TBC1D7 Is a Third Subunit of the TSC1-TSC2 Complex Upstream of mTORC1
Dibble, Christian C., Elis, Winfried, Menon, Suchithra, Qin, Wei, Klekota, Justin, Asara, John M., Finan, Peter M., Kwiatkowski, David J., Murphy, Leon O., Manning, Brendan D.
Published in Molecular cell (24.08.2012)
Published in Molecular cell (24.08.2012)
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Activation of a Metabolic Gene Regulatory Network Downstream of mTOR Complex 1
Düvel, Katrin, Yecies, Jessica L., Menon, Suchithra, Raman, Pichai, Lipovsky, Alex I., Souza, Amanda L., Triantafellow, Ellen, Ma, Qicheng, Gorski, Regina, Cleaver, Stephen, Vander Heiden, Matthew G., MacKeigan, Jeffrey P., Finan, Peter M., Clish, Clary B., Murphy, Leon O., Manning, Brendan D.
Published in Molecular cell (30.07.2010)
Published in Molecular cell (30.07.2010)
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Bidirectional Transport of Amino Acids Regulates mTOR and Autophagy
Nicklin, Paul, Bergman, Philip, Zhang, Bailin, Triantafellow, Ellen, Wang, Henry, Nyfeler, Beat, Yang, Haidi, Hild, Marc, Kung, Charles, Wilson, Christopher, Myer, Vic E., MacKeigan, Jeffrey P., Porter, Jeffrey A., Wang, Y. Karen, Cantley, Lewis C., Finan, Peter M., Murphy, Leon O.
Published in Cell (06.02.2009)
Published in Cell (06.02.2009)
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ZNRF3 promotes Wnt receptor turnover in an R-spondin-sensitive manner
HAO, Huai-Xiang, YANG XIE, XIAOHONG MAO, QICHENG MA, ZAMPONI, Raffaella, BOUWMEESTER, Tewis, FINAN, Peter M, KIRSCHNER, Marc W, PORTER, Jeffery A, SERLUCA, Fabrizio C, FENG CONG, YUE ZHANG, CHARLAT, Olga, OSTER, Emma, AVELLO, Monika, HONG LEI, MICKANIN, Craig, DONG LIU, RUFFNER, Heinz
Published in Nature (London) (10.05.2012)
Published in Nature (London) (10.05.2012)
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RNF146 is a poly(ADP-ribose)-directed E3 ligase that regulates axin degradation and Wnt signalling
Zhang, Yue, Liu, Shanming, Mickanin, Craig, Feng, Yan, Charlat, Olga, Michaud, Gregory A, Schirle, Markus, Shi, Xiaoying, Hild, Marc, Bauer, Andreas, Myer, Vic E, Finan, Peter M, Porter, Jeffery A, Huang, Shih-Min A, Cong, Feng
Published in Nature cell biology (01.05.2011)
Published in Nature cell biology (01.05.2011)
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Tankyrase inhibition stabilizes axin and antagonizes Wnt signalling
Bauer, Andreas, Myer, Vic, Fawell, Stephen, Ghidelli, Sonja, Shi, Xiaoying, Rau, Christina, Schirle, Markus, Serluca, Fabrizio, Zhang, Yue, Bouwmeester, Tewis, Charlat, Olga, Mickanin, Craig, Curtis, Daniel, Stegmeier, Frank, Hild, Marc, Cong, Feng, Mishina, Yuji M, Wilson, Christopher J, Liu, Shanming, Wiessner, Stephanie, Tomlinson, Ronald, Fazal, Aleem, Shao, Wenlin, Shultz, Michael, Wiellette, Elizabeth, Michaud, Gregory A, Cheng, Hong, Schlegl, Judith, Finan, Peter M, Porter, Jeffery A, Lu, Chris, Cheung, Atwood, Lengauer, Christoph, Tallarico, John A, Kirschner, Marc W, Huang, Shih-Min A
Published in Nature (01.10.2009)
Published in Nature (01.10.2009)
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Identification and characterization of NVP-BEZ235, a new orally available dual phosphatidylinositol 3-kinase/mammalian target of rapamycin inhibitor with potent in vivo antitumor activity
Maira, Sauveur-Michel, Stauffer, Frédéric, Brueggen, Josef, Furet, Pascal, Schnell, Christian, Fritsch, Christine, Brachmann, Saskia, Chène, Patrick, De Pover, Alain, Schoemaker, Kevin, Fabbro, Doriano, Gabriel, Daniela, Simonen, Marjo, Murphy, Leon, Finan, Peter, Sellers, William, García-Echeverría, Carlos
Published in Molecular cancer therapeutics (01.07.2008)
Published in Molecular cancer therapeutics (01.07.2008)
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Relieving Autophagy and 4EBP1 from Rapamycin Resistance
Nyfeler, Beat, Bergman, Philip, Triantafellow, Ellen, Wilson, Christopher J., Zhu, Yanyi, Radetich, Branko, Finan, Peter M., Klionsky, Daniel J., Murphy, Leon O.
Published in Molecular and Cellular Biology (01.07.2011)
Published in Molecular and Cellular Biology (01.07.2011)
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Defective Autophagy and mTORC1 Signaling in Myotubularin Null Mice
Fetalvero, Kristina M., Yu, Yenyen, Goetschkes, Margaret, Liang, Guiqing, Valdez, Reginald A., Gould, Ty, Triantafellow, Ellen, Bergling, Sebastian, Loureiro, Joseph, Eash, John, Lin, Victor, Porter, Jeffrey A., Finan, Peter M., Walsh, Kenneth, Yang, Yi, Mao, Xiaohong, Murphy, Leon O.
Published in Molecular and Cellular Biology (01.01.2013)
Published in Molecular and Cellular Biology (01.01.2013)
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R-Spondin potentiates Wnt/β-catenin signaling through orphan receptors LGR4 and LGR5
Ruffner, Heinz, Sprunger, Joëlle, Charlat, Olga, Leighton-Davies, Juliet, Grosshans, Bianka, Salathe, Adrian, Zietzling, Svenja, Beck, Valérie, Therier, Maxime, Isken, Andrea, Xie, Yang, Zhang, Yue, Hao, Huaixiang, Shi, Xiaoying, Liu, Dong, Song, Qinhui, Clay, Ieuan, Hintzen, Gabriele, Tchorz, Jan, Bouchez, Laure C, Michaud, Gregory, Finan, Peter, Myer, Vic E, Bouwmeester, Tewis, Porter, Jeff, Hild, Marc, Bassilana, Fred, Parker, Christian N, Cong, Feng
Published in PloS one (16.07.2012)
Published in PloS one (16.07.2012)
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Inhibition of tumorigenesis driven by different Wnt proteins requires blockade of distinct ligand-binding regions by LRP6 antibodies
Ettenberg, Seth A., Charlat, Olga, Daley, Michael P., Liu, Shanming, Vincent, Karen J., Stuart, Darrin D., Schuller, Alwin G., Yuan, Jing, Ospina, Beatriz, Green, John, Yu, Qunyan, Walsh, Renee, Li, Sharon, Schmitz, Rita, Heine, Holger, Bilic, Sanela, Ostrom, Lance, Mosher, Rebecca, Hartlepp, K. Felix, Zhu, Zhenping, Fawell, Stephen, Yao, Yung-Mae, Stover, David, Finan, Peter M., Porter, Jeffery A., Sellers, William R., Klagge, Ingo M., Cong, Feng, Nusse, Roeland
Published in Proceedings of the National Academy of Sciences - PNAS (31.08.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (31.08.2010)
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RAD001 enhances the potency of BEZ235 to inhibit mTOR signaling and tumor growth
Nyfeler, Beat, Chen, Yan, Li, Xiaoyan, Pinzon-Ortiz, Maria, Wang, Zuncai, Reddy, Anupama, Pradhan, Elina, Das, Rita, Lehár, Joseph, Schlegel, Robert, Finan, Peter M, Cao, Z Alexander, Murphy, Leon O, Huang, Alan
Published in PloS one (14.11.2012)
Published in PloS one (14.11.2012)
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Rescue screens with secreted proteins reveal compensatory potential of receptor tyrosine kinases in driving cancer growth
Harbinski, Fred, Craig, Vanessa J, Sanghavi, Sneha, Jeffery, Douglas, Liu, Lijuan, Sheppard, Kelly Ann, Wagner, Sabrina, Stamm, Christelle, Buness, Andreas, Chatenay-Rivauday, Christian, Yao, Yao, He, Feng, Lu, Chris X, Guagnano, Vito, Metz, Thomas, Finan, Peter M, Hofmann, Francesco, Sellers, William R, Porter, Jeffrey A, Myer, Vic E, Graus-Porta, Diana, Wilson, Christopher J, Buckler, Alan, Tiedt, Ralph
Published in Cancer discovery (01.10.2012)
Published in Cancer discovery (01.10.2012)
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Selective VPS34 inhibitor blocks autophagy and uncovers a role for NCOA4 in ferritin degradation and iron homeostasis in vivo
Dowdle, William E, Nyfeler, Beat, Nagel, Jane, Elling, Robert A, Liu, Shanming, Triantafellow, Ellen, Menon, Suchithra, Wang, Zuncai, Honda, Ayako, Pardee, Gwynn, Cantwell, John, Luu, Catherine, Cornella-Taracido, Ivan, Harrington, Edmund, Fekkes, Peter, Lei, Hong, Fang, Qing, Digan, Mary Ellen, Burdick, Debra, Powers, Andrew F, Helliwell, Stephen B, D'Aquin, Simon, Bastien, Julie, Wang, Henry, Wiederschain, Dmitri, Kuerth, Jenny, Bergman, Philip, Schwalb, David, Thomas, Jason, Ugwonali, Savuth, Harbinski, Fred, Tallarico, John, Wilson, Christopher J, Myer, Vic E, Porter, Jeffery A, Bussiere, Dirksen E, Finan, Peter M, Labow, Mark A, Mao, Xiaohong, Hamann, Lawrence G, Manning, Brendan D, Valdez, Reginald A, Nicholson, Thomas, Schirle, Markus, Knapp, Mark S, Keaney, Erin P, Murphy, Leon O
Published in Nature cell biology (01.11.2014)
Published in Nature cell biology (01.11.2014)
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Potent, Selective, and Orally Bioavailable Inhibitors of VPS34 Provide Chemical Tools to Modulate Autophagy in Vivo
Honda, Ayako, Harrington, Edmund, Cornella-Taracido, Ivan, Furet, Pascal, Knapp, Mark S, Glick, Meir, Triantafellow, Ellen, Dowdle, William E, Wiedershain, Dmitri, Maniara, Wieslawa, Moore, Christine, Finan, Peter M, Hamann, Lawrence G, Firestone, Brant, Murphy, Leon O, Keaney, Erin P
Published in ACS medicinal chemistry letters (14.01.2016)
Published in ACS medicinal chemistry letters (14.01.2016)
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COT drives resistance to RAF inhibition through MAP kinase pathway reactivation
Emery, Caroline M, Hieronymus, Haley, Zhao, Jean J, Boehm, Jesse S, Golub, Todd, Yang, Xiaoping, Root, David E, Roberts, Thomas M, Hahn, William C, Hill, David E, Wilson, Christopher J, Weber, Barbara L, Garraway, Levi A, Johnson, Laura A, Kim, Sungjoon, Harris, Jennifer L, Kim, So Young, Vidal, Marc, Finan, Peter M, Myer, Vic E, Sellers, William R, Barretina, Jordi, Alkan, Ozan, Thomas, Sapana R, Wardwell, Leslie, Cogdill, Alexandria P, Dummer, Reinhard, Schlegel, Robert, Stransky, Nicolas, Flaherty, Keith T, Wargo, Jennifer A, Murray, Ryan R, Johannessen, Cory M, Salehi-Ashtiani, Kourosh, Caponigro, Giordano
Published in Nature (London) (16.12.2010)
Published in Nature (London) (16.12.2010)
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Genetic ablation of PI3Kγ results in defective IL‐17RA signalling in T lymphocytes and increased IL‐17 levels
Harris, Stephanie J., Ciuclan, Loredana, Finan, Peter M., Wymann, Matthias P., Walker, Christoph, Westwick, John, Ward, Stephen G., Thomas, Matthew J.
Published in European journal of immunology (01.12.2012)
Published in European journal of immunology (01.12.2012)
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Down-Regulation of Class II Phosphoinositide 3-Kinase α Expression below a Critical Threshold Induces Apoptotic Cell Death
Elis, Winfried, Triantafellow, Ellen, Wolters, Natalie M, Sian, Katie R, Caponigro, Giordano, Borawski, Jason, Gaither, L Alex, Murphy, Leon O, Finan, Peter M, Mackeigan, Jeffrey P
Published in Molecular cancer research (01.04.2008)
Published in Molecular cancer research (01.04.2008)
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Regulation of P-Rex1 by Phosphatidylinositol (3,4,5)-Trisphosphate and Gβγ Subunits
Hill, Kirsti, Krugmann, Sonja, Andrews, Simon R., Coadwell, W. John, Finan, Peter, Welch, Heidi C.E., Hawkins, Phillip T., Stephens, Len R.
Published in The Journal of biological chemistry (11.02.2005)
Published in The Journal of biological chemistry (11.02.2005)
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IL-10 expression profiling in human monocytes
Williams, Lynn, Jarai, Gabor, Smith, Alexandra, Finan, Peter
Published in Journal of leukocyte biology (01.10.2002)
Published in Journal of leukocyte biology (01.10.2002)
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