Enantiospecific inhibition of emesis induced by nicotine in the house musk shrew (Suncus murinus) by the neurokinin sub(1) (NK sub(1)) receptor antagonist CP-99,994
Tattersall, F D, Rycroft, W, Marmont, N, Cascieri, M, Hill, R G, Hargreaves, R J
Published in Neuropharmacology (01.01.1995)
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Published in Neuropharmacology (01.01.1995)
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Tachykinin NK sub(1) receptor antagonists act centrally to inhibit emesis induced by the chemotherapeutic agent cisplatin in ferrets
Tattersall, F D, Rycroft, W, Francis, B, Pearce, D, Merchant, K, MacLeod, A M, Ladduwahetty, T, Keown, L, Swain, C
Published in Neuropharmacology (01.01.1996)
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Published in Neuropharmacology (01.01.1996)
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Structural optimization affording 2-(R)-1-((R)-3,5-bis(trifluoromethyl)phenylethoxy)-3-(S)-(4-fluoro)phenyl-4-(3- oxo-1,2,4-triazol-5-yl)methylmorpholine, a potent, orally active, long-acting morpholine acetal human NK-1 receptor antagonist
HALE, J. J, MILLS, S. G, EIERMANN, G, TSOU, N. N, TATTERSALL, F. D, RUPNIAK, N. M. J, WILLIAMS, A. R, RYCROFT, W, HARGREAVES, R, MACINTYRE, D. E, MACCOSS, M, FINKE, P. E, CASCIERI, M. A, SADOWSKI, S, BER, E, CHICCHI, G. G, KURTZ, M, METZGER, J
Published in Journal of medicinal chemistry (1998)
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Published in Journal of medicinal chemistry (1998)
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Novel lactam NK1 antagonists with anti-emetic activity
HOLLINGWORTH, Gregory J, CARLSON, Emma J, KURTZ, Marc M, RYCROFT, Wayne, TATTERSALL, F. David, TSAO, Kwei-Lan, SWAIN, Christopher J, CASTRO, José L, CHICCHI, Gary G, CLARK, Natalie, COOPER, Laura C, DIRAT, Olivier, DI SALVO, Jerry, ELLIOTT, Jason M, KILBURN, Ruth
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
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N -Heteroaryl-2-phenyl-3-(benzyloxy)piperidines: A Novel Class of Potent Orally Active Human NK 1 Antagonists
Ladduwahetty, T., Baker, R., Cascieri, M. A., Chambers, M. S., Haworth, K., Keown, L. E., MacIntyre, D. E., Metzger, J. M., Owen, S., Rycroft, W., Sadowski, S., Seward, E. M., Shepheard, S. L., Swain, C. J., Tattersall, F. D., Watt, A. P., Williamson, D. W., Hargreaves, R. J.
Published in Journal of medicinal chemistry (01.01.1996)
Published in Journal of medicinal chemistry (01.01.1996)
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Spirocyclic NK1 antagonists II: [4.5]-Spiroethers
WILLIAMS, Brian J, CASCIERI, Margaret A, CHICCHI, Gary G, HARRISON, Timothy, OWENS, Andrew P, OWEN, Simon N, RUPNIAK, Nadia M. J, TATTERSALL, David F, WILLIAMS, Angela, SWAIN, Christopher J
Published in Bioorganic & medicinal chemistry letters (07.10.2002)
Published in Bioorganic & medicinal chemistry letters (07.10.2002)
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Imidazo[1,2-a]pyrimidines as functionally selective GABA sub(A) ligands
Blackaby, Wesley P, Atack, John R, Bromidge, Frances, Castro, Jose L, Goodacre, Simon C, Hallett, David J, Lewis, Richard T, Marshall, George R, Pike, Andrew, Smith, Alison J, Street, Leslie J, Tattersall, David FD, Wafford, Keith A
Published in Bioorganic & medicinal chemistry letters (01.01.2006)
Published in Bioorganic & medicinal chemistry letters (01.01.2006)
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