Discovery and development of Janus kinase (JAK) inhibitors for inflammatory diseases
Clark, James D, Flanagan, Mark E, Telliez, Jean-Baptiste
Published in Journal of medicinal chemistry (26.06.2014)
Published in Journal of medicinal chemistry (26.06.2014)
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Chemical and Computational Methods for the Characterization of Covalent Reactive Groups for the Prospective Design of Irreversible Inhibitors
Flanagan, Mark E, Abramite, Joseph A, Anderson, Dennis P, Aulabaugh, Ann, Dahal, Upendra P, Gilbert, Adam M, Li, Chao, Montgomery, Justin, Oppenheimer, Stacey R, Ryder, Tim, Schuff, Brandon P, Uccello, Daniel P, Walker, Gregory S, Wu, Yan, Brown, Matthew F, Chen, Jinshan M, Hayward, Matthew M, Noe, Mark C, Obach, R. Scott, Philippe, Laurence, Shanmugasundaram, Veerabahu, Shapiro, Michael J, Starr, Jeremy, Stroh, Justin, Che, Ye
Published in Journal of medicinal chemistry (11.12.2014)
Published in Journal of medicinal chemistry (11.12.2014)
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Discovery of CP-690,550: A Potent and Selective Janus Kinase (JAK) Inhibitor for the Treatment of Autoimmune Diseases and Organ Transplant Rejection
Flanagan, Mark E, Blumenkopf, Todd A, Brissette, William H, Brown, Matthew F, Casavant, Jeffrey M, Shang-Poa, Chang, Doty, Jonathan L, Elliott, Eileen A, Fisher, Michael B, Hines, Michael, Kent, Craig, Kudlacz, Elizabeth M, Lillie, Brett M, Magnuson, Kelly S, McCurdy, Sandra P, Munchhof, Michael J, Perry, Bret D, Sawyer, Perry S, Strelevitz, Timothy J, Subramanyam, Chakrapani, Sun, Jianmin, Whipple, David A, Changelian, Paul S
Published in Journal of medicinal chemistry (23.12.2010)
Published in Journal of medicinal chemistry (23.12.2010)
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Toward the assembly and characterization of an encoded library hit confirmation platform: Bead-Assisted Ligand Isolation Mass Spectrometry (BALI-MS)
Ratnayake, Anokha S., Flanagan, Mark E., Foley, Timothy L., Hultgren, Scott L., Bellenger, Justin, Montgomery, Justin I., Lall, Manjinder S., Liu, Bo, Ryder, Tim, Kölmel, Dominik K., Shavnya, Andre, Feng, Xidong, Lefker, Bruce, Byrnes, Laura J., Sahasrabudhe, Parag V., Farley, Kathleen A., Chen, Shi, Wan, Jinqiao
Published in Bioorganic & medicinal chemistry (01.07.2021)
Published in Bioorganic & medicinal chemistry (01.07.2021)
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Non-traditional antibacterial screening approaches for the identification of novel inhibitors of the glyoxylate shunt in gram-negative pathogens
Fahnoe, Kelly C, Flanagan, Mark E, Gibson, Glenn, Shanmugasundaram, Veerabahu, Che, Ye, Tomaras, Andrew P
Published in PloS one (11.12.2012)
Published in PloS one (11.12.2012)
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Selecting Approaches for Hit Identification and Increasing Options by Building the Efficient Discovery of Actionable Chemical Matter from DNA-Encoded Libraries
Foley, Timothy L., Burchett, Woodrow, Chen, Qiuxia, Flanagan, Mark E., Kapinos, Brendon, Li, Xianyang, Montgomery, Justin I., Ratnayake, Anokha S., Zhu, Hongyao, Peakman, Marie-Claire
Published in SLAS discovery (01.02.2021)
Published in SLAS discovery (01.02.2021)
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The specificity of JAK3 kinase inhibitors
Changelian, Paul S., Moshinsky, Deborah, Kuhn, Cyrille F., Flanagan, Mark E., Munchhof, Michael J., Harris, Thomas M., Whipple, David A., Doty, Jonathan L., Sun, Jianmin, Kent, Craig R., Magnuson, Kelly S., Perregaux, David G., Sawyer, Perry S., Kudlacz, Elizabeth M.
Published in Blood (15.02.2008)
Published in Blood (15.02.2008)
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Designing DNA Encoded Libraries of Diverse Products in a Focused Property Space
Zhu, Hongyao, Flanagan, Mark E, Stanton, Robert V
Published in Journal of chemical information and modeling (25.11.2019)
Published in Journal of chemical information and modeling (25.11.2019)
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Photoredox cross-electrophile coupling in DNA-encoded chemistry
Kölmel, Dominik K., Ratnayake, Anokha S., Flanagan, Mark E.
Published in Biochemical and biophysical research communications (03.12.2020)
Published in Biochemical and biophysical research communications (03.12.2020)
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Employing Photoredox Catalysis for DNA‐Encoded Chemistry: Decarboxylative Alkylation of α‐Amino Acids
Kölmel, Dominik K., Loach, Richard P., Knauber, Thomas, Flanagan, Mark E.
Published in ChemMedChem (22.10.2018)
Published in ChemMedChem (22.10.2018)
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Photocatalytic [2 + 2] Cycloaddition in DNA-Encoded Chemistry
Kölmel, Dominik K, Ratnayake, Anokha S, Flanagan, Mark E, Tsai, Mei-Hsuan, Duan, Cong, Song, Chao
Published in Organic letters (17.04.2020)
Published in Organic letters (17.04.2020)
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On-DNA Decarboxylative Arylation: Merging Photoredox with Nickel Catalysis in Water
Kölmel, Dominik K, Meng, Jiang, Tsai, Mei-Hsuan, Que, Jiamin, Loach, Richard P, Knauber, Thomas, Wan, Jinqiao, Flanagan, Mark E
Published in ACS combinatorial science (12.08.2019)
Published in ACS combinatorial science (12.08.2019)
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Expanding Reactivity in DNA-Encoded Library Synthesis via Reversible Binding of DNA to an Inert Quaternary Ammonium Support
Flood, Dillon T, Asai, Shota, Zhang, Xuejing, Wang, Jie, Yoon, Leonard, Adams, Zoë C, Dillingham, Blythe C, Sanchez, Brittany B, Vantourout, Julien C, Flanagan, Mark E, Piotrowski, David W, Richardson, Paul, Green, Samantha A, Shenvi, Ryan A, Chen, Jason S, Baran, Phil S, Dawson, Philip E
Published in Journal of the American Chemical Society (26.06.2019)
Published in Journal of the American Chemical Society (26.06.2019)
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Identification of N‑{cis-3-[Methyl(7H‑pyrrolo[2,3‑d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide (PF-04965842): A Selective JAK1 Clinical Candidate for the Treatment of Autoimmune Diseases
Vazquez, Michael L, Kaila, Neelu, Strohbach, Joseph W, Trzupek, John D, Brown, Matthew F, Flanagan, Mark E, Mitton-Fry, Mark J, Johnson, Timothy A, TenBrink, Ruth E, Arnold, Eric P, Basak, Arindrajit, Heasley, Steven E, Kwon, Soojin, Langille, Jonathan, Parikh, Mihir D, Griffin, Sarah H, Casavant, Jeffrey M, Duclos, Brian A, Fenwick, Ashley E, Harris, Thomas M, Han, Seungil, Caspers, Nicole, Dowty, Martin E, Yang, Xin, Banker, Mary Ellen, Hegen, Martin, Symanowicz, Peter T, Li, Li, Wang, Lu, Lin, Tsung H, Jussif, Jason, Clark, James D, Telliez, Jean-Baptiste, Robinson, Ralph P, Unwalla, Ray
Published in Journal of medicinal chemistry (08.02.2018)
Published in Journal of medicinal chemistry (08.02.2018)
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Merging C(sp)-H activation with DNA-encoding
Fan, Zhoulong, Zhao, Shuai, Liu, Tao, Shen, Peng-Xiang, Cui, Zi-Ning, Zhuang, Zhe, Shao, Qian, Chen, Jason S, Ratnayake, Anokha S, Flanagan, Mark E, Kölmel, Dominik K, Piotrowski, David W, Richardson, Paul, Yu, Jin-Quan
Published in Chemical science (Cambridge) (07.12.2020)
Published in Chemical science (Cambridge) (07.12.2020)
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RASS‐Enabled S/P−C and S−N Bond Formation for DEL Synthesis
Flood, Dillon T., Zhang, Xuejing, Fu, Xiang, Zhao, Zhenxiang, Asai, Shota, Sanchez, Brittany B., Sturgell, Emily J., Vantourout, Julien C., Richardson, Paul, Flanagan, Mark E., Piotrowski, David W., Kölmel, Dominik K., Wan, Jinqiao, Tsai, Mei‐Hsuan, Chen, Jason S., Baran, Phil S., Dawson, Philip E.
Published in Angewandte Chemie International Edition (04.05.2020)
Published in Angewandte Chemie International Edition (04.05.2020)
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A Solution Phase Platform to Characterize Chemical Reaction Compatibility with DNA-Encoded Chemical Library Synthesis
Ratnayake, Anokha S, Flanagan, Mark E, Foley, Timothy L, Smith, Justin D, Johnson, Jillian G, Bellenger, Justin, Montgomery, Justin I, Paegel, Brian M
Published in ACS combinatorial science (14.10.2019)
Published in ACS combinatorial science (14.10.2019)
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Ultra-High-Throughput Acoustic Droplet Ejection-Open Port Interface-Mass Spectrometry for Parallel Medicinal Chemistry
DiRico, Kenneth J, Hua, Wenyi, Liu, Chang, Tucker, Joseph W, Ratnayake, Anokha S, Flanagan, Mark E, Troutman, Matthew D, Noe, Mark C, Zhang, Hui
Published in ACS medicinal chemistry letters (11.06.2020)
Published in ACS medicinal chemistry letters (11.06.2020)
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Chiral Sulfoxide-Induced Single Turn Peptide α-Helicity
Zhang, Qingzhou, Jiang, Fan, Zhao, Bingchuan, Lin, Huacan, Tian, Yuan, Xie, Mingsheng, Bai, Guoyun, Gilbert, Adam M, Goetz, Gilles H, Liras, Spiros, Mathiowetz, Alan A, Price, David A, Song, Kun, Tu, Meihua, Wu, Yujie, Wang, Tao, Flanagan, Mark E, Wu, Yun-Dong, Li, Zigang
Published in Scientific reports (09.12.2016)
Published in Scientific reports (09.12.2016)
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