Hydrophobic Vancomycin Derivatives with Improved ADME Properties: Discovery of Telavancin (TD-6424)
LEADBETTER, MICHAEL R., ADAMS, STACY M., BAZZINI, BETTINA, FATHEREE, PAUL R., KARR, DANE E., KRAUSE, KEVIN M., LAM, BERNICE M. T., LINSELL, MARTIN S., NODWELL, MATTHEW B., PACE, JOHN L., QUAST, KELLY, SHAW, JENG-PYNG, SORIANO, ELIZABETH, TRAPP, SEAN G., VILLENA, JENNY D., WU, TERRY X., CHRISTENSEN, BURTON G., JUDICE, J. KEVIN
Published in Journal of antibiotics (01.05.2004)
Published in Journal of antibiotics (01.05.2004)
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Exploring the Positional Attachment of Glycopeptide/β-lactam Heterodimers
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Published in Journal of antibiotics (01.10.2008)
Published in Journal of antibiotics (01.10.2008)
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Discovery of TD-8954, a clinical stage 5-HT4 receptor agonist with gastrointestinal prokinetic properties
McKinnell, R. Murray, Armstrong, Scott R., Beattie, David T., Fatheree, Paul R., Long, Daniel D., Marquess, Daniel G., Shaw, Jeng-Pyng, Vickery, Ross G.
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
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Discovery, oral pharmacokinetics and in vivo efficacy of velusetrag, a highly selective 5-HT4 receptor agonist that has achieved proof-of-concept in patients with chronic idiopathic constipation
Long, Daniel D., Armstrong, Scott R., Beattie, David T., Choi, Seok-Ki, Fatheree, Paul R., Gendron, Roland A.L., Genov, Daniel, Goldblum, Adam A., Humphrey, Patrick P., Jiang, Lan, Marquess, Daniel G., Shaw, Jeng-Pyng, Smith, Jacqueline A.M., Turner, S. Derek, Vickery, Ross G.
Published in Bioorganic & medicinal chemistry letters (01.10.2012)
Published in Bioorganic & medicinal chemistry letters (01.10.2012)
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페닐 아세트아미드 기재 IL-17A 조정제 및 그의 용도
AQUINO CLAUDIO, CHURCH TIMOTHY J, REILLY MAUREEN, FATHEREE PAUL R, FREIDBERG MICHAEL
Year of Publication 05.04.2024
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Year of Publication 05.04.2024
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Discovery, oral pharmacokinetics and in vivo efficacy of a highly selective 5-HT4 receptor agonist: Clinical compound TD-2749
Long, Daniel D., Armstrong, Scott R., Beattie, David T., Choi, Seok-Ki, Fatheree, Paul R., Gendron, Roland A.L., Goldblum, Adam A., Humphrey, Patrick P., Marquess, Daniel G., Shaw, Jeng-Pyng, Smith, Jacqueline A.M., Derek Turner, S., Vickery, Ross G.
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
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A Multivalent Approach to the Design and Discovery of Orally Efficacious 5-HT4 Receptor Agonists
McKinnell, R. Murray, Armstrong, Scott R, Beattie, David T, Choi, Seok-Ki, Fatheree, Paul R, Gendron, Roland A. L, Goldblum, Adam, Humphrey, Patrick P, Long, Daniel D, Marquess, Daniel G, Shaw, J. P, Smith, Jacqueline A. M, Turner, S. Derek, Vickery, Ross G
Published in Journal of medicinal chemistry (10.09.2009)
Published in Journal of medicinal chemistry (10.09.2009)
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IL-17A 조절인자 및 이의 용도
LINSELL MARTIN S, AQUINO CLAUDIO, CHURCH TIMOTHY J, VAN DER LINDEN WOUTER A, JACOBSEN JOHN R, PAULICK MARGOT G, FATHEREE PAUL R
Year of Publication 19.07.2022
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Year of Publication 19.07.2022
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NAPHTHYRIDINE COMPOUNDS AS JAK KINASE INHIBITORS
DANTE D PODESTO, JENNIFER KOZAK, MELISSA FLEURY, HUANG XIAOJUN, VENKAT R THALLADI, RYAN HUDSON, GARY E L BLANT, ANNE-MARIE BEAUSOLEIL, FATHEREE PAUL R
Year of Publication 01.07.2021
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NAPHTHYRIDINE COMPOUNDS AS JAK KINASE INHIBITORS
DANTE D PODESTO, JENNIFER KOZAK, MELISSA FLEURY, HUANG XIAOJUN, VENKAT R THALLADI, RYAN HUDSON, GARY E L BLANT, ANNE-MARIE BEAUSOLEIL, FATHEREE PAUL R
Year of Publication 07.01.2021
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Year of Publication 07.01.2021
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NAPHTHYRIDINE COMPOUNDS AS JAK KINASE INHIBITORS
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Year of Publication 27.07.2020
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Year of Publication 26.12.2019
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Year of Publication 26.12.2019
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JAK 키나제 저해제로서 피리미딘 화합물
HUANG XIAOJUN, KOZAK JENNIFER, HUDSON RYAN, FLEURY MELISSA, BEAUSOLEIL ANNE MARIE, PODESTO DANTE D, FATHEREE PAUL R
Year of Publication 08.01.2019
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Year of Publication 08.01.2019
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융합된 이미다조-피페리딘 JAK 저해제
SMITH CAMERON, KLEINSCHEK MELANIE A, CRATER GLENN D, SULLIVAN STEVEN D.E, VAN ORDEN LORI JEAN, FATHEREE PAUL R, BRANDT GARY E.L
Year of Publication 13.11.2019
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Year of Publication 13.11.2019
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SMITH CAMERON, KLEINSCHEK MELANIE A, CRATER GLENN D, SULLIVAN STEVEN D.E, VAN ORDEN LORI JEAN, FATHEREE PAUL R, BRANDT GARY E.L
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Year of Publication 31.01.2018
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Year of Publication 31.01.2018
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FASS GENE TIMOTHY, BENJAMIN NOAH, BEAUSOLEIL ANNE MARIE, FLEURY MELISSA, COLSON PIERRE JEAN, SULLIVAN STEVEN D.E, VAN ORDEN LORI JEAN, SMITH CAMERON, JACOBSEN JOHN R, THALLADI VENKAT R, JIANG LAN, DABROS MARTA, RAPTA MIROSLAV, FATHEREE PAUL R, BRANDT GARY E.L
Year of Publication 02.07.2018
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Year of Publication 02.07.2018
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