radosław P., Donovan, Katherine A., Yang, Guang, Li, Zhengnian, Fischer, Eric S., Treon, Steven P., Weinstock, David M., Gray, Nathanael S.
Published in Blood (28.02.2019)
Published in Blood (28.02.2019)
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Journal Article
Functional Segregation of Overlapping Genes in HIV
Fernandes, Jason D., Faust, Tyler B., Strauli, Nicolas B., Smith, Cynthia, Crosby, David C., Nakamura, Robert L., Hernandez, Ryan D., Frankel, Alan D.
Published in Cell (15.12.2016)
Published in Cell (15.12.2016)
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Journal Article
The HIV-1 Tat protein recruits a ubiquitin ligase to reorganize the 7SK snRNP for transcriptional activation
Faust, Tyler B, Li, Yang, Bacon, Curtis W, Jang, Gwendolyn M, Weiss, Amit, Jayaraman, Bhargavi, Newton, Billy W, Krogan, Nevan J, D'Orso, Iván, Frankel, Alan D
Published in eLife (30.05.2018)
Published in eLife (30.05.2018)
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Journal Article
Small-Molecule Approaches to Targeted Protein Degradation
Faust, Tyler B, Donovan, Katherine A, Yue, Hong, Chamberlain, Philip P, Fischer, Eric S
Published in Annual review of cancer biology (04.03.2021)
Published in Annual review of cancer biology (04.03.2021)
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Journal Article
PJA2 ubiquitinates the HIV-1 Tat protein with atypical chain linkages to activate viral transcription
Faust, Tyler B, Li, Yang, Jang, Gwendolyn M, Johnson, Jeffrey R, Yang, Shumin, Weiss, Amit, Krogan, Nevan J, Frankel, Alan D
Published in Scientific reports (27.03.2017)
Published in Scientific reports (27.03.2017)
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Journal Article
Transition Step during Assembly of HIV Tat:P-TEFb Transcription Complexes and Transfer to TAR RNA
D'Orso, Iván, Jang, Gwendolyn M, Pastuszak, Alexander W, Faust, Tyler B, Quezada, Elizabeth, Booth, David S, Frankel, Alan D
Published in Molecular and Cellular Biology (01.12.2012)
Published in Molecular and Cellular Biology (01.12.2012)
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Journal Article
Triple Degradation of BTK, IKZF1 and IKZF3 in B-Cell Malignancies
Morrow, Sara, Dobrovolsky, Dennis, Wang, Eric, Nowak, Radosław P., Donovan, Katherine, Faust, Tyler, Yang, Guang, Li, Zhengnian, Fischer, Eric, Treon, Steven P, Weinstock, David M, Gray, Nathanael S.
Published in Blood (29.11.2018)
Published in Blood (29.11.2018)
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Journal Article
Abstract LB123: Poorer outcomes in EGFR L858R-driven NSCLC treated with osimertinib may be addressed with novel combination of BLU-945 and osimertinib
Elamin, Yasir Y., Rouskin-Faust, Tyler, Zhang, Nicole, Green, Teresa, Dhande, Aditya, Mar, Brenton G., Heymach, John V., Conti, Chiara
Published in Cancer research (Chicago, Ill.) (14.04.2023)
Published in Cancer research (Chicago, Ill.) (14.04.2023)
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Journal Article
PROTEIN TAG TO INDUCE LIGAND DEPENDENT DEGRADATION OF PROTEIN/PROTEIN-FUSIONS
NOWAK, Radoslaw P, BURMAN, Shourya Sonkar Roy, FISCHER, Eric S, FAUST, Tyler, YOON, Hojong
Year of Publication 13.09.2023
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Year of Publication 13.09.2023
Patent
SULFONAMIDE DERIVATIVES FOR PROTEIN DEGRADATION
Gray, Nathanael S, Fischer, Eric, Li, Zhengnian, Zhang, Tinghu, Cai, Quan, Faust, Tyler, Donovan, Katherine, Yoon, Hojong
Year of Publication 14.03.2024
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Year of Publication 14.03.2024
Patent
PROTEIN TAG TO INDUCE LIGAND DEPENDENT DEGRADATION OF PROTEIN/PROTEIN-FUSIONS
Burman, Shourya Sonkar Roy, Nowak, Radoslaw P, Faust, Tyler, Fischer, Eric S, Yoon, Hojong
Year of Publication 22.12.2022
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Year of Publication 22.12.2022
Patent
Sulfonamide derivatives for protein degradation
Gray, Nathanael S, Fischer, Eric, Li, Zhengnian, Zhang, Tinghu, Cai, Quan, Faust, Tyler, Donovan, Katherine, Yoon, Hojong
Year of Publication 07.11.2023
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Year of Publication 07.11.2023
Patent
PROTEIN TAG TO INDUCE LIGAND DEPENDENT DEGRADATION OF PROTEIN/PROTEIN-FUSIONS
NOWAK, Radoslaw P, BURMAN, Shourya Sonkar Roy, FISCHER, Eric S, FAUST, Tyler, YOON, Hojong
Year of Publication 27.07.2022
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Year of Publication 27.07.2022
Patent
Protein tag to induce ligand dependent degradation of protein/protein-fusions
NOWAK, Radoslaw P, BURMAN, Shourya Sonkar Roy, FISCHER, Eric S, FAUST, Tyler, YOON, Hojong
Year of Publication 24.02.2022
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Year of Publication 24.02.2022
Patent
PROTEIN TAG TO INDUCE LIGAND DEPENDENT DEGRADATION OF PROTEIN/PROTEIN-FUSIONS
NOWAK, Radoslaw P, BURMAN, Shourya Sonkar Roy, FISCHER, Eric S, FAUST, Tyler, YOON, Hojong
Year of Publication 25.03.2021
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Year of Publication 25.03.2021
Patent
PROTEIN TAG TO INDUCE LIGAND DEPENDENT DEGRADATION OF PROTEIN/PROTEIN-FUSIONS
FAUST, TYLER, BURMAN, SHOURYA SONKAR ROY, NOWAK, RADOSLAW P, YOON, HOJONG, FISCHER, ERIC S
Year of Publication 25.03.2021
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Year of Publication 25.03.2021
Patent