In silico drug discovery of SIRT2 inhibitors from natural source as anticancer agents
Ibrahim, Mahmoud A. A., Abdeljawaad, Khlood A. A., Roshdy, Eslam, Mohamed, Dina E. M., Ali, Taha F. S., Gabr, Gamal A., Jaragh-Alhadad, Laila A., Mekhemer, Gamal A. H., Shawky, Ahmed M., Sidhom, Peter A., Abdelrahman, Alaa H. M.
Published in Scientific reports (07.02.2023)
Published in Scientific reports (07.02.2023)
Get full text
Journal Article
Combination of an Oxindole Derivative with (-)-β-Elemene Alters Cell Death Pathways in FLT3/ITD + Acute Myeloid Leukemia Cells
Alanazi, Jowaher, Bender, Onur, Dogan, Rumeysa, Malik, Jonaid Ahmad, Atalay, Arzu, Ali, Taha F S, Beshr, Eman A M, Shawky, Ahmed M, Aly, Omar M, Alqahtani, Yasir Nasser H, Anwar, Sirajudheen
Published in Molecules (Basel, Switzerland) (01.07.2023)
Published in Molecules (Basel, Switzerland) (01.07.2023)
Get full text
Journal Article
The First Pentacyclic Triterpenoid Gypsogenin Derivative Exhibiting Anti-ABL1 Kinase and Anti-chronic Myelogenous Leukemia Activities
Ciftci, Halil Ibrahim, Ozturk, Safiye Emirdag, Ali, Taha F. S., Radwan, Mohamed O., Tateishi, Hiroshi, Koga, Ryoko, Ocak, Zeynep, Can, Mustafa, Otsuka, Masami, Fujita, Mikako
Published in Biological & pharmaceutical bulletin (01.04.2018)
Published in Biological & pharmaceutical bulletin (01.04.2018)
Get full text
Journal Article
Discovery and Anticancer Screening of Novel Oxindole-Based Derivative Bearing Pyridyl Group as Potent and Selective Dual FLT3/CDK2 Kinase Inhibitor
Soudi, Aya, Bender, Onur, Celik, Ismail, El-Hafeez, Amer Ali Abd, Dogan, Rumeysa, Atalay, Arzu, Elkaeed, Eslam B, Alsfouk, Aisha A, Abdelhafez, Elshimaa M N, Aly, Omar M, Sippl, Wolfgang, Ali, Taha F S
Published in Pharmaceuticals (Basel, Switzerland) (01.05.2024)
Published in Pharmaceuticals (Basel, Switzerland) (01.05.2024)
Get full text
Journal Article
In Vitro and In Silico Evaluation of Anticancer Activity of New Indole-Based 1,3,4-Oxadiazoles as EGFR and COX-2 Inhibitors
Sever, Belgin, Altıntop, Mehlika Dilek, Özdemir, Ahmet, Akalın Çiftçi, Gülşen, Ellakwa, Doha E, Tateishi, Hiroshi, Radwan, Mohamed O, Ibrahim, Mahmoud A A, Otsuka, Masami, Fujita, Mikako, Ciftci, Halil I, Ali, Taha F S
Published in Molecules (Basel, Switzerland) (07.11.2020)
Published in Molecules (Basel, Switzerland) (07.11.2020)
Get full text
Journal Article
Design, Synthesis, and Biological Evaluation of Novel 1,3,4-Thiadiazole Derivatives as Potential Antitumor Agents against Chronic Myelogenous Leukemia: Striking Effect of Nitrothiazole Moiety
Altıntop, Mehlika Dilek, Ciftci, Halil Ibrahim, Radwan, Mohamed O, Sever, Belgin, Kaplancıklı, Zafer Asım, Ali, Taha F S, Koga, Ryoko, Fujita, Mikako, Otsuka, Masami, Özdemir, Ahmet
Published in Molecules (Basel, Switzerland) (27.12.2017)
Published in Molecules (Basel, Switzerland) (27.12.2017)
Get full text
Journal Article
Novel Inhibitor for Downstream Targeting of Transforming Growth Factor-β Signaling to Suppress Epithelial to Mesenchymal Transition and Cell Migration
Toma, Tsugumasa, Tateishi, Hiroshi, Kawakami, Kensaku, Ali, Taha F S, Kamo, Masahiro, Monde, Kazuaki, Nakashima, Yuta, Fujita, Mikako, Otsuka, Masami
Published in International journal of molecular sciences (02.05.2022)
Published in International journal of molecular sciences (02.05.2022)
Get full text
Journal Article
Antiproliferative S -Trityl-l-Cysteine -Derived Compounds as SIRT2 Inhibitors: Repurposing and Solubility Enhancement
Radwan, Mohamed O, Ciftci, Halil I, Ali, Taha F S, Ellakwa, Doha E, Koga, Ryoko, Tateishi, Hiroshi, Nakata, Akiko, Ito, Akihiro, Yoshida, Minoru, Okamoto, Yoshinari, Fujita, Mikako, Otsuka, Masami
Published in Molecules (Basel, Switzerland) (10.09.2019)
Published in Molecules (Basel, Switzerland) (10.09.2019)
Get full text
Journal Article
New Multi-Targeted Antiproliferative Agents: Design and Synthesis of IC261-Based Oxindoles as Potential Tubulin, CK1 and EGFR Inhibitors
Fareed, Momen R, Shoman, Mai E, Hamed, Mohammed I A, Badr, Mohamed, Bogari, Hanin A, Elhady, Sameh S, Ibrahim, Tarek S, Abuo-Rahma, Gamal El-Din A, Ali, Taha F S
Published in Pharmaceuticals (Basel, Switzerland) (30.10.2021)
Published in Pharmaceuticals (Basel, Switzerland) (30.10.2021)
Get full text
Journal Article
A Dithiol Compound Binds to the Zinc Finger Protein TRAF6 and Suppresses Its Ubiquitination
Koga, Ryoko, Radwan, Mohamed O., Ejima, Tomohiko, Kanemaru, Yosuke, Tateishi, Hiroshi, Ali, Taha F. S., Ciftci, Halil Ibrahim, Shibata, Yuri, Taguchi, Yuu, Inoue, Jun‐ichiro, Otsuka, Masami, Fujita, Mikako
Published in ChemMedChem (07.12.2017)
Published in ChemMedChem (07.12.2017)
Get full text
Journal Article
Discovery of Azaindolin-2-One as a Dual Inhibitor of GSK3β and Tau Aggregation with Potential Neuroprotective Activity
Ali, Taha F S, Ciftci, Halil I, Radwan, Mohamed O, Roshdy, Eslam, Shawky, Ahmed M, Abourehab, Mohammed A S, Tateishi, Hiroshi, Otsuka, Masami, Fujita, Mikako
Published in Pharmaceuticals (Basel, Switzerland) (31.03.2022)
Published in Pharmaceuticals (Basel, Switzerland) (31.03.2022)
Get full text
Journal Article
Design and synthesis of new dihydropyrimidine/sulphonamide hybrids as promising anti-inflammatory agents via dual mPGES-1/5-LOX inhibition
Al-Wahaibi, Lamya H, Elshamsy, Ali M, Ali, Taha F S, Youssif, Bahaa G M, Bräse, S, Abdel-Aziz, Mohamed, El-Koussi, Nawal A
Published in Frontiers in chemistry (2024)
Published in Frontiers in chemistry (2024)
Get full text
Journal Article
Design and Synthesis of New Dihydropyrimidine Derivatives with a Cytotoxic Effect as Dual EGFR/VEGFR‑2 Inhibitors
Al-Wahaibi, Lamya H., Elshamsy, Ali M., Ali, Taha F. S., Youssif, Bahaa G. M., Bräse, Stefan, Abdel-Aziz, Mohamed, El-Koussi, Nawal A.
Published in ACS omega (13.08.2024)
Published in ACS omega (13.08.2024)
Get full text
Journal Article
Design, Synthesis and Biological Evaluation of Pentacyclic Triterpene Derivatives: Optimization of Anti-ABL Kinase Activity
I Ciftci, Halil, O Radwan, Mohamed, E Ozturk, Safiye, Ulusoy, N Gokce, Sozer, Ece, E Ellakwa, Doha, Ocak, Zeynep, Can, Mustafa, F S Ali, Taha, I Abd-Alla, Howaida, Yayli, Nurettin, Tateishi, Hiroshi, Otsuka, Masami, Fujita, Mikako
Published in Molecules (Basel, Switzerland) (30.09.2019)
Published in Molecules (Basel, Switzerland) (30.09.2019)
Get full text
Journal Article
An antifibrotic compound that ameliorates hyperglycaemia and fat accumulation in cell and HFD mouse models
Toma, Tsugumasa, Miyakawa, Nobukazu, Arakaki, Yuiichi, Watanabe, Takuro, Nakahara, Ryosei, Ali, Taha F S, Biswas, Tanima, Todaka, Mikio, Kondo, Tatsuya, Fujita, Mikako, Otsuka, Masami, Araki, Eiichi, Tateishi, Hiroshi
Published in Diabetologia (09.09.2024)
Published in Diabetologia (09.09.2024)
Get full text
Journal Article
The protective role of two oxindole derivatives is mediated by modulating NLRP3/caspase-1 and PI3K/AKT pathways in a preclinical animal model of hepatic ischemia reperfusion injury
Eldafashi, Nardeen, Waaz, Shaimaa, Ali, Taha F.S., Zaki, Marco Y.W., Nazmy, Maiiada Hassan, Fathy, Moustafa
Published in Life sciences (1973) (01.09.2024)
Published in Life sciences (1973) (01.09.2024)
Get full text
Journal Article
Structure activity study of S-trityl-cysteamine dimethylaminopyridine derivatives as SIRT2 inhibitors: Improvement of SIRT2 binding and inhibition
Radwan, Mohamed O., Ciftci, Halil I., Ali, Taha F.S., Koga, Ryoko, Tateishi, Hiroshi, Nakata, Akiko, Ito, Akihiro, Yoshida, Minoru, Fujita, Mikako, Otsuka, Masami
Published in Bioorganic & medicinal chemistry letters (01.10.2020)
Published in Bioorganic & medicinal chemistry letters (01.10.2020)
Get full text
Journal Article