Structure−Function Studies on the New Growth Hormone-Releasing Peptide, Ghrelin: Minimal Sequence of Ghrelin Necessary for Activation of Growth Hormone Secretagogue Receptor 1a
Bednarek, Maria A, Feighner, Scott D, Pong, Sheng-Shung, McKee, Karen Kulju, Hreniuk, Donna L, Silva, Maria V, Warren, Vivien A, Howard, Andrew D, Van der Ploeg, Lex H. Y, Heck, James V
Published in Journal of medicinal chemistry (16.11.2000)
Published in Journal of medicinal chemistry (16.11.2000)
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Journal Article
Orphan G-protein-coupled receptors and natural ligand discovery
Howard, Andrew D, McAllister, George, Feighner, Scott D, Liu, Qingyun, Nargund, Ravi P, Van der Ploeg, Lex H.T, Patchett, Arthur A
Published in Trends in Pharmacological Sciences (01.03.2001)
Published in Trends in Pharmacological Sciences (01.03.2001)
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Book Review
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Melanin-Concentrating Hormone Receptor Subtypes 1 and 2: Species-Specific Gene Expression
Tan, Carina P., Sano, Hideki, Iwaasa, Hisashi, Pan, Jie, Sailer, Andreas W., Hreniuk, Donna L., Feighner, Scott D., Palyha, Oksana C., Pong, Sheng-Shung, Figueroa, David J., Austin, Christopher P., Jiang, Michael M., Yu, Hong, Ito, Junko, Ito, Makoto, Ito, Masahiko, Guan, Xiao Ming, MacNeil, Douglas J., Kanatani, Akio, Van der Ploeg, Lex H.T., Howard, Andrew D.
Published in Genomics (San Diego, Calif.) (01.06.2002)
Published in Genomics (San Diego, Calif.) (01.06.2002)
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Journal Article
Chronic MCH-1 receptor modulation alters appetite, body weight and adiposity in rats
Shearman, Lauren P., Camacho, Ramon E., Sloan Stribling, D., Zhou, Dan, Bednarek, Maria A., Hreniuk, Donna L., Feighner, Scott D., Tan, Carina P., Howard, Andrew D., Van der Ploeg, Lex H.T., MacIntyre, D.Euan, Hickey, Gerard J., Strack, Alison M.
Published in European journal of pharmacology (15.08.2003)
Published in European journal of pharmacology (15.08.2003)
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Journal Article
Molecular Analysis of Rat Pituitary and Hypothalamic Growth Hormone Secretagogue Receptors
McKee, Karen Kulju, Palyha, Oksana C, Feighner, Scott D, Hreniuk, Donna L, Tan, Carina P, Phillips, Michael S, Smith, Roy G, Van der Ploeg, Lex H. T, Howard, Andrew D
Published in Molecular endocrinology (Baltimore, Md.) (01.04.1997)
Published in Molecular endocrinology (Baltimore, Md.) (01.04.1997)
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Journal Article
Peptidomimetic Regulation of Growth Hormone Secretion
Smith, Roy G, Van der Ploeg, Lex H. T, Howard, Andrew D, Feighner, Scott D, Cheng, Kang, Hickey, Gerard J, Wyvratt, Matthew J, Fisher, Mike H, Nargund, Ravi P, Patchett, Arthur A
Published in Endocrine reviews (01.10.1997)
Published in Endocrine reviews (01.10.1997)
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Journal Article
Discovery and optimization of novel 4-[(aminocarbonyl)amino]- N-[4-(2-aminoethyl)phenyl]benzenesulfonamide ghrelin receptor antagonists
Pasternak, Alexander, Goble, Stephen D., deJesus, Reynalda K., Hreniuk, Donna L., Chung, Christine C., Tota, Michael R., Mazur, Paul, Feighner, Scott D., Howard, Andrew D., Mills, Sander G., Yang, Lihu
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
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Journal Article
Characterization of the bombesin-like peptide receptor family in primates
Sano, Hideki, Feighner, Scott D, Hreniuk, Donna L, Iwaasa, Hisashi, Sailer, Andreas W, Pan, Jie, Reitman, Marc L, Kanatani, Akio, Howard, Andrew D, Tan, Carina P
Published in Genomics (San Diego, Calif.) (01.07.2004)
Published in Genomics (San Diego, Calif.) (01.07.2004)
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Journal Article
Hypothalamic Growth Hormone Secretagogue-Receptor (GHS-R) Expression Is Regulated by Growth Hormone in the Rat
Bennett, Pamela A, Thomas, Gregory B, Howard, Andrew D, Feighner, Scott D, Van der Ploeg, Lex H. T, Smith, Roy G, Robinson, Iain C. A. F
Published in Endocrinology (Philadelphia) (01.11.1997)
Published in Endocrinology (Philadelphia) (01.11.1997)
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Journal Article
Discovery of substituted biphenyl imidazoles as potent, bioavailable bombesin receptor subtype-3 agonists
He, Shuwen, Dobbelaar, Peter H., Liu, Jian, Jian, Tianying, Sebhat, Iyassu K., Lin, Linus S., Goodman, Allan, Guo, Cheng, Guzzo, Peter R., Hadden, Mark, Henderson, Alan J., Ruenz, Megan, Sargent, Bruce J., Yet, Larry, Kelly, Theresa M., Palyha, Oksana, Kan, Yanqing, Pan, Jie, Chen, Howard, Marsh, Donald J., Shearman, Lauren P., Strack, Alison M., Metzger, Joseph M., Feighner, Scott D., Tan, Carina, Howard, Andrew D., Tamvakopoulos, Constantin, Peng, Qianping, Guan, Xiao-Ming, Reitman, Marc L., Patchett, Arthur A., Wyvratt, Matthew J., Nargund, Ravi P.
Published in Bioorganic & medicinal chemistry letters (15.03.2010)
Published in Bioorganic & medicinal chemistry letters (15.03.2010)
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Journal Article
Ligand Activation Domain of Human Orphan Growth Hormone (GH) Secretagogue Receptor (GHS-R) Conserved from Pufferfish to Humans
Palyha, Oksana C, Feighner, Scott D, Tan, Carina P, McKee, Karen Kulju, Hreniuk, Donna L, Gao, Ying-Duo, Schleim, Klaus D, Yang, Lihu, Morriello, Gregori J, Nargund, Ravi, Patchett, Arthur A, Howard, Andrew D, Smith, Roy G
Published in Molecular endocrinology (Baltimore, Md.) (01.01.2000)
Published in Molecular endocrinology (Baltimore, Md.) (01.01.2000)
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Journal Article
Molecular cloning and characterization of a new receptor for galanin
Howard, Andrew D, Tan, Carina, Shiao, Lin-Lin, Palyha, Oksana C, McKee, Karen Kulju, Weinberg, David H, Feighner, Scott D, Cascieri, Margaret A, Smith, Roy G, Van Der Ploeg, Lex H.T, Sullivan, Kathleen A
Published in FEBS letters (01.04.1997)
Published in FEBS letters (01.04.1997)
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Journal Article
Synthesis and Biological Evaluation in Vitro of Selective, High Affinity Peptide Antagonists of Human Melanin-Concentrating Hormone Action at Human Melanin-Concentrating Hormone Receptor 1
Bednarek, Maria A, Hreniuk, Donna L, Tan, Carina, Palyha, Oksana C, MacNeil, Douglas J, Van der Ploeg, Lex H. Y, Howard, Andrew D, Feighner, Scott D
Published in Biochemistry (Easton) (21.05.2002)
Published in Biochemistry (Easton) (21.05.2002)
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Journal Article
Growth hormone secretagogue receptor family members and ligands
Smith, R G, Leonard, R, Bailey, A R, Palyha, O, Feighner, S, Tan, C, Mckee, K K, Pong, S S, Griffin, P, Howard, A
Published in Endocrine (01.02.2001)
Published in Endocrine (01.02.2001)
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Journal Article
Identification and Characterization of a Second Melanin-Concentrating Hormone Receptor, MCH-2R
Sailer, Andreas W., Sano, Hideki, Zeng, Zhizhen, McDonald, Terrence P., Pan, Jie, Pong, Sheng-Shung, Feighner, Scott D., Tan, Carina P., Fukami, Takehiro, Iwaasa, Hisashi, Hreniuk, Donna L., Morin, Nancy R., Sadowski, Sharon J., Ito, Makoto, Ito, Masahiko, Bansal, Alka, Ky, Betty, Figueroa, David J., Jiang, Qingping, Austin, Christopher P., MacNeil, Douglas J., Ishihara, Akane, Ihara, Masaki, Kanatani, Akio, Lex H. T. Van der Ploeg, Howard, Andrew D., Liu, Qingyun
Published in Proceedings of the National Academy of Sciences - PNAS (19.06.2001)
Published in Proceedings of the National Academy of Sciences - PNAS (19.06.2001)
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Journal Article
Structural Requirements for the Activation of the Human Growth Hormone Secretagogue Receptor by Peptide and Nonpeptide Secretagogues
Feighner, Scott D, Howard, Andrew D, Prendergast, Kristine, Palyha, Oksana C, Hreniuk, Donna L, Nargund, Ravi, Underwood, Dennis, Tata, James R, Dean, Dennis C, Tan, Carina P, McKee, Karen Kulju, Woods, John W, Patchett, Arthur A, Smith, Roy G, Van der Ploeg, Lex H. T
Published in Molecular endocrinology (Baltimore, Md.) (01.01.1998)
Published in Molecular endocrinology (Baltimore, Md.) (01.01.1998)
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Journal Article
Synthesis and Biological Evaluation in Vitro of a Selective, High Potency Peptide Agonist of Human Melanin-concentrating Hormone Action at Human Melanin-concentrating Hormone Receptor 1
Bednarek, Maria A., Tan, Carina, Hreniuk, Donna L., Palyha, Oksana C., MacNeil, Douglas J., Van der Ploeg, Lex H.Y., Howard, Andrew D., Feighner, Scott D.
Published in The Journal of biological chemistry (19.04.2002)
Published in The Journal of biological chemistry (19.04.2002)
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Journal Article
A New Orphan Receptor Involved in Pulsatile Growth Hormone Release
Smith, Roy G, Feighner, Scott, Prendergast, Kris, Guan, Xiaoming, Howard, Andrew
Published in Trends in Endocrinology & Metabolism (01.05.1999)
Published in Trends in Endocrinology & Metabolism (01.05.1999)
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Book Review
Journal Article
Phylogenetic relationships among eight Eimeria species infecting domestic fowl inferred using complete small subunit ribosomal DNA sequences
Barta, J R, Martin, D S, Liberator, P A, Dashkevicz, M, Anderson, J W, Feighner, S D, Elbrecht, A, Perkins-Barrow, A, Jenkins, M C, Danforth, H D, Ruff, M D, Profous-Juchelka, H
Published in The Journal of parasitology (01.04.1997)
Published in The Journal of parasitology (01.04.1997)
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Journal Article
Increased Melanin Concentrating Hormone Receptor Type I in the Human Hypothalamic Infundibular Nucleus in Cachexia
Unmehopa, Unga A, van Heerikhuize, Joop J, Spijkstra, Wenda, Woods, John W, Howard, Andrew D, Zycband, Emanuel, Feighner, Scott D, Hreniuk, Donna L, Palyha, Oksana C, Guan, Xiao-Ming, MacNeil, Douglas J, Van der Ploeg, Lex H. T, Swaab, Dick F
Published in The journal of clinical endocrinology and metabolism (01.04.2005)
Published in The journal of clinical endocrinology and metabolism (01.04.2005)
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