Action for Increasing Diversity, Market Access, and Capacity in Oncology Registration Trials—Is Africa the Answer? Report From a Satellite Session of the Accelerating Anti-Cancer Agent Development and Validation Workshop
Kizub, Darya, Manner, Cathyryne K., Graef, Katy, Abubakar, Bello, Orem, Jackson, Odedina, Folakemi, Adeyeye, Mojisola Christianah, Nakigudde, Gertrude, Ayalew, Kassa, Kalidas, Chitkala, Lyerly, Herbert Kim, Norman, Thea, Fashoyin-Aje, Lola, Freedman, Jamie, Dent, Jennifer, Cance, Bill, Gralow, Julie
Published in JCO global oncology (01.06.2022)
Published in JCO global oncology (01.06.2022)
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Characterization of 2-(2,6-dichloro-benzyl)-thiazolo[5,4- d]pyrimidin-7-yl]-(4-trifluoromethyl-phenyl)-amine (JNJ-39729209) as a novel TRPV1 antagonist
Maher, Michael P., Bhattacharya, Anindya, Ao, Hong, Swanson, Nadia, Wu, Nyan-Tsz, Freedman, Jamie, Kansagara, Mena, Scott, Brian, Li, Dong H., Eckert, William A., Liu, Yi, Sepassi, Kia, Rizzolio, Michele, Fitzgerald, Anne, Liu, Jing, Branstetter, Bryan J., Rech, Jason C., Lebsack, Alec D., Breitenbucher, J. Guy, Wickenden, Alan D., Chaplan, Sandra R.
Published in European journal of pharmacology (01.08.2011)
Published in European journal of pharmacology (01.08.2011)
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Discovery and synthesis of 6,7,8,9-tetrahydro-5H-pyrimido-[4,5-d]azepines as novel TRPV1 antagonists
HAWRYLUK, Natalie A, MERIT, Jeffrey E, FREEDMAN, Jamie M, SCOTT, Brian P, WICKENDEN, Alan D, CHAPLAN, Sandra R, BREITENBUCHER, J. Guy, LEBSACK, Alec D, BRANSTETTER, Bryan J, HACK, Michael D, SWANSON, Nadia, HONG AO, MAHER, Michael P, BHATTACHARYA, Anindya, QI WANG
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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3-[5-(3,4-Dichloro-phenyl)-1-(4-methoxy-phenyl)-1H-pyrazol-3-yl]-2-m-tolyl-propionate (JNJ-17156516), a Novel, Potent, and Selective Cholecystokinin 1 Receptor Antagonist: In Vitro and in Vivo Pharmacological Comparison with Dexloxiglumide
Morton, Magda F, Barrett, Terrance D, Yan, Wen, Freedman, Jamie M, Lagaud, Guy, Prendergast, Clodagh E, Moreno, Veronica, Pyati, Jayashree, Figueroa, Katherine, Li, Lina, Wu, Xiaodong, Rizzolio, Michele, Breitenbucher, James G, McClure, Kelly, Shankley, Nigel P
Published in The Journal of pharmacology and experimental therapeutics (01.11.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2007)
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Tocilizumab in Patients Hospitalized with Covid-19 Pneumonia
Salama, Carlos, Han, Jian, Yau, Linda, Reiss, William G, Kramer, Benjamin, Neidhart, Jeffrey D, Criner, Gerard J, Kaplan-Lewis, Emma, Baden, Rachel, Pandit, Lavannya, Cameron, Miriam L, Garcia-Diaz, Julia, Chávez, Victoria, Mekebeb-Reuter, Martha, Lima de Menezes, Ferdinando, Shah, Reena, González-Lara, Maria F, Assman, Beverly, Freedman, Jamie, Mohan, Shalini V
Published in New England Journal of Medicine (07.01.2021)
Published in New England Journal of Medicine (07.01.2021)
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Discovery of potent cholecystokinin-2 receptor antagonists: Elucidation of key pharmacophore elements by X-ray crystallographic and NMR conformational analysis
Rosen, Mark D., Hack, Michael D., Allison, Brett D., Phuong, Victor K., Woods, Craig R., Morton, Magda F., Prendergast, Clodagh E., Barrett, Terrance D., Schubert, Carsten, Li, Lina, Wu, Xiaodong, Wu, Jiejun, Freedman, Jamie M., Shankley, Nigel P., Rabinowitz, Michael H.
Published in Bioorganic & medicinal chemistry (01.04.2008)
Published in Bioorganic & medicinal chemistry (01.04.2008)
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Niraparib in patients (pts) with metastatic castration-resistant prostate cancer (mCRPC) and biallelic DNA-repair gene defects (DRD): Correlative measures of tumor response in phase II GALAHAD study
Smith, Matthew Raymond, Fizazi, Karim, Sandhu, Shahneen Kaur, Kelly, William Kevin, Efstathiou, Eleni, Lara, Primo, Yu, Evan Y., George, Daniel J., Chi, Kim N., Saad, Fred, Summa, Jason, Freedman, Jamie M., Mason, Gary, Espina, Byron M., Zhu, Eugene, Ricci, Deborah S., Snyder, Linda A., Simon, Jason S., Cheng, Shinta, Scher, Howard I.
Published in Journal of clinical oncology (20.02.2020)
Published in Journal of clinical oncology (20.02.2020)
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Advancing Inclusive Research: Establishing Collaborative Strategies to Improve Diversity in Clinical Trials
Garrick, Owen, Mesa, Ruben, Ferris, Andrea, Kim, Edward S, Mitchell, Edith, Brawley, Otis W, Carpten, John, Carter, Keith D, Coney, Joseph, Winn, Robert, Monroe, Stephanie, Sandoval, Fabian, Perez, Edith, Williams, Mitzi, Grove, Evan, Highsmith, Quita, Richie, Nicole, Begelman, Susan M, Collins, Asha S, Freedman, Jamie, Gonzales, Melissa S, Wilson, Gerren
Published in Ethnicity & disease (01.01.2022)
Published in Ethnicity & disease (01.01.2022)
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JNJ-26070109 [(R)4-bromo-N-[1-(2,4-difluoro-phenyl)-ethyl]-2-(quinoxaline-5-sulfonylamino)-benzamide]: a novel, potent, and selective cholecystokinin 2 receptor antagonist with good oral bioavailability
Morton, Magda F, Barrett, Terrance D, Freedman, Jamie, Li, Lina, Rizzolio, Michele C, Prendergast, Clodagh E, Wu, Xiaodong, Moreno, Veronica, Pyati, Jayashree, Figueroa, Katherine, Cagnon, Laurence, Lagaud, Guy, Ver Donck, Luc, Ghoos, Etienne, Allison, Brett, Rabinowitz, Michael H, Shankley, Nigel P
Published in The Journal of pharmacology and experimental therapeutics (01.07.2011)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2011)
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Identification and Optimization of Anthranilic Sulfonamides as Novel, Selective Cholecystokinin-2 Receptor Antagonists
Allison, Brett D, Phuong, Victor K, McAtee, Laura C, Rosen, Mark, Morton, Magda, Prendergast, Clodagh, Barrett, Terry, Lagaud, Guy, Freedman, Jamie, Li, Lina, Wu, Xiaodong, Venkatesan, Hariharan, Pippel, Marna, Woods, Craig, Rizzolio, Michèle C, Hack, Michael, Hoey, Kenway, Deng, Xiaohu, King, Christopher, Shankley, Nigel P, Rabinowitz, Michael H
Published in Journal of medicinal chemistry (19.10.2006)
Published in Journal of medicinal chemistry (19.10.2006)
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Discovery and synthesis of 6,7,8,9-tetrahydro-5 H-pyrimido-[4,5- d]azepines as novel TRPV1 antagonists
Hawryluk, Natalie A., Merit, Jeffrey E., Lebsack, Alec D., Branstetter, Bryan J., Hack, Michael D., Swanson, Nadia, Ao, Hong, Maher, Michael P., Bhattacharya, Anindya, Wang, Qi, Freedman, Jamie M., Scott, Brian P., Wickenden, Alan D., Chaplan, Sandra R., Breitenbucher, J. Guy
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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1,2-Diamino-ethane-substituted-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepines as TRPV1 antagonists with improved properties
LEBSACK, Alec D, RECH, Jason C, HONG AO, MAHER, Michael P, HERRMANN, Michelle, FREEDMAN, Jamie, SCOTT, Brian P, LIN LUO, BHATTACHARYA, Anindya, QI WANG, CHAPLAN, Sandra R, WICKENDEN, Alan D, BRANSTETTER, Bryan J, BREITENBUCHER, J. Guy, HAWRYLUK, Natalie A, MERIT, Jeffrey E, ALLISON, Brett, RYNBERG, Raymond, BUMA, Johnathan, RIZZOLIO, Michele, SWANSON, Nadia
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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1,2-Diamino-ethane-substituted-6,7,8,9-tetrahydro-5 H-pyrimido[4,5- d]azepines as TRPV1 antagonists with improved properties
Lebsack, Alec D., Rech, Jason C., Branstetter, Bryan J., Hawryluk, Natalie A., Merit, Jeffrey E., Allison, Brett, Rynberg, Raymond, Buma, Johnathan, Rizzolio, Michele, Swanson, Nadia, Ao, Hong, Maher, Michael P., Herrmann, Michelle, Freedman, Jamie, Scott, Brian P., Luo, Lin, Bhattacharya, Anindya, Wang, Qi, Chaplan, Sandra R., Wickenden, Alan D., Breitenbucher, J. Guy
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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