The European Lead Factory: Results from a decade of collaborative, public–private, drug discovery programs
van Vlijmen, Herman, Pannifer, Andrew D., Cochrane, Phil, Basting, Daniel, Li, Volkhart M, Engkvist, Ola, Ortholand, Jean-Yves, Wagener, Markus, Duffy, James, Finsinger, Dirk, Davis, Jeremy, van Helden, Steven P., de Vlieger, Jon S.B.
Published in Drug discovery today (01.03.2024)
Published in Drug discovery today (01.03.2024)
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The European Federation for Medicinal Chemistry (EFMC) Best Practice Initiative: Validating Chemical Probes
Quancard, Jean, Cox, Brian, Finsinger, Dirk, Guéret, Stéphanie M., Hartung, Ingo V., Koolman, Hannes F., Messinger, Josef, Sbardella, Gianluca, Laufer, Stefan
Published in ChemMedChem (15.12.2020)
Published in ChemMedChem (15.12.2020)
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The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Phenotypic Drug Discovery
Quancard, Jean, Bach, Anders, Cox, Brian, Craft, Russell, Finsinger, Dirk, Guéret, Stéphanie M., Hartung, Ingo V., Laufer, Stefan, Messinger, Josef, Sbardella, Gianluca, Koolman, Hannes F.
Published in ChemMedChem (07.06.2021)
Published in ChemMedChem (07.06.2021)
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IMI European Lead Factory - democratizing access to high-throughput screening
Jones, Philip S, Boucharens, Sylviane, McElroy, Stuart P, Morrison, Angus, Honarnejad, Saman, van Boeckel, Stan, van den Hurk, Helma, Basting, Daniel, Hüser, Jörg, Jaroch, Stefan, Ottow, Eckhard, Benningshof, Jorg, Folmer, Rutger H A, Leemhuis, Frank, Kramer-Verhulst, Patricia M, Nies, Vera J M, Orrling, Kristina M, Rijnders, Ton, Pfander, Claudia, Engkvist, Ola, Pairaudeau, Garry, Simpson, Peter B, Ortholand, Jean-Yves, Roche, Didier, Dömling, Alexander, Kühnert, Sven M, Roevens, Peter W M, van Vlijmen, Herman, van Wanrooij, Eva J A, Verbruggen, Christophe, Nussbaumer, Peter, Ovaa, Huib, van der Stelt, Mario, Simonsen, Klaus Baek, Tagmose, Lena, Waldmann, Herbert, Duffy, James, Finsinger, Dirk, Jurzak, Mirek, Burgess-Brown, Nicola A, Lee, Wen H, Rutjes, Floris P J T, Haag, Hubert, Kallus, Christopher, Mors, Hartmut, Dorval, Thierry, Lesur, Brigitte, Ramon Olayo, Fernando, Hamza, Daniel, Jones, Geraint, Pearce, Christopher, Piechot, Alexander, Tzalis, Dimitrios, Clausen, Mads H, Davis, Jeremy, Derouane, Daphné, Vermeiren, Céline, Kaiser, Markus, Stockman, Robert A, Barrault, Denise V, Pannifer, Andrew D, Swedlow, Jason R, Nelson, Adam S, Orru, Romano V A, Ruijter, Eelco, van Helden, Steven P, Li, Volkhart M, Vries, Ton, de Vlieger, Jon S B
Published in Nature reviews. Drug discovery (01.04.2022)
Published in Nature reviews. Drug discovery (01.04.2022)
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The discovery and optimization of hexahydro-2H-pyrano[3,2-c]quinolines (HHPQs) as potent and selective inhibitors of the mitotic kinesin-5
SCHIEMANN, Kai, FINSINGER, Dirk, ZENKE, Frank, AMENDT, Christiane, KNÖCHEL, Thorsten, BRUGE, David, BUCHSTALLER, Hans-Peter, EMDE, Ulrich, STÄHLE, Wolfgang, ANZALI, Soheila
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
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Discovery of novel 7-azaindoles as PDK1 inhibitors
Wucherer-Plietker, Margarita, Merkul, Eugen, Müller, Thomas J.J., Esdar, Christina, Knöchel, Thorsten, Heinrich, Timo, Buchstaller, Hans-Peter, Greiner, Hartmut, Dorsch, Dieter, Finsinger, Dirk, Calderini, Michel, Bruge, David, Grädler, Ulrich
Published in Bioorganic & medicinal chemistry letters (01.07.2016)
Published in Bioorganic & medicinal chemistry letters (01.07.2016)
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Design and synthesis of isoquinolines and benzimidazoles as RAF kinase inhibitors
Buchstaller, Hans-Peter, Burgdorf, Lars, Finsinger, Dirk, Stieber, Frank, Sirrenberg, Christian, Amendt, Christiane, Grell, Matthias, Zenke, Frank, Krier, Mireille
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
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Surface Coating with Cyclic RGD Peptides Stimulates Osteoblast Adhesion and Proliferation as well as Bone Formation
Kantlehner, Martin, Schaffner, Patricia, Finsinger, Dirk, Meyer, Jörg, Jonczyk, Alfred, Diefenbach, Beate, Nies, Berthold, Hölzemann, Günter, Goodman, Simon L., Kessler, Horst
Published in Chembiochem : a European journal of chemical biology (18.08.2000)
Published in Chembiochem : a European journal of chemical biology (18.08.2000)
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PYRROLOPYRIDINYL-PYRIMIDIN-2-YL-AMIN-DERIVATE
DAVID BRUGE, FINSINGER DIRK, ULRICH GRAEDLER, DIETER DORSCH, CHRISTINA ESDAR, MARGARITA WUCHERER-PLIETKER
Year of Publication 25.12.2014
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Year of Publication 25.12.2014
Patent
The discovery and optimization of hexahydro-2 H-pyrano[3,2- c]quinolines (HHPQs) as potent and selective inhibitors of the mitotic kinesin-5
Schiemann, Kai, Finsinger, Dirk, Zenke, Frank, Amendt, Christiane, Knöchel, Thorsten, Bruge, David, Buchstaller, Hans-Peter, Emde, Ulrich, Stähle, Wolfgang, Anzali, Soheila
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Selective RGD-Mediated Adhesion of Osteoblasts at Surfaces of Implants
Kantlehner, Martin, Finsinger, Dirk, Meyer, Jörg, Schaffner, Patricia, Jonczyk, Alfred, Diefenbach, Beate, Nies, Berthold, Kessler, Horst
Published in Angewandte Chemie (International ed.) (15.02.1999)
Published in Angewandte Chemie (International ed.) (15.02.1999)
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Access to Variously Substituted 5,6,7,8‐Tetrahydro‐3 H ‐quinazolin‐4‐ones via Diels–Alder Adducts of Phenyl Vinyl Sulfone to Cyclobutene‐Annelated Pyrimidinones
Dalai, Suryakanta, Belov, Vladimir N., Nizamov, Shamil, Rauch, Karsten, Finsinger, Dirk, de Meijere, Armin
Published in European journal of organic chemistry (01.06.2006)
Published in European journal of organic chemistry (01.06.2006)
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PYRROLOPYRIDINYLPYRIMIDIN-2-YLAMINE DERIVATIVES
GRAEDLER ULRICH, ESDAR CHRISTINA, BRUGE DAVID, FINSINGER DIRK, DORSCH DIETER, WUCHERER PLIETKER MARGARITA
Year of Publication 16.03.2011
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Year of Publication 16.03.2011
Patent
Two novel probes reveal tubular and vascular Arg-Gly-Asp (RGD) binding sites in the ischemic rat kidney
Romanov, Victor, Noiri, Eisei, Czerwinski, Grzegorz, Finsinger, Dirk, Kessler, Horst, Goligorsky, Michael S.
Published in Kidney international (01.07.1997)
Published in Kidney international (01.07.1997)
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Conference Proceeding
COMPOUNDS FOR THE TREATMENT OF VIRAL INFECTIONS
BETZ, Ulrich, POETZSCH, Sven Carsten, FINSINGER, Dirk, KLEIN, Markus, BURGDORF, Lars
Year of Publication 21.04.2022
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Year of Publication 21.04.2022
Patent