A Robust Process for an mGluR5 Negative Allosteric Modulator: Difluoromethylation and Sonogashira Coupling on Large Scale
Sperry, Jeffrey B, Farr, Roger M, Levent, Mahmut, Ghosh, Mousumi, Hoagland, Steven M, Varsolona, Richard J, Sutherland, Karen
Published in Organic process research & development (16.11.2012)
Published in Organic process research & development (16.11.2012)
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Highly Regioselective Friedländer Annulations with Unmodified Ketones Employing Novel Amine Catalysts: Syntheses of 2-Substituted Quinolines, 1,8-Naphthyridines, and Related Heterocycles
Dormer, Peter G, Eng, Kan K, Farr, Roger N, Humphrey, Guy R, McWilliams, J. Christopher, Reider, P. J, Sager, Jess W, Volante, R. P
Published in Journal of organic chemistry (24.01.2003)
Published in Journal of organic chemistry (24.01.2003)
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Practical Enantioselective Synthesis of a 3-Aryl-3-trifluoromethyl-2-aminopropanol Derivative
Alimardanov, Asaf, Nikitenko, Antonia, Connolly, Terrence J, Feigelson, Gregg, Chan, Anita W, Ding, Zhixian, Ghosh, Mousumi, Shi, Xinxu, Ren, Jianxin, Hansen, Eric, Farr, Roger, MacEwan, Michael, Tadayon, Sam, Springer, Dane M, Kreft, Anthony F, Ho, Douglas M, Potoski, John R
Published in Organic process research & development (20.11.2009)
Published in Organic process research & development (20.11.2009)
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Enantiospecific and regioselective opening of 2-alkyl nosylaziridines by indoles mediated by boron trifluoride. Application to a practical synthesis of a GnRH antagonist
Farr, Roger N, Alabaster, Ramon J, Chung, John Y.L, Craig, Bridgette, Edwards, John S, Gibson, Andrew W, Ho, Guo-Jie, Humphrey, Guy R, Johnson, Simon A, Grabowski, E.J.J
Published in Tetrahedron: asymmetry (14.11.2003)
Published in Tetrahedron: asymmetry (14.11.2003)
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8-Ethenyl-1-hydroxy-4-.beta.-D-ribofuranosylbenzo[d]naphtho[1,2-b]pyran-6-one and 8-ethenyl-1-hydroxy-4-(2'-deoxy-.beta.-D-ribofuranosyl)benzo[d]naphtho[1,2-b]pyran-6-one. Synthetic C-glycosides related to the gilvocarcin, ravidomycin, and chrysomycin antibiotics
Farr, Roger N, Kwok, Daw Iong, Daves, G. Doyle
Published in Journal of organic chemistry (01.03.1992)
Published in Journal of organic chemistry (01.03.1992)
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Palladium-mediated coupling of a 3-deoxy pyranoid glycal: stereochemistry of C-glycosyl bond formation
Kwok, Daw Long, Farr, Roger N, Daves, G. Doyle
Published in Journal of organic chemistry (01.05.1991)
Published in Journal of organic chemistry (01.05.1991)
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A Convenient and Stable Synthon for Ethyl Azide and Its Evaluation in a [3 + 2]-Cycloaddition Reaction under Continuous-Flow Conditions
Tinder, Rob, Farr, Roger, Heid, Richard, Zhao, Ralph, Rarig, Randy S, Storz, Thomas
Published in Organic process research & development (20.11.2009)
Published in Organic process research & development (20.11.2009)
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Journal Article
C-Glycoside synthesis by palladium-catalyzed iodoaglycon-glycal coupling
Farr, Roger N, Outten, Robert A, Cheng, Jane Chi Ya, Daves, G. Doyle
Published in Organometallics (01.12.1990)
Published in Organometallics (01.12.1990)
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Synthesis of a selective estrogen receptor β-modulator via asymmetric phase-transfer catalysis
Huffman, Mark A., Rosen, Jonathan D., Farr, Roger N., Lynch, Joseph E.
Published in Tetrahedron (21.05.2007)
Published in Tetrahedron (21.05.2007)
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Assignment of anomeric configuration of C-glycopyranosides and C-glycofuranosides. A proton, carbon-13, and nuclear Overhauser enhancement spectrometric study
Brakta, Mohamed, Farr, Roger N, Chaguir, Brahim, Massiot, Georges, Lavaud, Catherine, Anderson, William R, Sinou, Denis, Daves, G. Doyle
Published in Journal of organic chemistry (01.05.1993)
Published in Journal of organic chemistry (01.05.1993)
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