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Published in PloS one (21.10.2016)
Published in PloS one (21.10.2016)
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CCX559 is a potent, orally-administered small molecule PD-L1 inhibitor that induces anti-tumor immunity
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Published in PloS one (07.06.2023)
Published in PloS one (07.06.2023)
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Correction: Characterization of Pharmacologic and Pharmacokinetic Properties of CCX168, a Potent and Selective Orally Administered Complement 5a Receptor Inhibitor, Based on Preclinical Evaluation and Randomized Phase 1 Clinical Study
Bekker, Pirow, Dairaghi, Daniel, Seitz, Lisa, Leleti, Manmohan, Wang, Yu, Ertl, Linda, Baumgart, Trageen, Shugarts, Sarah, Lohr, Lisa, Dang, Ton, Miao, Shichang, Zeng, Yibin, Fan, Pingchen, Zhang, Penglie, Johnson, Daniel, Powers, Jay, Jaen, Juan, Charo, Israel, Schall, Thomas J
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Published in PloS one (04.01.2019)
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Discovery of a novel melanin concentrating hormone receptor 1 (MCHR1) antagonist with reduced hERG inhibition
Mihalic, Jeffrey T., Fan, Pingchen, Chen, Xiaoqi, Chen, Xi, Fu, Ying, Motani, Alykhan, Liang, Lingming, Lindstrom, Michelle, Tang, Liang, Chen, Jin-Long, Jaen, Juan, Dai, Kang, Li, Leping
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
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Discovery of a novel series of melanin-concentrating hormone receptor 1 antagonists for the treatment of obesity
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Published in Bioorganic & medicinal chemistry letters (01.12.2011)
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
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Discovery and characterization of a potent and selective antagonist of melanin-concentrating hormone receptor 2
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Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
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Stereoselective Synthesis of a MCHr1 Antagonist
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The synthesis and SAR of novel diarylsulfone 11β-HSD1 inhibitors
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Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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Substituted indoloquinolines as new antifungal agents
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Structure−Activity Relationships of the Antimalarial Agent Artemisinin. 3. Total Synthesis of (+)-13-Carbaartemisinin and Related Tetra- and Tricyclic Structures
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Published in Journal of medicinal chemistry (26.04.1996)
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Abstract 1274: CCX559 is a potent orally-administered small molecule PD-L1 inhibitor that induces anti-tumor immunity
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Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Abstract 5693: Anti-tumor effect of orally available small molecule PD-L1 inhibitors in a murine model of colon adenocarcinoma
Li, Shijie "Chris", Vilalta, Marta, Ertl, Linda S., Wang, Yu, Zeng, Yibin, Fan, Pingchen, Lange, Christopher, McMurtrie, Darren, Yang, Ju, Lui, Rebecca, Ong, Ryan, Chhina, Vicky, Kumamoto, Alice, Yau, Simon, Dang, Ton, Easterday, Ashton, Liu, Shirley, Singh, Rajinder, Charo, Israel, Schall, Thomas J., Zhang, Penglie
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Year of Publication 31.10.2023
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Li, Zhihong, Wang, Xianghong, Eksterowicz, John, Gribble, Michael W, Alba, Grace Q, Ayres, Merrill, Carlson, Timothy J, Chen, Ada, Chen, Xiaoqi, Cho, Robert, Connors, Richard V, DeGraffenreid, Michael, Deignan, Jeffrey T, Duquette, Jason, Fan, Pingchen, Fisher, Benjamin, Fu, Jiasheng, Huard, Justin N, Kaizerman, Jacob, Keegan, Kathleen S, Li, Cong, Li, Kexue, Li, Yunxiao, Liang, Lingming, Liu, Wen, Lively, Sarah E, Lo, Mei-Chu, Ma, Ji, McMinn, Dustin L, Mihalic, Jeffrey T, Modi, Kriti, Ngo, Rachel, Pattabiraman, Kanaka, Piper, Derek E, Queva, Christophe, Ragains, Mark L, Suchomel, Julia, Thibault, Steve, Walker, Nigel, Wang, Xiaodong, Wang, Zhulun, Wanska, Malgorzata, Wehn, Paul M, Weidner, Margaret F, Zhang, Alex J, Zhao, Xiaoning, Kamb, Alexander, Wickramasinghe, Dineli, Dai, Kang, McGee, Lawrence R, Medina, Julio C
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Published in Journal of medicinal chemistry (24.04.2014)
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