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Tetrahydroquinoline-based tricyclic amines as potent and selective agonists of the 5-HT 2C receptor

Tetrahydroquinoline-based tricyclic amines as potent and selective agonists of the 5-HT 2C receptor

by Schrader, Thomas O, Kasem, Michelle, Ren, Albert, Feichtinger, Konrad, Al Doori, Bilal, Wei, Jing, Wu, Chunrui, Dang, Huong, Le, Minh, Gatlin, Joel, Chase, Kelli, Dong, Jenny, Whelan, Kevin T, Sage, Carleton, Grottick, Andrew J, Semple, Graeme
Published in Bioorganic & medicinal chemistry letters (01.12.2016)

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Journal Article

Diprotected Triflylguanidines: A New Class of Guanidinylation Reagents

Diprotected Triflylguanidines: A New Class of Guanidinylation Reagents

by Feichtinger, Konrad, Zapf, Christoph, Sings, Heather L, Goodman, Murray
Published in Journal of organic chemistry (12.06.1998)

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Journal Article

Triurethane-Protected Guanidines and Triflyldiurethane-Protected Guanidines: New Reagents for Guanidinylation Reactions

Triurethane-Protected Guanidines and Triflyldiurethane-Protected Guanidines: New Reagents for Guanidinylation Reactions

by Feichtinger, Konrad, Sings, Heather L, Baker, Tracy J, Matthews, Kenneth, Goodman, Murray
Published in Journal of organic chemistry (13.11.1998)

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Journal Article

Novel (R)-6,6a,7,8,9,10-hexahydro-5H-pyrazino[1,2-a][1,n]naphthyridines as potent and selective agonists of the 5-HT2C receptor

Novel (R)-6,6a,7,8,9,10-hexahydro-5H-pyrazino[1,2-a][1,n]naphthyridines as potent and selective agonists of the 5-HT2C receptor

by Schrader, Thomas O., Zhu, Xiuwen, Kasem, Michelle, Ren, Albert, Liu, Chunyan, Wu, Chunrui, Dang, Huong, Le, Minh, Gatlin, Joel, Chase, Kelli, Frazer, John, Whelan, Kevin T., Grottick, Andrew J., Hutton, Clayton, Barden, Jeremy, Chen, Chuan, Ortiz, Alvaro, Feichtinger, Konrad, Semple, Graeme
Published in Bioorganic & medicinal chemistry letters (15.04.2021)

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Journal Article

Discovery of a lead series of potent benzodiazepine 5-HT2C receptor agonists with high selectivity in functional and binding assays

Discovery of a lead series of potent benzodiazepine 5-HT2C receptor agonists with high selectivity in functional and binding assays

by Ren, Albert, Zhu, Xiuwen, Feichtinger, Konrad, Lehman, Juerg, Kasem, Michelle, Schrader, Thomas O., Wong, Amy, Dang, Huong, Le, Minh, Frazer, John, Unett, David J., Grottick, Andrew J., Whelan, Kevin T., Morgan, Michael E., Sage, Carleton R., Semple, Graeme
Published in Bioorganic & medicinal chemistry letters (01.03.2020)

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Journal Article

Tetrahydroquinoline-based tricyclic amines as potent and selective agonists of the 5-HT2C receptor

Tetrahydroquinoline-based tricyclic amines as potent and selective agonists of the 5-HT2C receptor

by Schrader, Thomas O., Kasem, Michelle, Ren, Albert, Feichtinger, Konrad, Al Doori, Bilal, Wei, Jing, Wu, Chunrui, Dang, Huong, Le, Minh, Gatlin, Joel, Chase, Kelli, Dong, Jenny, Whelan, Kevin T., Sage, Carleton, Grottick, Andrew J., Semple, Graeme
Published in Bioorganic & medicinal chemistry letters (15.12.2016)

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Journal Article

5-HT2C 수용체 효능제 및 조성물 및 사용 방법

5-HT2C 수용체 효능제 및 조성물 및 사용 방법

by REN ALBERT S, FEICHTINGER KONRAD, LEHMANN JUERG, SEMPLE GRAEME
Year of Publication 27.03.2018

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Patent

Novel (R)-6,6a,7,8,9,10-hexahydro-5H-pyrazino[1,2-a][1,n]naphthyridines as potent and selective agonists of the 5-HT 2C receptor

Novel (R)-6,6a,7,8,9,10-hexahydro-5H-pyrazino[1,2-a][1,n]naphthyridines as potent and selective agonists of the 5-HT 2C receptor

by Schrader, Thomas O, Zhu, Xiuwen, Kasem, Michelle, Ren, Albert, Liu, Chunyan, Wu, Chunrui, Dang, Huong, Le, Minh, Gatlin, Joel, Chase, Kelli, Frazer, John, Whelan, Kevin T, Grottick, Andrew J, Hutton, Clayton, Barden, Jeremy, Chen, Chuan, Ortiz, Alvaro, Feichtinger, Konrad, Semple, Graeme
Published in Bioorganic & medicinal chemistry letters (15.04.2021)

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Journal Article

Discovery of a lead series of potent benzodiazepine 5-HT 2C receptor agonists with high selectivity in functional and binding assays

Discovery of a lead series of potent benzodiazepine 5-HT 2C receptor agonists with high selectivity in functional and binding assays

by Ren, Albert, Zhu, Xiuwen, Feichtinger, Konrad, Lehman, Juerg, Kasem, Michelle, Schrader, Thomas O, Wong, Amy, Dang, Huong, Le, Minh, Frazer, John, Unett, David J, Grottick, Andrew J, Whelan, Kevin T, Morgan, Michael E, Sage, Carleton R, Semple, Graeme
Published in Bioorganic & medicinal chemistry letters (01.03.2020)

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Journal Article

Identification of fused bicyclic heterocycles as potent and selective 5-HT2A receptor antagonists for the treatment of insomnia

Identification of fused bicyclic heterocycles as potent and selective 5-HT2A receptor antagonists for the treatment of insomnia

by Xiong, Yifeng, Ullman, Brett, Choi, Jin-Sun Karoline, Cherrier, Martin, Strah-Pleynet, Sonja, Decaire, Marc, Feichtinger, Konrad, Frazer, John M., Yoon, Woo H., Whelan, Kevin, Sanabria, Erin K., Grottick, Andrew J., Al-Shamma, Hussien, Semple, Graeme
Published in Bioorganic & medicinal chemistry letters (01.03.2012)

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Journal Article

Discovery and Structure-Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine(2A) Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

Discovery and Structure-Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine(2A) Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

by Xiong, Yifeng, Teegarden, Bradley R., Choi, Jin-Sun Karoline, Strah-Pleynet, Sonja, Decaire, Marc, Jayakumar, Honnappa, Dosa, Peter I., Casper, Martin D., Pham, Lan, Feichtinger, Konrad, Ullman, Brett, Adams, John, Yuskin, Diane, Frazer, John, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Webb, Robert R., Connolly, Daniel T., Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (10.06.2010)

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Journal Article

Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine(2A) Receptor Antagonists for the Treatment of Insomnia

Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine(2A) Receptor Antagonists for the Treatment of Insomnia

by Xiong, Yifeng, Ullman, Brett, Choi, Jin-Sun Karoline, Cherrier, Martin, Strah-Pleynet, Sonja, Decaire, Marc, Dosa, Peter I., Feichtinger, Konrad, Teegarden, Bradley R., Frazer, John M., Yoon, Woo H., Shan, Yun, Whelan, Kevin, Hauser, Erin K., Grottick, Andrew J., Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (12.08.2010)

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Journal Article

Discovery and Structure−Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

Discovery and Structure−Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

by Xiong, Yifeng, Teegarden, Bradley R, Choi, Jin-Sun Karoline, Strah-Pleynet, Sonja, Decaire, Marc, Jayakumar, Honnappa, Dosa, Peter I, Casper, Martin D, Pham, Lan, Feichtinger, Konrad, Ullman, Brett, Adams, John, Yuskin, Diane, Frazer, John, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Webb, Robert R, Connolly, Daniel T, Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (10.06.2010)

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Journal Article

Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine2A Receptor Antagonists for the Treatment of Insomnia

Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine2A Receptor Antagonists for the Treatment of Insomnia

by Xiong, Yifeng, Ullman, Brett, Choi, Jin-Sun Karoline, Cherrier, Martin, Strah-Pleynet, Sonja, Decaire, Marc, Dosa, Peter I, Feichtinger, Konrad, Teegarden, Bradley R, Frazer, John M, Yoon, Woo H, Shan, Yun, Whelan, Kevin, Hauser, Erin K, Grottick, Andrew J, Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (12.08.2010)

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Journal Article

GUANIDINYLATION REAGENTS

GUANIDINYLATION REAGENTS

by ROMOFF TODD T. ROMOFF TODD T, GOODMAN MURRAY GOODMAN MURRAY, FEICHTINGER KONRAD FEICHTINGER KONRAD
Year of Publication 28.03.2001

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Patent

Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine 2A Receptor Antagonists for the Treatment of Insomnia

Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine 2A Receptor Antagonists for the Treatment of Insomnia

by Xiong, Yifeng, Ullman, Brett, Choi, Jin-Sun Karoline, Cherrier, Martin, Strah-Pleynet, Sonja, Decaire, Marc, Dosa, Peter I., Feichtinger, Konrad, Teegarden, Bradley R., Frazer, John M., Yoon, Woo H., Shan, Yun, Whelan, Kevin, Hauser, Erin K., Grottick, Andrew J., Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (12.08.2010)

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Journal Article

Discovery and Structure−Activity Relationship of 3-Methoxy- N -(3-(1-methyl-1 H -pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine 2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

Discovery and Structure−Activity Relationship of 3-Methoxy- N -(3-(1-methyl-1 H -pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine 2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

by Xiong, Yifeng, Teegarden, Bradley R., Choi, Jin-Sun Karoline, Strah-Pleynet, Sonja, Decaire, Marc, Jayakumar, Honnappa, Dosa, Peter I., Casper, Martin D., Pham, Lan, Feichtinger, Konrad, Ullman, Brett, Adams, John, Yuskin, Diane, Frazer, John, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Webb, Robert R., Connolly, Daniel T., Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (10.06.2010)

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Journal Article

5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE

5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE

by Ren, Albert S, Feichtinger, Konrad, Semple, Graeme, Lehmann, Juerg
Year of Publication 23.02.2023

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Patent

3-PHENYL-PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

3-PHENYL-PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

by XIONG YIFENG, JONES ROBERT M, UNETT DAVID J, JAYAKUMAR HONNAPPA, CHOI JIN SUN KAROLINE, DOSA PETER I, FEICHTINGER KONRAD, CASPER MARTIN, LEHMANN JUERG, TEEGARDEN BRADLEY, STRAH PLEYNET SONJA
Year of Publication 14.03.2013

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Patent

5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE

5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE

by SEMPLE, Graeme, LEHMANN, Juerg, REN, Albert S, FEICHTINGER, Konrad
Year of Publication 12.10.2022

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Patent

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