A landmark in drug discovery based on complex natural product synthesis
Kawano, Satoshi, Ito, Ken, Yahata, Kenzo, Kira, Kazunobu, Abe, Takanori, Akagi, Tsuyoshi, Asano, Makoto, Iso, Kentaro, Sato, Yuki, Matsuura, Fumiyoshi, Ohashi, Isao, Matsumoto, Yasunobu, Isomura, Minetaka, Sasaki, Takeo, Fukuyama, Takashi, Miyashita, Yusuke, Kaburagi, Yosuke, Yokoi, Akira, Asano, Osamu, Owa, Takashi, Kishi, Yoshito
Published in Scientific reports (17.06.2019)
Published in Scientific reports (17.06.2019)
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Journal Article
Total Synthesis and Stereochemistry of Pinnatoxins B and C
Matsuura, Fumiyoshi, Hao, Junliang, Reents, Reinhard, Kishi, Yoshito
Published in Organic letters (20.07.2006)
Published in Organic letters (20.07.2006)
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Journal Article
Stereochemistry of Pteriatoxins A, B, and C
Hao, Junliang, Matsuura, Fumiyoshi, Kishi, Yoshito, Kita, Masaki, Uemura, Daisuke, Asai, Naoki, Iwashita, Takashi
Published in Journal of the American Chemical Society (21.06.2006)
Published in Journal of the American Chemical Society (21.06.2006)
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Journal Article
Antidiabetic and Hypolipidemic Effects of a Novel Dual Peroxisome Proliferator-Activated Receptor (PPAR) α/γ Agonist, E3030, in db/db Mice and Beagle Dogs
Kasai, Shunji, Inoue, Takashi, Yoshitomi, Hideki, Hihara, Taro, Matsuura, Fumiyoshi, Harada, Hitoshi, Shinoda, Masanobu, Tanaka, Isao
Published in Journal of Pharmacological Sciences (2008)
Published in Journal of Pharmacological Sciences (2008)
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Journal Article
O3H-4-4 Finding of selective tissue factor/factor VIIa complex inhibitor as a novel anticoagulant with lower bleeding risk
Nagakura Tadashi, Kimiyo Tabata, Kazunobu Kira, Shinsuke Hirota, Clark Richard, Fumiyoshi Matsuura, Hironobu Hisyohi
Published in Journal of Pharmacological Sciences (15.02.2014)
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Published in Journal of Pharmacological Sciences (15.02.2014)
Journal Article
Antidiabetic and Hypolipidemic Effects of a Novel Dual Peroxisome Proliferator-Activated Receptor (PPAR) a/γ Agonist, E3030, in db/db Mice and Beagle Dogs
Shunji Kasai, Takashi Inoue, Hideki Yoshitomi, Taro Hihara, Fumiyoshi Matsuura, Hitoshi Harada, Masanobu Shinoda, Isao Tanaka
Published in Journal of Pharmacological Sciences (2008)
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Published in Journal of Pharmacological Sciences (2008)
Journal Article
Ten-Gram-Scale Total Synthesis of the Anticancer Drug Candidate E7130 to Supply Clinical Trials
Kaburagi, Yosuke, Kira, Kazunobu, Yahata, Kenzo, Iso, Kentaro, Sato, Yuki, Matsuura, Fumiyoshi, Ohashi, Isao, Matsumoto, Yasunobu, Isomura, Minetaka, Sasaki, Takeo, Fukuyama, Takashi, Miyashita, Yusuke, Azuma, Hiroshi, Iida, Daisuke, Ishida, Tasuku, Itano, Wataru, Matsuda, Masaaki, Matsukura, Masayuki, Murai, Norio, Nagao, Satoshi, Seki, Masashi, Yamamoto, Akihiko, Yamamoto, Yuji, Yoneda, Naoki, Watanabe, Yuzo, Kamada, Atsushi, Kayano, Akio, Tagami, Katsuya, Asano, Osamu, Owa, Takashi, Kishi, Yoshito
Published in Organic letters (12.04.2024)
Published in Organic letters (12.04.2024)
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Journal Article
What Does It Take to Develop Structurally Complex Molecules by Total Synthesis? Rapid Process Development and GMP Manufacturing of E7130 Drug Substance for First-in-Human Clinical Study
Sasaki, Takeo, Yahata, Kenzo, Isomura, Minetaka, Ohashi, Isao, Fukuyama, Takashi, Miyashita, Yusuke, Watanabe, Yuzo, Murai, Norio, Matsuda, Masaaki, Kamada, Atsushi, Kaburagi, Yosuke, Kira, Kazunobu, Iso, Kentaro, Sato, Yuki, Matsuura, Fumiyoshi, Matsumoto, Yasunobu, Azuma, Hiroshi, Iida, Daisuke, Ishida, Tasuku, Itano, Wataru, Nagao, Satoshi, Seki, Masashi, Yamamoto, Akihiko, Yamamoto, Yuji, Yoneda, Naoki, Matsukura, Masayuki, Asano, Osamu, Kayano, Akio, Tagami, Katsuya, Owa, Takashi, Kishi, Yoshito
Published in Organic process research & development (21.06.2024)
Published in Organic process research & development (21.06.2024)
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Journal Article
Abstract 4183: Mechanism of action analysis of anti-CAF activity of E7130, a novel tumor-microenvironment ameliorator
Abe, Takanori, Kawano, Satoshi, Ito, Ken, Yahata, Kenzo, Kira, Kazunobu, Akagi, Tsuyoshi, Asano, Makoto, Iso, Kentaro, Sato, Yuki, Matsuura, Fumiyoshi, Ohashi, Isao, Matsumoto, Yasunobu, Isomura, Minetaka, Sasaki, Takeo, Fukuyama, Takashi, Miyashita, Yusuke, Kaburagi, Yosuke, Yokoi, Akira, Asano, Osamu, Owa, Takashi, Kishi, Yoshito
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Journal Article
Abstract 4179: E7130 derived from total synthesis of halichondrin as a novel tumor-microenvironment ameliorator
Kawano, Satoshi, Abe, Takanori, Ito, Ken, Yahata, Kenzo, Kira, Kazunobu, Akagi, Tsuyoshi, Asano, Makoto, Iso, Kentaro, Sato, Yuki, Matsuura, Fumiyoshi, Ohashi, Isao, Matsumoto, Yasunobu, Isomura, Minetaka, Sasaki, Takeo, Fukuyama, Takashi, Miyashita, Yusuke, Kaburagi, Yosuke, Yokoi, Akira, Asano, Osamu, Owa, Takashi, Kishi, Yoshito
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Journal Article
E3024, 3-but-2-ynyl-5-methyl-2-piperazin-1-yl-3,5-dihydro-4H-imidazo [4,5-d]pyridazin-4-one tosylate, is a novel, selective and competitive dipeptidyl peptidase-IV inhibitor
YASUDA, Nobuyuki, NAGAKURA, Tadashi, KIRA, Kazunobu, IKUTA, Hironori, OKADA, Toshimi, SAEKI, Takao, ASANO, Osamu, TANAKA, Isao, INOUE, Takashi, YAMAZAKI, Kazuto, KATSUTANI, Naruo, TAKENAKA, Osamu, CLARK, Richard, MATSUURA, Fumiyoshi, EMORI, Eita, YOSHIKAWA, Seiji
Published in European journal of pharmacology (01.10.2006)
Published in European journal of pharmacology (01.10.2006)
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Journal Article
Selective tissue factor/factor VIIa Inhibitor, ER-410660, and its prodrug, E5539, have anti-venous and anti-arterial thrombotic effects with a low risk of bleeding
Nagakura, Tadashi, Tabata, Kimiyo, Kira, Kazunobu, Hirota, Shinsuke, Clark, Richard, Matsuura, Fumiyoshi, Hiyoshi, Hironobu
Published in Thrombosis research (01.08.2013)
Published in Thrombosis research (01.08.2013)
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Journal Article
Unified Total Synthesis of Pteriatoxins and Their Diastereomers
Matsuura, Fumiyoshi, Peters, René, Anada, Masahiro, Harried, Scott S, Hao, Junliang, Kishi, Yoshito
Published in Journal of the American Chemical Society (14.06.2006)
Published in Journal of the American Chemical Society (14.06.2006)
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