Carbamoyl Pyridone HIV‑1 Integrase Inhibitors. 1. Molecular Design and Establishment of an Advanced Two-Metal Binding Pharmacophore
Kawasuji, Takashi, Johns, Brian A, Yoshida, Hiroshi, Taishi, Teruhiko, Taoda, Yoshiyuki, Murai, Hitoshi, Kiyama, Ryuichi, Fuji, Masahiro, Yoshinaga, Tomokazu, Seki, Takahiro, Kobayashi, Masanori, Sato, Akihiko, Fujiwara, Tamio
Published in Journal of medicinal chemistry (25.10.2012)
Published in Journal of medicinal chemistry (25.10.2012)
Get full text
Journal Article
Highly Selective and Orally Active Inhibitors of Type IV Collagenase (MMP-9 and MMP-2): N-Sulfonylamino Acid Derivatives
Tamura, Yoshinori, Watanabe, Fumihiko, Nakatani, Takuji, Yasui, Ken, Fuji, Masahiro, Komurasaki, Tadafumi, Tsuzuki, Hiroshige, Maekawa, Ryuji, Yoshioka, Takayuki, Kawada, Kenji, Sugita, Kenji, Ohtani, Mitsuaki
Published in Journal of medicinal chemistry (12.02.1998)
Published in Journal of medicinal chemistry (12.02.1998)
Get full text
Journal Article
Carbamoyl Pyridone HIV‑1 Integrase Inhibitors 3. A Diastereomeric Approach to Chiral Nonracemic Tricyclic Ring Systems and the Discovery of Dolutegravir (S/GSK1349572) and (S/GSK1265744)
Johns, Brian A, Kawasuji, Takashi, Weatherhead, Jason G, Taishi, Teruhiko, Temelkoff, David P, Yoshida, Hiroshi, Akiyama, Toshiyuki, Taoda, Yoshiyuki, Murai, Hitoshi, Kiyama, Ryuichi, Fuji, Masahiro, Tanimoto, Norihiko, Jeffrey, Jerry, Foster, Scott A, Yoshinaga, Tomokazu, Seki, Takahiro, Kobayashi, Masanori, Sato, Akihiko, Johnson, Matthew N, Garvey, Edward P, Fujiwara, Tamio
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
Get full text
Journal Article
Total Synthesis of Terprenin, a Highly Potent and Novel Immunoglobulin E Antibody Suppressant
Kawada, Kenji, Arimura, Akinori, Tsuri, Tatsuo, Fuji, Masahiro, Komurasaki, Tadafumi, Yonezawa, Shuji, Kugimiya, Akira, Haga, Nobuhiro, Mitsumori, Susumu, Inagaki, Masanao, Nakatani, Takuji, Tamura, Yoshinori, Takechi, Shozo, Taishi, Teruhiko, Kishino, Junji, Ohtani, Mitsuaki
Published in Angewandte Chemie International Edition (20.04.1998)
Published in Angewandte Chemie International Edition (20.04.1998)
Get full text
Journal Article
Hyponatremic - Hypertensive Syndrome Associated With Renovascular Hypertension: A Case Report
Tetsuou, Yayoi Tsukada, Miyatake, Yoshiko Yamazaki, Tanaka, Kunio, Suzuki, Takeshi, Ohtsu, Fumio, Nagasawa, Koichi, Fuji-i, Masahiro, Tanaka, Shigeo, Iino, Yasuhiko, Tamura, Koichi
Published in Circulation Journal (2002)
Published in Circulation Journal (2002)
Get full text
Journal Article
Carbamoyl Pyridone HIV‑1 Integrase Inhibitors. 2. Bi- and Tricyclic Derivatives Result in Superior Antiviral and Pharmacokinetic Profiles
Kawasuji, Takashi, Johns, Brian A, Yoshida, Hiroshi, Weatherhead, Jason G, Akiyama, Toshiyuki, Taishi, Teruhiko, Taoda, Yoshiyuki, Mikamiyama-Iwata, Minako, Murai, Hitoshi, Kiyama, Ryuichi, Fuji, Masahiro, Tanimoto, Norihiko, Yoshinaga, Tomokazu, Seki, Takahiro, Kobayashi, Masanori, Sato, Akihiko, Garvey, Edward P, Fujiwara, Tamio
Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
Get full text
Journal Article
A platform for designing HIV integrase inhibitors. Part 2: A two-metal binding model as a potential mechanism of HIV integrase inhibitors
Kawasuji, Takashi, Fuji, Masahiro, Yoshinaga, Tomokazu, Sato, Akihiko, Fujiwara, Tamio, Kiyama, Ryuichi
Published in Bioorganic & medicinal chemistry (15.12.2006)
Published in Bioorganic & medicinal chemistry (15.12.2006)
Get full text
Journal Article
Transcriptional activation of survivin through the NF‐κB pathway by human T‐cell leukemia virus type I tax
Kawakami, Hirochika, Tomita, Mariko, Matsuda, Takehiro, Ohta, Takao, Tanaka, Yuetsu, Fujii, Masahiro, Hatano, Masahiko, Tokuhisa, Takeshi, Mori, Naoki
Published in International journal of cancer (20.07.2005)
Published in International journal of cancer (20.07.2005)
Get full text
Journal Article
A Study on Indoor Positioning Based on Attitude and Distance Estimations by Grid Search with Penalty Term
Taki, Fumiya, Fuji, Masahiro
Published in 2021 IEEE 10th Global Conference on Consumer Electronics (GCCE) (12.10.2021)
Published in 2021 IEEE 10th Global Conference on Consumer Electronics (GCCE) (12.10.2021)
Get full text
Conference Proceeding
Human T‐cell leukemia virus type 1 Tax oncoprotein represses the expression of the BCL11B tumor suppressor in T‐cells
Takachi, Takayuki, Takahashi, Masahiko, Takahashi‐Yoshita, Manami, Higuchi, Masaya, Obata, Miki, Mishima, Yukio, Okuda, Shujiro, Tanaka, Yuetsu, Matsuoka, Masao, Saitoh, Akihiko, Green, Patrick L., Fujii, Masahiro
Published in Cancer science (01.04.2015)
Published in Cancer science (01.04.2015)
Get full text
Journal Article
Synthesis and Antiviral Activity of 7-Benzyl-4-hydroxy-1,5-naphthyridin-2(1H)-one HIV Integrase Inhibitors
Boros, Eric E, Edwards, Cynthia E, Foster, Scott A, Fuji, Masahiro, Fujiwara, Tamio, Garvey, Edward P, Golden, Pamela L, Hazen, Richard J, Jeffrey, Jerry L, Johns, Brian A, Kawasuji, Takashi, Kiyama, Ryuichi, Koble, Cecilia S, Kurose, Noriyuki, Miller, Wayne H, Mote, Angela L, Murai, Hitoshi, Sato, Akihiko, Thompson, James B, Woodward, Mark C, Yoshinaga, Tomokazu
Published in Journal of medicinal chemistry (14.05.2009)
Published in Journal of medicinal chemistry (14.05.2009)
Get full text
Journal Article
Preparation of Alkyl-Substituted Indoles in the Benzene Portion. Part 9. Synthesis of (1aS,8bS)-1-tert-Butyloxycarbonyl-8-formyl-1,1a,2,8b-tetrahydroazirino(2',3':3,4)pyrrolo(1,2-a)indole. Model Study for the Enantiospecific Synthesis of Aziridinomitosenes
UTSUNOMIYA, Iwao, FUJI, Masahiro, SATO, Tomohiro, NATSUME, Mitsutaka
Published in Chemical & pharmaceutical bulletin (1993)
Published in Chemical & pharmaceutical bulletin (1993)
Get full text
Journal Article