Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum—The η-carbonic anhydrases
Del Prete, Sonia, Vullo, Daniela, Fisher, Gillian M., Andrews, Katherine T., Poulsen, Sally-Ann, Capasso, Clemente, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry letters (15.09.2014)
Published in Bioorganic & medicinal chemistry letters (15.09.2014)
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Isolation and In Vitro and In Vivo Activity of Secondary Metabolites from Clerodendrum polycephalum Baker against Plasmodium Malaria Parasites
Tamuli, Roktima, Nguyen, Thanh, Macdonald, Jacinta R., Pierens, Gregory K., Fisher, Gillian M., Andrews, Katherine T., Adewoyin, Francis B., Omisore, Nusrat O., Odaibo, Alexander B., Feng, Yunjiang
Published in Journal of natural products (Washington, D.C.) (22.12.2023)
Published in Journal of natural products (Washington, D.C.) (22.12.2023)
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Sulfonamide inhibition studies of the η-class carbonic anhydrase from the malaria pathogen Plasmodium falciparum
Vullo, Daniela, Del Prete, Sonia, Fisher, Gillian M., Andrews, Katherine T., Poulsen, Sally-Ann, Capasso, Clemente, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (01.02.2015)
Published in Bioorganic & medicinal chemistry (01.02.2015)
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Journal Article
Discovery of 1,3,4-oxadiazoles with slow-action activity against Plasmodium falciparum malaria parasites
Andrews, Katherine T., Fisher, Gillian M., Firmin, Meaghan, Liepa, Andris J., Wilson, Tony, Gardiner, James, Mohri, Yacine, Debele, Emmanuel, Rai, Anjana, Davey, Andrew K., Masurier, Antoine, Delion, Alix, Mouratidis, Alexandros A., Hutt, Oliver E., Forsyth, Craig M., Burrows, Jeremy N., Ryan, John H., Riches, Andrew G., Skinner-Adams, Tina S.
Published in European journal of medicinal chemistry (15.11.2024)
Published in European journal of medicinal chemistry (15.11.2024)
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Journal Article
Activity of alkoxyamide-based histone deacetylase inhibitors against Plasmodium falciparum malaria parasites
Dawood, Wisam A., Fisher, Gillian M., Kinnen, Franziska J.M., Anzenhofer, Christian, Skinner-Adams, Tina, Alves Avelar, Leandro, Asfaha, Yodita, Kurz, Thomas, Andrews, Katherine T.
Published in Experimental parasitology (01.03.2024)
Published in Experimental parasitology (01.03.2024)
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Journal Article
Antimalarial activity of compounds comprising a primary benzene sulfonamide fragment
Andrews, Katherine T., Fisher, Gillian M., Sumanadasa, Subathdrage D.M., Skinner-Adams, Tina, Moeker, Janina, Lopez, Marie, Poulsen, Sally-Ann
Published in Bioorganic & medicinal chemistry letters (15.11.2013)
Published in Bioorganic & medicinal chemistry letters (15.11.2013)
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Journal Article
An ELISA method to assess HDAC inhibitor-induced alterations to P. falciparum histone lysine acetylation
Hesping, Eva, Skinner-Adams, Tina S., Fisher, Gillian M., Kurz, Thomas, Andrews, Katherine T.
Published in International journal for parasitology -- drugs and drug resistance (01.12.2020)
Published in International journal for parasitology -- drugs and drug resistance (01.12.2020)
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Journal Article
Deguelin exerts potent nematocidal activity via the mitochondrial respiratory chain
Preston, Sarah, Korhonen, Pasi K, Mouchiroud, Laurent, Cornaglia, Matteo, McGee, Sean L, Young, Neil D, Davis, Rohan A, Crawford, Simon, Nowell, Cameron, Ansell, Brendan R E, Fisher, Gillian M, Andrews, Katherine T, Chang, Bill C H, Gijs, Martin A M, Sternberg, Paul W, Auwerx, Johan, Baell, Jonathan, Hofmann, Andreas, Jabbar, Abdul, Gasser, Robin B
Published in The FASEB journal (01.10.2017)
Published in The FASEB journal (01.10.2017)
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Journal Article
Defining the targets of antiparasitic compounds
Skinner-Adams, Tina S., Sumanadasa, Subathdrage D.M., Fisher, Gillian M., Davis, Rohan A., Doolan, Denise L., Andrews, Katherine T.
Published in Drug discovery today (01.05.2016)
Published in Drug discovery today (01.05.2016)
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Journal Article
The Key Glycolytic Enzyme Phosphofructokinase Is Involved in Resistance to Antiplasmodial Glycosides
Fisher, Gillian M, Cobbold, Simon A, Jezewski, Andrew, Carpenter, Emma F, Arnold, Megan, Cowell, Annie N, Tjhin, Erick T, Saliba, Kevin J, Skinner-Adams, Tina S, Lee, Marcus C S, Odom John, Audrey, Winzeler, Elizabeth A, McConville, Malcolm J, Poulsen, Sally-Ann, Andrews, Katherine T
Published in mBio (08.12.2020)
Published in mBio (08.12.2020)
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Journal Article
Histone deacetylase inhibitor AR-42 and achiral analogues kill malaria parasites in vitro and in mice
Chua, Ming Jang, Tng, Jiahui, Hesping, Eva, Fisher, Gillian M., Goodman, Christopher D., Skinner-Adams, Tina, Do, Darren, Lucke, Andrew J., Reid, Robert C., Fairlie, David P., Andrews, Katherine T.
Published in International journal for parasitology -- drugs and drug resistance (01.12.2021)
Published in International journal for parasitology -- drugs and drug resistance (01.12.2021)
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Journal Article
Adaptation of the [3H]Hypoxanthine Uptake Assay for In Vitro-Cultured Plasmodium knowlesi Malaria Parasites
Arnold, Megan S J, Engel, Jessica A, Chua, Ming Jang, Fisher, Gillian M, Skinner-Adams, Tina S, Andrews, Katherine T
Published in Antimicrobial agents and chemotherapy (01.07.2016)
Published in Antimicrobial agents and chemotherapy (01.07.2016)
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Assessing the anthelmintic activity of pyrazole-5-carboxamide derivatives against Haemonchus contortus
Jiao, Yaqing, Preston, Sarah, Song, Hongjian, Jabbar, Abdul, Liu, Yuxiu, Baell, Jonathan, Hofmann, Andreas, Hutchinson, Dana, Wang, Tao, Koehler, Anson V, Fisher, Gillian M, Andrews, Katherine T, Laleu, Benoît, Palmer, Michael J, Burrows, Jeremy N, Wells, Timothy N C, Wang, Qingmin, Gasser, Robin B
Published in Parasites & vectors (31.05.2017)
Published in Parasites & vectors (31.05.2017)
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QSAR Classification Models for Prediction of Hydroxamate Histone Deacetylase Inhibitor Activity against Malaria Parasites
Hesping, Eva, Chua, Ming Jang, Pflieger, Marc, Qian, Yunan, Dong, Lilong, Bachu, Prabhakar, Liu, Ligong, Kurz, Thomas, Fisher, Gillian M, Skinner-Adams, Tina S, Reid, Robert C, Fairlie, David P, Andrews, Katherine T, Gorse, Alain-Dominique J.P
Published in ACS infectious diseases (14.01.2022)
Published in ACS infectious diseases (14.01.2022)
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Investigating the antiplasmodial activity of primary sulfonamide compounds identified in open source malaria data
Fisher, Gillian M., Bua, Silvia, Del Prete, Sonia, Arnold, Megan S.J., Capasso, Clemente, Supuran, Claudiu T., Andrews, Katherine T., Poulsen, Sally-Ann
Published in International journal for parasitology -- drugs and drug resistance (01.04.2017)
Published in International journal for parasitology -- drugs and drug resistance (01.04.2017)
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Journal Article
Cyclization-blocked proguanil as a strategy to improve the antimalarial activity of atovaquone
Skinner-Adams, Tina S., Fisher, Gillian M., Riches, Andrew G., Hutt, Oliver E., Jarvis, Karen E., Wilson, Tony, von Itzstein, Mark, Chopra, Pradeep, Antonova-Koch, Yevgeniya, Meister, Stephan, Winzeler, Elizabeth A., Clarke, Mary, Fidock, David A., Burrows, Jeremy N., Ryan, John H., Andrews, Katherine T.
Published in Communications biology (03.05.2019)
Published in Communications biology (03.05.2019)
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