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Komatsu, Shun-ichiro, Kayukawa, Yoko, Miyazaki, Yoko, Kaneko, Akihisa, Ikegami, Hisashi, Ishiguro, Takahiro, Nakamura, Mikiko, Frings, Werner, Ono, Natsuki, Sakata, Kiyoaki, Fujii, Toshihiko, Kishishita, Shohei, Kitazawa, Takehisa, Endo, Mika, Sano, Yuji
Published in Scientific reports (19.07.2022)
Published in Scientific reports (19.07.2022)
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Selective TRK Inhibitor CH7057288 against TRK Fusion-Driven Cancer
Tanaka, Hiroshi, Sase, Hitoshi, Tsukaguchi, Toshiyuki, Hasegawa, Masami, Tanimura, Hiromi, Yoshida, Miyuki, Sakata, Kiyoaki, Fujii, Toshihiko, Tachibana, Yukako, Takanashi, Kenji, Higashida, Atsuko, Hasegawa, Kiyoshi, Ono, Yoshiyuki, Oikawa, Nobuhiro, Mio, Toshiyuki
Published in Molecular cancer therapeutics (01.12.2018)
Published in Molecular cancer therapeutics (01.12.2018)
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ERK Signal Suppression and Sensitivity to CH5183284/Debio 1347, a Selective FGFR Inhibitor
Nakanishi, Yoshito, Mizuno, Hideaki, Sase, Hitoshi, Fujii, Toshihiko, Sakata, Kiyoaki, Akiyama, Nukinori, Aoki, Yuko, Aoki, Masahiro, Ishii, Nobuya
Published in Molecular cancer therapeutics (01.12.2015)
Published in Molecular cancer therapeutics (01.12.2015)
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Enhanced antitumor activity of erlotinib in combination with the Hsp90 inhibitor CH5164840 against non‐small‐cell lung cancer
Ono, Naomi, Yamazaki, Toshikazu, Tsukaguchi, Toshiyuki, Fujii, Toshihiko, Sakata, Kiyoaki, Suda, Atsushi, Tsukuda, Takuo, Mio, Toshiyuki, Ishii, Nobuya, Kondoh, Osamu, Aoki, Yuko
Published in Cancer science (01.10.2013)
Published in Cancer science (01.10.2013)
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Preclinical antitumor activity of the novel heat shock protein 90 inhibitor CH5164840 against human epidermal growth factor receptor 2 (HER2)‐overexpressing cancers
Ono, Naomi, Yamazaki, Toshikazu, Nakanishi, Yoshito, Fujii, Toshihiko, Sakata, Kiyoaki, Tachibana, Yukako, Suda, Atsushi, Hada, Kihito, Miura, Takaaki, Sato, Shigeo, Saitoh, Ryoichi, Nakano, Kohnosuke, Tsukuda, Takuo, Mio, Toshiyuki, Ishii, Nobuya, Kondoh, Osamu, Aoki, Yuko
Published in Cancer science (01.02.2012)
Published in Cancer science (01.02.2012)
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Development of a targeted flip-in system in avian DT40 cells
Kobayashi, Kaori, Fujii, Toshihiko, Asada, Ryuta, Ooka, Masato, Hirota, Kouji
Published in PloS one (23.03.2015)
Published in PloS one (23.03.2015)
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In vitro activity of isavuconazole against 140 reference fungal strains and 165 clinically isolated yeasts from Japan
Yamazaki, Toshikazu, Inagaki, Yukiko, Fujii, Toshihiko, Ohwada, Jun, Tsukazaki, Masao, Umeda, Isao, Kobayashi, Kazuko, Shimma, Nobuo, Page, Malcolm G.P, Arisawa, Mikio
Published in International journal of antimicrobial agents (01.10.2010)
Published in International journal of antimicrobial agents (01.10.2010)
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Involvement of CYP2J2 and CYP4F12 in the Metabolism of Ebastine in Human Intestinal Microsomes
Hashizume, Takanori, Imaoka, Susumu, Mise, Masashi, Terauchi, Yoshiaki, Fujii, Toshihiko, Miyazaki, Hisashi, Kamataki, Tetsuya, Funae, Yoshihiko
Published in The Journal of pharmacology and experimental therapeutics (01.01.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2002)
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Synthesis and biological activities of benzofuran antifungal agents targeting fungal N-myristoyltransferase
Masubuchi, Miyako, Ebiike, Hirosato, Kawasaki, Ken-ichi, Sogabe, Satoshi, Morikami, Kenji, Shiratori, Yasuhiko, Tsujii, Shinji, Fujii, Toshihiko, Sakata, Kiyoaki, Hayase, Michiko, Shindoh, Hidetoshi, Aoki, Yuko, Ohtsuka, Tatsuo, Shimma, Nobuo
Published in Bioorganic & medicinal chemistry (01.10.2003)
Published in Bioorganic & medicinal chemistry (01.10.2003)
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Design and synthesis of novel benzofurans as a new class of antifungal agents targeting fungal N-myristoyltransferase. Part 3
Kawasaki, Ken-ichi, Masubuchi, Miyako, Morikami, Kenji, Sogabe, Satoshi, Aoyama, Tsunehisa, Ebiike, Hirosato, Niizuma, Satoshi, Hayase, Michiko, Fujii, Toshihiko, Sakata, Kiyoaki, Shindoh, Hidetoshi, Shiratori, Yasuhiko, Aoki, Yuko, Ohtsuka, Tatsuo, Shimma, Nobuo
Published in Bioorganic & medicinal chemistry letters (06.01.2003)
Published in Bioorganic & medicinal chemistry letters (06.01.2003)
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Journal Article
Design and synthesis of novel benzofurans as a new class of antifungal agents targeting fungal N-myristoyltransferase. Part 1
MASUBUCHI, Miyako, KAWASAKI, Ken-Ichi, OHTSUKA, Tatsuo, SHIMMA, Nobuo, EBIIKE, Hirosato, IKEDA, Yoshihiko, TSUJII, Shinji, SOGABE, Satoshi, FUJII, Toshihiko, SAKATA, Kiyoaki, SHIRATORI, Yasuhiko, AOKI, Yuko
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
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Neuroimaging of histamine H1‐receptor occupancy in human brain by positron emission tomography (PET): A comparative study of ebastine, a second‐generation antihistamine, and (+)‐chlorpheniramine, a classical antihistamine
Tagawa, Masaaki, Kano, Michiko, Okamura, Nobuyuki, Higuchi, Makoto, Matsuda, Michiaki, Mizuki, Yasuyuki, Arai, Hiroyuki, Iwata, Ren, Fujii, Toshihiko, Komemushi, Sadao, Ido, Tatsuo, Itoh, Masatoshi, Sasaki, Hidetada, Watanabe, Takehiko, Yanai, Kazuhiko
Published in British journal of clinical pharmacology (01.11.2001)
Published in British journal of clinical pharmacology (01.11.2001)
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Conference Proceeding
Uridine diphosphate sugar-selective conjugation of an aldose reductase inhibitor (AS-3201) by UDP-glucuronosyltransferase 2B subfamily in human liver microsomes
Toide, Kenji, Terauchi, Yoshiaki, Fujii, Toshihiko, Yamazaki, Hiroshi, Kamataki, Tetsuya
Published in Biochemical pharmacology (01.04.2004)
Published in Biochemical pharmacology (01.04.2004)
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cDNA Cloning and Expression of a Novel Cytochrome P450 (CYP4F12) from Human Small Intestine
Hashizume, Takanori, Imaoka, Susumu, Hiroi, Toyoko, Terauchi, Yoshiaki, Fujii, Toshihiko, Miyazaki, Hisashi, Kamataki, Tetsuya, Funae, Yoshihiko
Published in Biochemical and biophysical research communications (02.02.2001)
Published in Biochemical and biophysical research communications (02.02.2001)
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