An end-to-end automated platform process for high-throughput engineering of next-generation multi-specific antibody therapeutics
Furtmann, Norbert, Schneider, Marion, Spindler, Nadja, Steinmann, Bjoern, Li, Ziyu, Focken, Ingo, Meyer, Joachim, Dimova, Dilyana, Kroll, Katja, Leuschner, Wulf Dirk, Debeaumont, Audrey, Mathieu, Magali, Lange, Christian, Dittrich, Werner, Kruip, Jochen, Schmidt, Thorsten, Birkenfeld, Joerg
Published in mAbs (01.01.2021)
Published in mAbs (01.01.2021)
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Journal Article
Comprehensive knowledge base of two- and three-dimensional activity cliffs for medicinal and computational chemistry
Hu, Ye, Furtmann, Norbert, Stumpfe, Dagmar, Bajorath, Jürgen
Published in F1000 research (25.06.2015)
Published in F1000 research (25.06.2015)
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Journal Article
Identification of New Chromenone Derivatives as Cholinesterase Inhibitors and Molecular Docking Studies
Iqbal, Jamshed, Abbasi, Muhammad S A, Zaib, Sumera, Afridi, Saifullah, Furtmann, Norbert, Bajorath, Jürgen, Langer, Peter
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2018)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2018)
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Journal Article
Best practices for machine learning in antibody discovery and development
Wossnig, Leonard, Furtmann, Norbert, Buchanan, Andrew, Kumar, Sandeep, Greiff, Victor
Published in Drug discovery today (01.07.2024)
Published in Drug discovery today (01.07.2024)
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Journal Article
Current compound coverage of the kinome
Hu, Ye, Furtmann, Norbert, Bajorath, Jürgen
Published in Journal of medicinal chemistry (08.01.2015)
Published in Journal of medicinal chemistry (08.01.2015)
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Journal Article
Active compounds from a diverse library of triazolothiadiazole and triazolothiadiazine scaffolds: Synthesis, crystal structure determination, cytotoxicity, cholinesterase inhibitory activity, and binding mode analysis
Khan, Imtiaz, Ibrar, Aliya, Zaib, Sumera, Ahmad, Sarfraz, Furtmann, Norbert, Hameed, Shahid, Simpson, Jim, Bajorath, Jürgen, Iqbal, Jamshed
Published in Bioorganic & medicinal chemistry (01.11.2014)
Published in Bioorganic & medicinal chemistry (01.11.2014)
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Journal Article
Computational Screening for mAb Colloidal Stability with Coarse-Grained, Molecular-Scale Simulations
Janke, J. Joel, Starr, Charles G., Kingsbury, Jonathan S., Furtmann, Norbert, Roberts, Christopher J., Calero-Rubio, Cesar
Published in The journal of physical chemistry. B (15.02.2024)
Published in The journal of physical chemistry. B (15.02.2024)
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Journal Article
Coumarin-thiazole and -oxadiazole derivatives: Synthesis, bioactivity and docking studies for aldose/aldehyde reductase inhibitors
Ibrar, Aliya, Tehseen, Yildiz, Khan, Imtiaz, Hameed, Abdul, Saeed, Aamer, Furtmann, Norbert, Bajorath, Jürgen, Iqbal, Jamshed
Published in Bioorganic chemistry (01.10.2016)
Published in Bioorganic chemistry (01.10.2016)
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Journal Article
High-Throughput and Format-Agnostic Mispairing Assay for Multispecific Antibodies Using Intact Mass Spectrometry
Ziegengeist, Tanja, Orth, Jennifer, Kroll, Katja, Schneider, Marion, Spindler, Nadja, Dimova, Dilyana, Handschuh, Severin, Brandenburg, Arnd, Ossola, Reto, Furtmann, Norbert, Birkenfeld, Joerg, Beil, Christian, Hoffmann, Dietmar, Schmidt, Thorsten, Sendak, Rebecca, Fischer, Melanie, Hölper, Soraya, Kühn, Jennifer
Published in Analytical chemistry (Washington) (11.07.2023)
Published in Analytical chemistry (Washington) (11.07.2023)
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Journal Article
Structural Optimization of Azadipeptide Nitriles Strongly Increases Association Rates and Allows the Development of Selective Cathepsin Inhibitors
Frizler, Maxim, Lohr, Friederike, Furtmann, Norbert, Kläs, Julia, Gütschow, Michael
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
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Journal Article
A Coumarin-Labeled Vinyl Sulfone as Tripeptidomimetic Activity-Based Probe for Cysteine Cathepsins
Mertens, Matthias D., Schmitz, Janina, Horn, Martin, Furtmann, Norbert, Bajorath, Jürgen, Mareš, Michael, Gütschow, Michael
Published in Chembiochem : a European journal of chemical biology (05.05.2014)
Published in Chembiochem : a European journal of chemical biology (05.05.2014)
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Journal Article
Novel structural hybrids of pyrazolobenzothiazines with benzimidazoles as cholinesterase inhibitors
Aslam, Sana, Zaib, Sumera, Ahmad, Matloob, Gardiner, John M., Ahmad, Aqeel, Hameed, Abdul, Furtmann, Norbert, Guetschow, Michael, Bajorath, Juergen, Iqbal, Jamshed
Published in European journal of medicinal chemistry (06.05.2014)
Published in European journal of medicinal chemistry (06.05.2014)
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Journal Article
Current Compound Coverage of the Kinome: Miniperspective
Hu, Ye, Furtmann, Norbert, Bajorath, Jürgen
Published in Journal of medicinal chemistry (08.01.2015)
Published in Journal of medicinal chemistry (08.01.2015)
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Journal Article
Trispecific antibody targeting HIV-1 and T cells activates and eliminates latently-infected cells in HIV/SHIV infections
Promsote, Wanwisa, Xu, Ling, Hataye, Jason, Fabozzi, Giulia, March, Kylie, Almasri, Cassandra G, DeMouth, Megan E, Lovelace, Sarah E, Talana, Chloe Adrienna, Doria-Rose, Nicole A, McKee, Krisha, Hait, Sabrina Helmold, Casazza, Joseph P, Ambrozak, David, Beninga, Jochen, Rao, Ercole, Furtmann, Norbert, Birkenfeld, Joerg, McCarthy, Elizabeth, Todd, John-Paul, Petrovas, Constantinos, Connors, Mark, Hebert, Andrew T, Beck, Jeremy, Shen, Junqing, Zhang, Bailin, Levit, Mikhail, Wei, Ronnie R, Yang, Zhi-Yong, Pegu, Amarendra, Mascola, John R, Nabel, Gary J, Koup, Richard A
Published in Nature communications (22.06.2023)
Published in Nature communications (22.06.2023)
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Journal Article