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Published in Nature communications (05.10.2020)
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Published in Journal of medicinal chemistry (23.10.2008)
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A GIPR antagonist conjugated to GLP-1 analogues promotes weight loss with improved metabolic parameters in preclinical and phase 1 settings
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Published in Nature metabolism (01.02.2024)
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Published in Organic letters (19.02.2010)
Published in Organic letters (19.02.2010)
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Published in Drug metabolism and disposition (01.10.2019)
Published in Drug metabolism and disposition (01.10.2019)
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Engineering Antibody Reactivity for Efficient Derivatization to Generate NaV1.7 Inhibitory GpTx‑1 Peptide–Antibody Conjugates
Biswas, Kaustav, Nixey, Thomas E, Murray, Justin K, Falsey, James R, Yin, Li, Liu, Hantao, Gingras, Jacinthe, Hall, Brian E, Herberich, Brad, Holder, Jerry Ryan, Li, Hongyan, Ligutti, Joseph, Lin, Min-Hwa Jasmine, Liu, Dong, Soriano, Brian D, Soto, Marcus, Tran, Linh, Tegley, Christopher M, Zou, Anrou, Gunasekaran, Kannan, Moyer, Bryan D, Doherty, Liz, Miranda, Les P
Published in ACS chemical biology (15.09.2017)
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Published in ACS chemical biology (19.04.2019)
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위 저해 펩타이드 수용체(GIPR)에 대한 길항제에 접합된 GLP-1 수용체 작용제를 사용하여 대사 장애를 치료 또는 개선하는 방법
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Year of Publication 28.07.2011
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METHOD OF TREATING OR AMELIORATING METABOLIC DISORDERS USING GLP-1 RECEPTOR AGONISTS CONJUGATED TO ANTAGONISTS FOR GASTRIC INHIBITORY PEPTIDE RECEPTOR (GIPR)
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