Search Results - "FUSHIMI, NOBUHIKO" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Mizagliflozin, a novel selective SGLT1 inhibitor, exhibits potential in the amelioration of chronic constipation

Mizagliflozin, a novel selective SGLT1 inhibitor, exhibits potential in the amelioration of chronic constipation

by Inoue, Toshihiro, Takemura, Masaaki, Fushimi, Nobuhiko, Fujimori, Yoshikazu, Onozato, Tomoya, Kurooka, Takao, Asari, Tetsuya, Takeda, Hiroo, Kobayashi, Mamoru, Nishibe, Hironori, Isaji, Masayuki
Published in European journal of pharmacology (05.07.2017)

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Journal Article

KGA-2727, a novel selective inhibitor of a high-affinity sodium glucose cotransporter (SGLT1), exhibits antidiabetic efficacy in rodent models

KGA-2727, a novel selective inhibitor of a high-affinity sodium glucose cotransporter (SGLT1), exhibits antidiabetic efficacy in rodent models

by Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Fushimi, Nobuhiko, Itoh, Fumiaki, Yamada, Mitsuhiko, Isaji, Masayuki
Published in The Journal of pharmacology and experimental therapeutics (01.08.2012)

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Journal Article

The juxtamembrane region of TrkA kinase is critical for inhibitor selectivity

The juxtamembrane region of TrkA kinase is critical for inhibitor selectivity

by Furuya, Noritaka, Momose, Takaki, Katsuno, Kenji, Fushimi, Nobuhiko, Muranaka, Hideyuki, Handa, Chiaki, Ozawa, Tomonaga, Kinoshita, Takayoshi
Published in Bioorganic & medicinal chemistry letters (01.03.2017)

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Journal Article

Pharmacological characterization of linzagolix, a novel, orally active, non‐peptide antagonist of gonadotropin‐releasing hormone receptors

Pharmacological characterization of linzagolix, a novel, orally active, non‐peptide antagonist of gonadotropin‐releasing hormone receptors

by Tezuka, Motohiro, Tamai, Yasuaki, Kuramochi, Yu, Kobayashi, Kaoru, Fushimi, Nobuhiko, Kiguchi, Sumiyoshi
Published in Clinical and experimental pharmacology & physiology (01.10.2022)

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Journal Article

An isoform-selective inhibitor of tropomyosin receptor kinase A behaves as molecular glue

An isoform-selective inhibitor of tropomyosin receptor kinase A behaves as molecular glue

by Furuya, Noritaka, Momose, Takaki, Katsuno, Kenji, Fushimi, Nobuhiko, Muranaka, Hideyuki, Handa, Chiaki, Sawa, Masaaki, Ozawa, Tomonaga, Kinoshita, Takayoshi
Published in Bioorganic & medicinal chemistry letters (01.01.2020)

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Journal Article

Discovery of remogliflozin etabonate: A potent and highly selective SGLT2 inhibitor

Discovery of remogliflozin etabonate: A potent and highly selective SGLT2 inhibitor

by Shimizu, Kazuo, Fujikura, Hideki, Fushimi, Nobuhiko, Nishimura, Toshihiro, Tatani, Kazuya, Katsuno, Kenji, Fujimori, Yoshikazu, Watanabe, Shinjiro, Hiratochi, Masahiro, Nakabayashi, Takeshi, Kamada, Noboru, Arakawa, Koichi, Hikawa, Hidemasa, Azumaya, Isao, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (15.03.2021)

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Journal Article

Synthesis and structure-activity relationships of 1-benzylindane derivatives as selective agonists for estrogen receptor beta

Synthesis and structure-activity relationships of 1-benzylindane derivatives as selective agonists for estrogen receptor beta

by Yonekubo, Shigeru, Fushimi, Nobuhiko, Miyagi, Takashi, Nakanishi, Osamu, Katsuno, Kenji, Ozawa, Motoyasu, Handa, Chiaki, Furuya, Noritaka, Muranaka, Hideyuki
Published in Bioorganic & medicinal chemistry (15.11.2016)

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Journal Article

Structure–activity relationship studies of 4-benzyl-1H-pyrazol-3-yl β-d-glucopyranoside derivatives as potent and selective sodium glucose co-transporter 1 (SGLT1) inhibitors with therapeutic activity on postprandial hyperglycemia

Structure–activity relationship studies of 4-benzyl-1H-pyrazol-3-yl β-d-glucopyranoside derivatives as potent and selective sodium glucose co-transporter 1 (SGLT1) inhibitors with therapeutic activity on postprandial hyperglycemia

by Fushimi, Nobuhiko, Fujikura, Hideki, Shiohara, Hiroaki, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Ozawa, Tomonaga, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (15.11.2012)

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Journal Article

Design, synthesis, and structure–activity relationships of a series of 4-benzyl-5-isopropyl-1H-pyrazol-3-yl β-d-glycopyranosides substituted with novel hydrophilic groups as highly potent inhibitors of sodium glucose co-transporter 1 (SGLT1)

Design, synthesis, and structure–activity relationships of a series of 4-benzyl-5-isopropyl-1H-pyrazol-3-yl β-d-glycopyranosides substituted with novel hydrophilic groups as highly potent inhibitors of sodium glucose co-transporter 1 (SGLT1)

by Fushimi, Nobuhiko, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Yamauchi, Yuji, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (01.02.2013)

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Journal Article

METHOD FOR PRODUCING PYRAZOLE DERIVATIVE

METHOD FOR PRODUCING PYRAZOLE DERIVATIVE

by KIJIMA YOSHIRO, MUTAI YOSUKE, FUSHIMI NOBUHIKO, HIRASAWA HIDEAKI, TANADA FUMIYA, KOBAYASHI JUNICHI
Year of Publication 12.07.2018

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Patent

TRPM8 INHIBITOR

TRPM8 INHIBITOR

by KIJIMA YOSHIRO, MUTAI YOSUKE, FUSHIMI NOBUHIKO, HIRASAWA HIDEAKI, TANADA FUMIYA, KOBAYASHI JUNICHI
Year of Publication 28.06.2018

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Patent

피라졸 유도체, 또는 그 약리학적으로 허용되는 염

피라졸 유도체, 또는 그 약리학적으로 허용되는 염

by MUTAI YOUSUKE, KIJIMA YOSHIRO, FUSHIMI NOBUHIKO, HIRASAWA HIDEAKI, TANADA FUMIYA, KOBAYASHI JUNICHI
Year of Publication 12.02.2018

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Patent

PYRAZOLE DERIVATIVE, OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF

PYRAZOLE DERIVATIVE, OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF

by TANADA, Fumiya, HIRASAWA, Hideaki, KIJIMA, Yoshiro, MUTAI, Yousuke, FUSHIMI, Nobuhiko, KOBAYASHI, Junichi
Year of Publication 29.12.2016

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Patent

Design, synthesis, and structure-activity relationships of a series of 4-benzyl-5-isopropyl-1H-pyrazol-3-yl I2-d-glycopyranosides substituted with novel hydrophilic groups as highly potent inhibitors of sodium glucose co-transporter 1 (SGLT1)

Design, synthesis, and structure-activity relationships of a series of 4-benzyl-5-isopropyl-1H-pyrazol-3-yl I2-d-glycopyranosides substituted with novel hydrophilic groups as highly potent inhibitors of sodium glucose co-transporter 1 (SGLT1)

by Fushimi, Nobuhiko, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Yamauchi, Yuji, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (01.02.2013)

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Journal Article

Design, synthesis, and structure-activity relationships of a series of 4-benzyl-5-isopropyl-1H-pyrazol-3-yl [beta]-d-glycopyranosides substituted with novel hydrophilic groups as highly potent inhibitors of sodium glucose co-transporter 1 (SGLT1)

Design, synthesis, and structure-activity relationships of a series of 4-benzyl-5-isopropyl-1H-pyrazol-3-yl [beta]-d-glycopyranosides substituted with novel hydrophilic groups as highly potent inhibitors of sodium glucose co-transporter 1 (SGLT1)

by Fushimi, Nobuhiko, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Yamauchi, Yuji, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (01.02.2013)

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Journal Article

Structure-activity relationship studies of 4-benzyl-1H-pyrazol-3-yl I2-d-glucopyranoside derivatives as potent and selective sodium glucose co-transporter 1 (SGLT1) inhibitors with therapeutic activity on postprandial hyperglycemia

Structure-activity relationship studies of 4-benzyl-1H-pyrazol-3-yl I2-d-glucopyranoside derivatives as potent and selective sodium glucose co-transporter 1 (SGLT1) inhibitors with therapeutic activity on postprandial hyperglycemia

by Fushimi, Nobuhiko, Fujikura, Hideki, Shiohara, Hiroaki, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Ozawa, Tomonaga, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (01.11.2012)

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Journal Article

1-SUBSTITUTED-3-ß-D-GLUCOPYRANOSYLATED NITROGENOUS HETERO- CYCLIC COMPOUNDS AND MEDICINES CONTAINING THE SAME

1-SUBSTITUTED-3-ß-D-GLUCOPYRANOSYLATED NITROGENOUS HETERO- CYCLIC COMPOUNDS AND MEDICINES CONTAINING THE SAME

by FUSHIMI, NOBUHIKO, YONEKUBO, SHIGERU
Year of Publication 26.05.2006

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Patent

NITROGENATED FUSED-RING DERIVATIVE, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND USE OF THE SAME FOR MEDICAL PURPOSES

NITROGENATED FUSED-RING DERIVATIVE, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND USE OF THE SAME FOR MEDICAL PURPOSES

by OHNO, KOHSUKE, FUSHIMI, NOBUHIKO, YONEKUBO, SHIGERU, MIYAGI, TAKASHI
Year of Publication 26.03.2009

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Patent

NAPHTHALENE DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF

NAPHTHALENE DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF

by FUJIKURA, HIDEKI, FUSHIMI, NOBUHIKO, ISAJI, MASAYUKI
Year of Publication 13.10.2005

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Patent

NAPHTHALENE DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF

NAPHTHALENE DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF

by FUJIKURA, HIDEKI, FUSHIMI, NOBUHIKO, ISAJI, MASAYUKI
Year of Publication 13.10.2005

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Patent

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