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Identification of Covalent Cyclic Peptide Inhibitors Targeting Protein–Protein Interactions Using Phage Display
Wang, Sijie, Faucher, Franco F., Bertolini, Matilde, Kim, Heeyoung, Yu, Bingchen, Cao, Li, Roeltgen, Katharina, Lovell, Scott, Shanker, Varun, Boyd, Scott D., Wang, Lei, Bartenschlager, Ralf, Bogyo, Matthew
Published in Journal of the American Chemical Society (05.03.2025)
Published in Journal of the American Chemical Society (05.03.2025)
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Macrocyclic Phage Display for Identification of Selective Protease Substrates
Faucher, Franco F., Blažková, Kristýna, Lovell, Scott, Bertolini, Matilde, Herrero-Bourdieu, Juan, Cosco, Emily D., Bogyo, Matthew, Barniol-Xicota, Marta
Published in Journal of the American Chemical Society (30.07.2025)
Published in Journal of the American Chemical Society (30.07.2025)
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Identification of covalent inhibitors of Staphylococcus aureus serine hydrolases important for virulence and biofilm formation
Upadhyay, Tulsi, Woods, Emily C., Dela Ahator, Stephen, Julin, Kjersti, Faucher, Franco F., Uddin, Md Jalal, Hollander, Marijn J., Pedowitz, Nichole J., Abegg, Daniel, Hammond, Isabella, Eke, Ifeanyichukwu E., Wang, Sijie, Chen, Shiyu, Bennett, John M., Jo, Jeyun, Lentz, Christian S., Adibekian, Alexander, Fellner, Matthias, Bogyo, Matthew
Published in Nature communications (30.05.2025)
Published in Nature communications (30.05.2025)
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Highlights from the Lowlands: Early Career Researchers Shine at Medicinal Chemistry Frontiers 2024
McKenna, Sean M., Borsari, Chiara, Chin Chan, Sean, Donckele, Etienne J., Faucher, Franco F., Grenier‐Davies, Melissa C., Haranahalli, Krupanandan, Matagne, Brieuc, Monastyrskyi, Andrii, Petracca, Rita
Published in ChemMedChem (16.02.2025)
Published in ChemMedChem (16.02.2025)
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Protease Activated Probes for Real-Time Ratiometric Imaging of Solid Tumors
Faucher, Franco F., Liu, Kevin J., Cosco, Emily D., Widen, John C., Sorger, Jonathan, Guerra, Matteo, Bogyo, Matthew
Published in ACS central science (24.05.2023)
Published in ACS central science (24.05.2023)
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New Insights into Aldol Reactions of Methyl Isocyanoacetate Catalyzed by Heterogenized Homogeneous Catalysts
Ye, Rong, Zhao, Jie, Yuan, Bing, Liu, Wen-Chi, Rodrigues De Araujo, Joyce, Faucher, Franco F, Chang, Matthew, Deraedt, Christophe V, Toste, F. Dean, Somorjai, Gabor A
Published in Nano letters (11.01.2017)
Published in Nano letters (11.01.2017)
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Covalent Macrocyclic Proteasome Inhibitors Mitigate Resistance in Plasmodium falciparum
Bennett, John M., Ward, Kurt E., Muir, Ryan K., Kabeche, Stephanie, Yoo, Euna, Yeo, Tomas, Lam, Grace, Zhang, Hao, Almaliti, Jehad, Berger, Gabriel, Faucher, Franco F., Lin, Gang, Gerwick, William H., Yeh, Ellen, Fidock, David A., Bogyo, Matthew
Published in ACS infectious diseases (13.10.2023)
Published in ACS infectious diseases (13.10.2023)
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Polymer-Tethered Quenched Fluorescent Probes for Enhanced Imaging of Tumor-Associated Proteases
Hadzima, Martin, Faucher, Franco F., Blažková, Kristýna, Yim, Joshua J., Guerra, Matteo, Chen, Shiyu, Woods, Emily C., Park, Ki Wan, Šácha, Pavel, Šubr, Vladimír, Kostka, Libor, Etrych, Tomáš, Majer, Pavel, Konvalinka, Jan, Bogyo, Matthew
Published in ACS sensors (26.07.2024)
Published in ACS sensors (26.07.2024)
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Macrocyclic phage display for identification of selective protease substrates
Faucher, Franco F, Lovell, Scott, Bertolini, Matilde, Blažková, Kristýna, Cosco, Emily D, Bogyo, Matthew, Barniol-Xicota, Marta
Published in bioRxiv (15.03.2025)
Published in bioRxiv (15.03.2025)
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Solid Phase Synthesis of Fluorosulfate Containing Macrocycles for Chemoproteomic Workflows
Faucher, Franco F, Abegg, Daniel, Ipock, Phillip, Adibekian, Alexander, Lovell, Scott, Bogyo, Matthew
Published in bioRxiv (18.02.2023)
Published in bioRxiv (18.02.2023)
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Identification of Covalent Cyclic Peptide Inhibitors Targeting Protein-Protein Interactions Using Phage Display
Wang, Sijie, Faucher, Franco F, Bertolini, Matilde, Kim, Heeyoung, Yu, Bingchen, Cao, Li, Roeltgen, Katharina, Lovell, Scott, Shanker, Varun, Boyd, Scott D, Wang, Lei, Bartenschlager, Ralf, Bogyo, Matthew
Published in bioRxiv (09.11.2024)
Published in bioRxiv (09.11.2024)
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Strategies for Tuning the Selectivity of Chemical Probes that Target Serine Hydrolases
Faucher, Franco, Bennett, John M., Bogyo, Matthew, Lovell, Scott
Published in Cell chemical biology (20.08.2020)
Published in Cell chemical biology (20.08.2020)
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Mixed Alkyl/Aryl Phosphonates Identify Metabolic Serine Hydrolases as Antimalarial Targets
Bennett, John M, Narwal, Sunil K, Kabeche, Stephanie, Abegg, Daniel, Hackett, Fiona, Yeo, Tomas, Li, Veronica L, Muir, Ryan K, Faucher, Franco F, Lovell, Scott, Blackman, Michael J, Adibekian, Alexander, Yeh, Ellen, Fidock, David A, Bogyo, Matthew
Published in bioRxiv (11.01.2024)
Published in bioRxiv (11.01.2024)
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EVIDENCE OF PROTEASE-MEDIATED PRO-NOCICEPTIVE EFFECTS IN INFLAMMATORY BOWEL DISEASE PATIENTS
Wood, Hannah, Blazkova, Kristyna, Faucher, Franco, Sheth, Prameet M., Vanner, Stephen J., Reed, David E., Bogyo, Matthew, Lomax, Alan
Published in Gastroenterology (New York, N.Y. 1943) (01.02.2025)
Published in Gastroenterology (New York, N.Y. 1943) (01.02.2025)
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EVIDENCE OF PROTEASE-MEDIATED PRO-NOCICEPTIVE EFFECTS IN INFLAMMATORY BOWEL DISEASE PATIENTS
Wood, Hannah, Blazkova, Kristyna, Faucher, Franco, Sheth, Prameet M, Vanner, Stephen J, Reed, David E, Bogyo, Matthew, Lomax, Alan
Published in Inflammatory bowel diseases (28.02.2025)
Published in Inflammatory bowel diseases (28.02.2025)
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Mixed alkyl/aryl phosphonates identify metabolic serine hydrolases as antimalarial targets
Bennett, John M., Narwal, Sunil K., Kabeche, Stephanie, Abegg, Daniel, Thathy, Vandana, Hackett, Fiona, Yeo, Tomas, Li, Veronica L., Muir, Ryan, Faucher, Franco, Lovell, Scott, Blackman, Michael J., Adibekian, Alexander, Yeh, Ellen, Fidock, David A., Bogyo, Matthew
Published in Cell chemical biology (19.09.2024)
Published in Cell chemical biology (19.09.2024)
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Chemoproteomic identification of a DPP4 homolog in Bacteroides thetaiotaomicron
Keller, Laura J., Nguyen, Taylor H., Liu, Lawrence J., Hurysz, Brianna M., Lakemeyer, Markus, Guerra, Matteo, Gelsinger, Danielle J., Chanin, Rachael, Ngo, Nhi, Lum, Kenneth M., Faucher, Franco, Ipock, Phillip, Niphakis, Micah J., Bhatt, Ami S., O’Donoghue, Anthony J., Huang, Kerwyn Casey, Bogyo, Matthew
Published in Nature chemical biology (01.12.2023)
Published in Nature chemical biology (01.12.2023)
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New Insights into Aldol Reactions of Methyl Isocyanoacetate Catalyzed by Heterogenized Homogeneous Catalysts
Ye, Rong, Zhao, Jie, Yuan, Bing, Liu, Wen-Chi, Rodrigues De Araujo, Joyce, Faucher, Franco F., Chang, Matthew, Deraedt, Christophe V., Toste, F. Dean, Somorjai, Gabor A.
Published in Nano letters (14.12.2016)
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Published in Nano letters (14.12.2016)
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