Stapled α−helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy
Chang, Yong S, Graves, Bradford, Guerlavais, Vincent, Tovar, Christian, Packman, Kathryn, To, Kwong-Him, Olson, Karen A, Kesavan, Kamala, Gangurde, Pranoti, Mukherjee, Aditi, Baker, Theresa, Darlak, Krzysztof, Elkin, Carl, Filipovic, Zoran, Qureshi, Farooq Z, Cai, Hongliang, Berry, Pamela, Feyfant, Eric, Shi, Xiangguo E, Horstick, James, Annis, D Allen, Manning, Anthony M, Fotouhi, Nader, Nash, Huw, Vassilev, Lyubomir T, Sawyer, Tomi K
Published in Proceedings of the National Academy of Sciences - PNAS (03.09.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (03.09.2013)
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Journal Article
The Tuberculosis Drug Accelerator at year 10: what have we learned?
Aldridge, Bree B, Barros-Aguirre, David, Barry, 3rd, Clifton E, Bates, Robert H, Berthel, Steven J, Boshoff, Helena I, Chibale, Kelly, Chu, Xin-Jie, Cooper, Christopher B, Dartois, Véronique, Duncan, Ken, Fotouhi, Nader, Gusovsky, Fabian, Hipskind, Philip A, Kempf, Dale J, Lelièvre, Joël, Lenaerts, Anne J, McNamara, Case W, Mizrahi, Valerie, Nathan, Carl, Olsen, David B, Parish, Tanya, Petrassi, H Michael, Pym, Alexander, Rhee, Kyu Y, Robertson, Gregory T, Rock, Jeremy Michael, Rubin, Eric J, Russell, Betsy, Russell, David G, Sacchettini, James C, Schnappinger, Dirk, Schrimpf, Michael, Upton, Anna M, Warner, Peter, Wyatt, Paul Graham, Yuan, Ying
Published in Nature medicine (01.08.2021)
Published in Nature medicine (01.08.2021)
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Journal Article
In vivo Activation of the p53 Pathway by Small-Molecule Antagonists of MDM2
Vassilev, Lyubomir T., Vu, Binh T., Graves, Bradford, Carvajal, Daisy, Podlaski, Frank, Filipovic, Zoran, Kong, Norman, Kammlott, Ursula, Lukacs, Christine, Klein, Christian, Fotouhi, Nader, Liu, Emily A.
Published in Science (American Association for the Advancement of Science) (06.02.2004)
Published in Science (American Association for the Advancement of Science) (06.02.2004)
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Journal Article
A Novel Tool to Identify Bactericidal Compounds against Vulnerable Targets in Drug-Tolerant M. tuberculosis found in Caseum
Sarathy, Jansy P, Xie, Min, Jones, Richard M, Chang, Adrienne, Osiecki, Paulina, Weiner, Danielle, Tsao, Wen-Shan, Dougher, Maureen, Blanc, Landry, Fotouhi, Nader, Via, Laura E, Barry, 3rd, Clifton E, De Vlaminck, Iwijn, Sherman, David R, Dartois, Véronique A
Published in mBio (25.04.2023)
Published in mBio (25.04.2023)
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Journal Article
The Novel Oxazolidinone TBI-223 Is Effective in Three Preclinical Mouse Models of Methicillin-Resistant Staphylococcus aureus Infection
Gordon, Oren, Dikeman, Dustin A, Ortines, Roger V, Wang, Yu, Youn, Christine, Mumtaz, Mohammed, Orlando, Nicholas, Zhang, Jeffrey, Patel, Aman M, Gough, Ethan, Kaushik, Amit, Nuermberger, Eric L, Upton, Anna M, Fotouhi, Nader, Miller, Lloyd S, Archer, Nathan K
Published in Microbiology spectrum (26.10.2022)
Published in Microbiology spectrum (26.10.2022)
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Journal Article
A Selective Phosphatase of Regenerating Liver Phosphatase Inhibitor Suppresses Tumor Cell Anchorage-Independent Growth by a Novel Mechanism Involving p130Cas Cleavage
DAOUTI, Sherif, LI, Wen-Hui, HONGJIN BIAN, REIDHAAR-OLSON, John F, BLISS, Sarah A, OLIVIER, Andree R, SERGI, Joseph A, FRY, David, DANHO, Waleed, RITLAND, Steve, FOTOUHI, Nader, HEIMBROOK, David, HONG QIAN, HUIFENG NIU, HUANG, Kuo-Sen, HOLMGREN, Janna, LEVIN, Wayne, REIK, Linda, MCGADY, Debra Lucas, GILLESPIE, Paul, PERROTTA, Agostino
Published in Cancer research (Chicago, Ill.) (15.02.2008)
Published in Cancer research (Chicago, Ill.) (15.02.2008)
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Journal Article
The discovery of VLA-4 antagonists
Tilley, Jefferson W, Chen, Li, Sidduri, Achyutharao, Fotouhi, Nader
Published in Current topics in medicinal chemistry (01.01.2004)
Published in Current topics in medicinal chemistry (01.01.2004)
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Journal Article
Contribution of Pretomanid to Novel Regimens Containing Bedaquiline with either Linezolid or Moxifloxacin and Pyrazinamide in Murine Models of Tuberculosis
Xu, Jian, Li, Si-Yang, Almeida, Deepak V, Tasneen, Rokeya, Barnes-Boyle, Kala, Converse, Paul J, Upton, Anna M, Mdluli, Khisimuzi, Fotouhi, Nader, Nuermberger, Eric L
Published in Antimicrobial agents and chemotherapy (01.05.2019)
Published in Antimicrobial agents and chemotherapy (01.05.2019)
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Journal Article
Comparative Efficacy of the Novel Diarylquinoline TBAJ-587 and Bedaquiline against a Resistant Rv0678 Mutant in a Mouse Model of Tuberculosis
Xu, Jian, Converse, Paul J, Upton, Anna M, Mdluli, Khisimuzi, Fotouhi, Nader, Nuermberger, Eric L
Published in Antimicrobial agents and chemotherapy (18.03.2021)
Published in Antimicrobial agents and chemotherapy (18.03.2021)
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Journal Article
Comparative Efficacy of the Novel Diarylquinoline TBAJ-876 and Bedaquiline against a Resistant Rv0678 Mutant in a Mouse Model of Tuberculosis
Almeida, Deepak, Converse, Paul J, Li, Si-Yang, Upton, Anna M, Fotouhi, Nader, Nuermberger, Eric L
Published in Antimicrobial agents and chemotherapy (17.11.2021)
Published in Antimicrobial agents and chemotherapy (17.11.2021)
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Journal Article
Contezolid can replace linezolid in a novel combination with bedaquiline and pretomanid in a murine model of tuberculosis
Almeida, Deepak, Li, Si-Yang, Lee, Jin, Hafkin, Barry, Mdluli, Khisimuzi, Fotouhi, Nader, Nuermberger, Eric L
Published in Antimicrobial agents and chemotherapy (14.12.2023)
Published in Antimicrobial agents and chemotherapy (14.12.2023)
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Journal Article
Combating antimicrobial resistance in malaria, HIV and tuberculosis
Duffey, Maëlle, Shafer, Robert W, Timm, Juliano, Burrows, Jeremy N, Fotouhi, Nader, Cockett, Mark, Leroy, Didier
Published in Nature reviews. Drug discovery (01.06.2024)
Published in Nature reviews. Drug discovery (01.06.2024)
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Journal Article
Next-Generation Diarylquinolines Improve Sterilizing Activity of Regimens with Pretomanid and the Novel Oxazolidinone TBI-223 in a Mouse Tuberculosis Model
Li, Si-Yang, Converse, Paul J, Betoudji, Fabrice, Lee, Jin, Mdluli, Khisimuzi, Upton, Anna, Fotouhi, Nader, Nuermberger, Eric L
Published in Antimicrobial agents and chemotherapy (18.04.2023)
Published in Antimicrobial agents and chemotherapy (18.04.2023)
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Journal Article
Dual mTORC1/mTORC2 Inhibition as a Host-Directed Therapeutic Target in Pathologically Distinct Mouse Models of Tuberculosis
Tasneen, Rokeya, Mortensen, Deborah S, Converse, Paul J, Urbanowski, Michael E, Upton, Anna, Fotouhi, Nader, Nuermberger, Eric, Hawryluk, Natalie
Published in Antimicrobial agents and chemotherapy (17.06.2021)
Published in Antimicrobial agents and chemotherapy (17.06.2021)
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Journal Article
The heme oxygenase-1 metalloporphyrin inhibitor stannsoporfin enhances the bactericidal activity of a novel regimen for multidrug-resistant tuberculosis in a murine model
Ruelas Castillo, Jennie, Neupane, Pranita, Karanika, Styliani, Krug, Stefanie, Quijada, Darla, Garcia, Andrew, Ayeh, Samuel, Yilma, Addis, Costa, Diego L, Sher, Alan, Fotouhi, Nader, Serbina, Natalya, Karakousis, Petros C
Published in Antimicrobial agents and chemotherapy (07.02.2024)
Published in Antimicrobial agents and chemotherapy (07.02.2024)
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