Stereoselective metabolism of pyrido[3,2-D]pyrimidine-containing compounds by aldehyde oxidase
He, Xiaowei, Amy Siu, Y., David Hong, W., Benayoud, Farid, George Lai, W.
Published in Drug metabolism and pharmacokinetics (01.01.2018)
Published in Drug metabolism and pharmacokinetics (01.01.2018)
Get full text
Journal Article
Halichondrin B: Synthesis of the C1−C22 Subunit
Lambert, William T, Hanson, Gregory H, Benayoud, Farid, Burke, Steven D
Published in Journal of organic chemistry (11.11.2005)
Published in Journal of organic chemistry (11.11.2005)
Get full text
Journal Article
AWZ1066S, a highly specific anti-Wolbachia drug candidate for a short-course treatment of filariasis
Hong, W. David, Benayoud, Farid, Nixon, Gemma L., Ford, Louise, Johnston, Kelly L., Clare, Rachel H., Cassidy, Andrew, Cook, Darren A. N., Siu, Amy, Shiotani, Motohiro, Webborn, Peter J. H., Kavanagh, Stefan, Aljayyoussi, Ghaith, Murphy, Emma, Steven, Andrew, Archer, John, Struever, Dominique, Frohberger, Stefan J., Ehrens, Alexandra, Hübner, Marc P., Hoerauf, Achim, Roberts, Adam P., Hubbard, Alasdair T. M., Tate, Edward W., Serwa, Remigiusz A., Leung, Suet C., Qie, Li, Berry, Neil G., Gusovsky, Fabian, Hemingway, Janet, Turner, Joseph D., Taylor, Mark J., Ward, Stephen A., O’Neill, Paul M.
Published in Proceedings of the National Academy of Sciences - PNAS (22.01.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (22.01.2019)
Get full text
Journal Article
Efficient Syntheses of (α-Fluoropropargyl)phosphonate Esters
Benayoud, Farid, deMendonca, Daniel J, Digits, Cheryl A, Moniz, George A, Sanders, Tanya C, Hammond, Gerald B
Published in Journal of organic chemistry (26.07.1996)
Published in Journal of organic chemistry (26.07.1996)
Get full text
Journal Article
Transformation of the Manufacturing Process from Discovery to Kilogram Scale for AWZ1066S: A Highly Specific Anti-Wolbachia Drug Candidate for a Short-Course Treatment of Filariasis
Hong, W. David, O’Neill, Paul M., Taylor, Mark J., Turner, Joseph D., Ward, Stephen A., Gusovsky, Fabian, Benayoud, Farid, Shibuguchi, Nao, Girish, Dixit, Fang, Francis Gerard, Talabhakthla, Ravi Kumar, Vaddi, Anand, Challa, Chiranjeevi, Reddy, Karri Satya Ammi, Kalla, Vijay, Srinivasa Rao, Sugandham, Nagireddi, Durga Mahesh Kumar, Patel, Jayesh, Khile, Anil Shahaji
Published in Organic process research & development (20.01.2023)
Published in Organic process research & development (20.01.2023)
Get full text
Journal Article
Synthesis of BACE1 Inhibitors E2609/E2071 via Oxime–Olefin Cycloaddition Following a Process Risk Mitigation Strategy
Kim, Dae-Shik, Yoshizawa, Kazuhiro, Mitasev, Branko, Schnaderbeck, Matthew, Zhang, Huiming, Omori, Masayuki, Kayano, Akio, Nagai, Mitsuo, Wakasugi, Kazunori, Watanabe, Yuzo, Benayoud, Farid, Suzuki, Yuichi, Motoki, Takafumi, Kaneko, Toshihiko, Takaishi, Mamoru, Ishida, Tasuku, Takeda, Kunitoshi, Kita, Yoichi, Yamamoto, Noboru, Khan, Afzal, Dimopoulos, Paschalis, Farthing, Christopher N, Hall, Adrian, Chanda, Arani, Lu, Lily, Bracke, Markus, Fang, Francis G
Published in Organic process research & development (18.03.2022)
Published in Organic process research & development (18.03.2022)
Get full text
Journal Article
INTERMEDIATES FOR PREPARATION OF HALICHONDRIN B ANALOGS
AUSTAD BRIAN, HU YONGBO, CHASE CHARLES E, FARID BENAYOUD, CALKINS TREVOR LEE, SCHNADERBECK MATTHEW, FRANCIS G FANG, PESANT MARC, CHRIST WILLIAM, CAMPAGNA SILVIO, ZHU XIAOJIE, WILKIE GORDON, LEWIS BRYAN M
Year of Publication 17.08.2017
Get full text
Year of Publication 17.08.2017
Patent
INTERMEDIATES FOR PREPARATION OF HALICHONDRIN B ANALOGS
AUSTAD BRIAN, HU YONGBO, CHASE CHARLES E, FARID BENAYOUD, CALKINS TREVOR LEE, SCHNADERBECK MATTHEW, FRANCIS G FANG, PESANT MARC, CHRIST WILLIAM, CAMPAGNA SILVIO, ZHU XIAOJIE, WILKIE GORDON, LEWIS BRYAN M
Year of Publication 20.10.2016
Get full text
Year of Publication 20.10.2016
Patent
INTERMEDIATES FOR PREPARATION OF ANALOGS OF HALICHONDRIN B
AUSTAD BRIAN, HU YONGBO, CHASE CHARLES E, FARID BENAYOUD, CALKINS TREVOR LEE, SCHNADERBECK MATTHEW, FRANCIS G FANG, PESANT MARC, CHRIST WILLIAM, CAMPAGNA SILVIO, ZHU XIAOJIE, WILKIE GORDON, LEWIS BRYAN M
Year of Publication 02.04.2015
Get full text
Year of Publication 02.04.2015
Patent
ANTI-WOLBACHIA PYRIDO[2,3-d]PYRIMIDINECOMPOUNDS
Ward, Stephen A, O'Neil, Paul M, Benayoud, Farid, Taylor, Mark J, Hong, Weiqian David
Year of Publication 02.11.2023
Get full text
Year of Publication 02.11.2023
Patent
Anti-Wolbachia pyrido[2,3-d]pyrimidine compounds
Ward, Stephen A, Benayoud, Farid, Taylor, Mark J, O'Neill, Paul M, Hong, Weiqian David
Year of Publication 06.12.2022
Get full text
Year of Publication 06.12.2022
Patent
INTERMEDIATES FOR THE PREPARATION OF ANALOGS OF HALICHONDRIN B
BENAYOUD, FARID, CALKINS, TREVOR LEE, CHASE, CHARLES E, CHRIST, WILLIAM
Year of Publication 12.02.2019
Get full text
Year of Publication 12.02.2019
Patent
Fluorinated Synthons: Reactivity of 1-RF-Epoxy Ethers with Lewis Acids
Begue, Jean-Pierre, Benayoud, Farid, Bonnet-Delpon, Daniele
Published in Journal of organic chemistry (01.08.1995)
Published in Journal of organic chemistry (01.08.1995)
Get full text
Journal Article
Intermediates for the preparation of halichondrin B
Chase, Charles E, Christ, William, Calkins, Trevor Lee, BENAYOUD, Farid, FANG, Francis G
Year of Publication 28.02.2020
Get full text
Year of Publication 28.02.2020
Patent