Selective Sensing of Darolutamide and Thalidomide in Pharmaceutical Preparations and in Spiked Biofluids
Talaat, Wael, Farahat, Abdelbasset A, Keshk, Reda Mohammed
Published in Biosensors (Basel) (11.11.2022)
Published in Biosensors (Basel) (11.11.2022)
Get full text
Journal Article
Heterocyclic Diamidine DNA Ligands as HOXA9 Transcription Factor Inhibitors: Design, Molecular Evaluation, and Cellular Consequences in a HOXA9-Dependant Leukemia Cell Model
Depauw, Sabine, Lambert, Mélanie, Jambon, Samy, Paul, Ananya, Peixoto, Paul, Nhili, Raja, Marongiu, Laura, Figeac, Martin, Dassi, Christelle, Paul-Constant, Charles, Billoré, Benjamin, Kumar, Arvind, Farahat, Abdelbasset A, Ismail, Mohamed A, Mineva, Ekaterina, Sweat, Daniel P, Stephens, Chad E, Boykin, David W, Wilson, W. David, David-Cordonnier, Marie-Hélène
Published in Journal of medicinal chemistry (14.02.2019)
Published in Journal of medicinal chemistry (14.02.2019)
Get full text
Journal Article
Pharmacological inhibition of the transcription factor PU.1 in leukemia
Antony-Debré, Iléana, Paul, Ananya, Leite, Joana, Mitchell, Kelly, Kim, Hye Mi, Carvajal, Luis A, Todorova, Tihomira I, Huang, Kenneth, Kumar, Arvind, Farahat, Abdelbasset A, Bartholdy, Boris, Narayanagari, Swathi-Rao, Chen, Jiahao, Ambesi-Impiombato, Alberto, Ferrando, Adolfo A, Mantzaris, Ioannis, Gavathiotis, Evripidis, Verma, Amit, Will, Britta, Boykin, David W, Wilson, W David, Poon, Gregory Mk, Steidl, Ulrich
Published in The Journal of clinical investigation (01.12.2017)
Published in The Journal of clinical investigation (01.12.2017)
Get full text
Journal Article
Investigation of the effect of structure modification of furamidine on the DNA minor groove binding and antiprotozoal activity
Farahat, Abdelbasset A., Kumar, Arvind, Wenzler, Tanja, Brun, Reto, Paul, Ananya, Guo, Pu, Wilson, W. David, Boykin, David W.
Published in European journal of medicinal chemistry (05.04.2023)
Published in European journal of medicinal chemistry (05.04.2023)
Get full text
Journal Article
G‐quadruplex‐binding small molecules ameliorate C9orf72 FTD/ALS pathology in vitro and in vivo
Simone, Roberto, Balendra, Rubika, Moens, Thomas G, Preza, Elisavet, Wilson, Katherine M, Heslegrave, Amanda, Woodling, Nathan S, Niccoli, Teresa, Gilbert‐Jaramillo, Javier, Abdelkarim, Samir, Clayton, Emma L, Clarke, Mica, Konrad, Marie‐Therese, Nicoll, Andrew J, Mitchell, Jamie S, Calvo, Andrea, Chio, Adriano, Houlden, Henry, Polke, James M, Ismail, Mohamed A, Stephens, Chad E, Vo, Tam, Farahat, Abdelbasset A, Wilson, W David, Boykin, David W, Zetterberg, Henrik, Partridge, Linda, Wray, Selina, Parkinson, Gary, Neidle, Stephen, Patani, Rickie, Fratta, Pietro, Isaacs, Adrian M
Published in EMBO molecular medicine (01.01.2018)
Published in EMBO molecular medicine (01.01.2018)
Get full text
Journal Article
Indole and Benzimidazole Bichalcophenes: Synthesis, DNA Binding and Antiparasitic Activity
Farahat, Abdelbasset A., Ismail, Mohamed A., Kumar, Arvind, Wenzler, Tanja, Brun, Reto, Paul, Ananya, Wilson, W. David, Boykin, David W.
Published in European journal of medicinal chemistry (01.01.2018)
Published in European journal of medicinal chemistry (01.01.2018)
Get full text
Journal Article
Extending the σ‑Hole Motif for Sequence-Specific Recognition of the DNA Minor Groove
Guo, Pu, Farahat, Abdelbasset A, Paul, Ananya, Kumar, Arvind, Boykin, David W, Wilson, W. David
Published in Biochemistry (Easton) (12.05.2020)
Published in Biochemistry (Easton) (12.05.2020)
Get full text
Journal Article
In Silico and In Vitro Evaluation of Some Amidine Derivatives as Hit Compounds towards Development of Inhibitors against Coronavirus Diseases
Hassan, Ahmed H E, El-Sayed, Selwan M, Yamamoto, Mizuki, Gohda, Jin, Matsumoto, Takehisa, Shirouzu, Mikako, Inoue, Jun-Ichiro, Kawaguchi, Yasushi, Mansour, Reem M A, Anvari, Abtin, Farahat, Abdelbasset A
Published in Viruses (15.05.2023)
Published in Viruses (15.05.2023)
Get full text
Journal Article
Pharmacological restriction of genomic binding sites redirects PU.1 pioneer transcription factor activity
Taylor, Samuel J, Stauber, Jacob, Bohorquez, Oliver, Tatsumi, Goichi, Kumari, Rajni, Chakraborty, Joyeeta, Bartholdy, Boris A, Schwenger, Emily, Sundaravel, Sriram, Farahat, Abdelbasset A, Wheat, Justin C, Goldfinger, Mendel, Verma, Amit, Kumar, Arvind, Boykin, David W, Stengel, Kristy R, Poon, Gregory M K, Steidl, Ulrich
Published in Nature genetics (18.09.2024)
Published in Nature genetics (18.09.2024)
Get full text
Journal Article
Targeting the DNA-binding activity of the human ERG transcription factor using new heterocyclic dithiophene diamidines
Nhili, Raja, Peixoto, Paul, Depauw, Sabine, Flajollet, Sébastien, Dezitter, Xavier, Munde, Manoj M, Ismail, Mohamed A, Kumar, Arvind, Farahat, Abdelbasset A, Stephens, Chad E, Duterque-Coquillaud, Martine, David Wilson, W, Boykin, David W, David-Cordonnier, Marie-Hélène
Published in Nucleic acids research (01.01.2013)
Published in Nucleic acids research (01.01.2013)
Get full text
Journal Article
Web Resource
The Thiophene "Sigma-Hole" as a Concept for Preorganized, Specific Recognition of G⋅C Base Pairs in the DNA Minor Groove
Guo, Pu, Paul, Ananya, Kumar, Arvind, Farahat, Abdelbasset A., Kumar, Dhiraj, Wang, Siming, Boykin, David W., Wilson, W. David
Published in Chemistry : a European journal (17.10.2016)
Published in Chemistry : a European journal (17.10.2016)
Get full text
Journal Article
REACTIVITY OF 4-BROMOACETYL-1,2,3-TRIAZOLES TOWARDS AMINES AND PHENOLS: SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF NOVEL HETEROCYCLES
Abdel-Wahab, Bakr F., Mohamed, Hanan A., Farahat, Abdelbasset A., Kariuki, Benson M., El-Hiti, Gamal A.
Published in Heterocycles (01.09.2022)
Published in Heterocycles (01.09.2022)
Get more information
Journal Article
The Thiophene "Sigma-Hole" as a Concept for Preorganized, Specific Recognition of G.C Base Pairs in the DNA Minor Groove
Guo, Pu, Paul, Ananya, Kumar, Arvind, Farahat, Abdelbasset A., Kumar, Dhiraj, Wang, Siming, Boykin, David W., Wilson, W. David
Published in Chemistry : a European journal (01.10.2016)
Published in Chemistry : a European journal (01.10.2016)
Get full text
Journal Article