Metal‐Free Activation of C(sp3)–H Bond, and a Practical and Rapid Synthesis of Privileged 1‐Substituted 1,2,3,4‐Tetrahydroisoquinolines
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Published in European journal of organic chemistry (25.09.2017)
Published in European journal of organic chemistry (25.09.2017)
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Metal-Free Activation of a C(sp)−H Bond of Aryl Acetylenes
Rout, Laxmidhar, Parida, Bibhuti Bhusan, Florent, Jean-Claude, Johannes, Ludger, Choudhury, Santosh Kumar, Phaomei, Ganngam, Scanlon, Joe, Bertounesque, Emmanuel
Published in Chemistry : a European journal (10.10.2016)
Published in Chemistry : a European journal (10.10.2016)
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Palladium-Catalyzed Direct Arylation of Polysubstituted Benzofurans
Carrër, Amandine, Brinet, Dimitri, Florent, Jean-Claude, Rousselle, Patricia, Bertounesque, Emmanuel
Published in Journal of organic chemistry (03.02.2012)
Published in Journal of organic chemistry (03.02.2012)
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2nd PSL Chemical Biology Symposium (2019): At the Crossroads of Chemistry and Biology
Lucchino, Marco, Billet, Anne, Versini, Antoine, Bavireddi, Harikrishna, Dasari, Bhanu‐Das, Debieu, Sylvain, Colombeau, Ludovic, Cañeque, Tatiana, Wagner, Alain, Masson, Géraldine, Taran, Frédéric, Karoyan, Philippe, Delepierre, Muriel, Gaillet, Christine, Houdusse, Anne, Britton, Sébastien, Schmidt, Frédéric, Florent, Jean‐Claude, Belmont, Philippe, Monchaud, David, Cossy, Janine, Thomas, Christophe, Gautier, Arnaud, Johannes, Ludger, Rodriguez, Raphaël
Published in Chembiochem : a European journal of chemical biology (01.04.2019)
Published in Chembiochem : a European journal of chemical biology (01.04.2019)
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New potent dual inhibitors of CK2 and Pim kinases: discovery and structural insights
López-Ramos, Miriam, Prudent, Renaud, Moucadel, Virginie, Sautel, Céline F, Barette, Caroline, Lafanechère, Laurence, Mouawad, Liliane, Grierson, David, Schmidt, Frédéric, Florent, Jean-Claude, Filippakopoulos, Panagis, Bullock, Alex N, Knapp, Stefan, Reiser, Jean-Baptiste, Cochet, Claude
Published in The FASEB journal (01.09.2010)
Published in The FASEB journal (01.09.2010)
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Pharmacological Inhibition of LIM Kinase Stabilizes Microtubules and Inhibits Neoplastic Growth
PRUDENT, Renaud, VASSAL-STERMANN, Emilie, VALDAMERI, Glaucio, HONORE, Stéphane, ACI-SECHE, Samia, GRIERSON, David, ANTONIPILLAI, Juliana, RONG LI, DI PIETRO, Attilio, DUMONTET, Charles, BRAGUER, Diane, FLORENT, Jean-Claude, NGUYEN, Chi-Hung, KNAPP, Stefan, BERNARD, Ora, LAFANECHERE, Laurence, PILLET, Catherine, MARTINEZ, Anne, PRUNIER, Chloe, BARETTE, Caroline, SOLEILHAC, Emmanuelle, FILHOL, Odile, BEGHIN, Anne
Published in Cancer research (Chicago, Ill.) (01.09.2012)
Published in Cancer research (Chicago, Ill.) (01.09.2012)
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Carbohydrate Conformation and Lipid Condensation in Monolayers Containing Glycosphingolipid Gb3: Influence of Acyl Chain Structure
Watkins, Erik B., Gao, Haifei, Dennison, Andrew J.C., Chopin, Nathalie, Struth, Bernd, Arnold, Thomas, Florent, Jean-Claude, Johannes, Ludger
Published in Biophysical journal (02.09.2014)
Published in Biophysical journal (02.09.2014)
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Selective Palladium-Catalyzed Direct Arylation of Furo[3,2-b]pyridines
Carrër, Amandine, Rousselle, Patricia, Florent, Jean-Claude, Bertounesque, Emmanuel
Published in Advanced synthesis & catalysis (08.10.2012)
Published in Advanced synthesis & catalysis (08.10.2012)
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Shiga Toxin-Mediated Retrograde Delivery of a Topoisomerase I Inhibitor Prodrug
El Alaoui, Abdessamad, Schmidt, Frédéric, Amessou, Mohamed, Sarr, Marianne, Decaudin, Didier, Florent, Jean-Claude, Johannes, Ludger
Published in Angewandte Chemie (International ed.) (01.01.2007)
Published in Angewandte Chemie (International ed.) (01.01.2007)
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Azaindole derivatives are inhibitors of microtubule dynamics, with anti‐cancer and anti‐angiogenic activities
Prudent, Renaud, Vassal‐Stermann, Émilie, Nguyen, Chi‐Hung, Mollaret, Marjorie, Viallet, Jean, Desroches‐Castan, Agnès, Martinez, Anne, Barette, Caroline, Pillet, Catherine, Valdameri, Glaucio, Soleilhac, Emmanuelle, Di Pietro, Attilio, Feige, Jean‐Jacques, Billaud, Marc, Florent, Jean‐Claude, Lafanechère, Laurence
Published in British journal of pharmacology (01.02.2013)
Published in British journal of pharmacology (01.02.2013)
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SNAP‐tag Based Proteomics Approach for the Study of the Retrograde Route
Shi, Getao, Azoulay, Michel, Dingli, Florent, Lamaze, Christophe, Loew, Damarys, Florent, Jean‐Claude, Johannes, Ludger
Published in Traffic (Copenhagen, Denmark) (01.07.2012)
Published in Traffic (Copenhagen, Denmark) (01.07.2012)
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Easy Access to Pyranoacridines, Pyranoxanthenes, and Arylchromenes Through a Domino Reaction
Commandeur, Claude, Florent, Jean-Claude, Rousselle, Patricia, Bertounesque, Emmanuel
Published in European Journal of Organic Chemistry (01.03.2011)
Published in European Journal of Organic Chemistry (01.03.2011)
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Synthesis and Structure-Activity Relationships of Constrained Heterocyclic Analogues of Combretastatin A4
Arthuis, Martin, Pontikis, Renée, Chabot, Guy G., Seguin, Johanne, Quentin, Lionel, Bourg, Stéphane, Morin-Allory, Luc, Florent, Jean-Claude
Published in ChemMedChem (05.09.2011)
Published in ChemMedChem (05.09.2011)
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Mechanism of Shiga Toxin Clustering on Membranes
Pezeshkian, Weria, Gao, Haifei, Arumugam, Senthil, Becken, Ulrike, Bassereau, Patricia, Florent, Jean-Claude, Ipsen, John Hjort, Johannes, Ludger, Shillcock, Julian C
Published in ACS nano (24.01.2017)
Published in ACS nano (24.01.2017)
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Shiga Toxin Induces Lipid Compression: A Mechanism for Generating Membrane Curvature
Watkins, Erik B, Majewski, Jaroslaw, Chi, Eva Y, Gao, Haifei, Florent, Jean-Claude, Johannes, Ludger
Published in Nano letters (09.10.2019)
Published in Nano letters (09.10.2019)
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Expanding the chemical diversity of CK2 inhibitors
Prudent, Renaud, Moucadel, Virginie, López-Ramos, Miriam, Aci, Samia, Laudet, Beatrice, Mouawad, Liliane, Barette, Caroline, Einhorn, Jacques, Einhorn, Cathy, Denis, Jean-Noel, Bisson, Gilles, Schmidt, Frédéric, Roy, Sylvaine, Lafanechere, Laurence, Florent, Jean-Claude, Cochet, Claude
Published in Molecular and cellular biochemistry (01.09.2008)
Published in Molecular and cellular biochemistry (01.09.2008)
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Synthesis and biological evaluation of vinylogous combretastatin A-4 derivatives
Kaffy, J, Pontikis, RE, Florent, JC, Monneret, C
Published in Organic & biomolecular chemistry (21.07.2005)
Published in Organic & biomolecular chemistry (21.07.2005)
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Chemistry-based protein modification strategy for endocytic pathway analysis
Christiano, Romain, Amessou, Mohamed, Shi, Getao, Azoulay, Michel, Blanpain, Annick, Drobecq, Hervé, Melnyk, Oleg, Florent, Jean-Claude, Johannes, Ludger
Published in Biology of the cell (01.06.2010)
Published in Biology of the cell (01.06.2010)
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Synthesis and Properties of a Mitochondrial Peripheral Benzodiazepine Receptor Conjugate
El Alaoui, Abdessamad, Schmidt, Frédéric, Sarr, Marianne, Decaudin, Didier, Florent, Jean-Claude, Johannes, Ludger
Published in ChemMedChem (17.11.2008)
Published in ChemMedChem (17.11.2008)
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