Optimization of the dipeptide motifs in the PSMA ligands linker structure: synthesis and in vitro evaluation
Uspenskaya, Anastasiia A., Nimenko, Ekaterina A., Shafikov, Radik R., Zyk, Nikolay Y., Evteev, Sergei A., Dashkova, Natalia S., Ivanenkov, Yan A., Majouga, Alexander G., Skvortsov, Dmitry A., Garanina, Anastasiia S., Beloglazkina, Elena K., Machulkin, Aleksei E.
Published in Medicinal chemistry research (2023)
Published in Medicinal chemistry research (2023)
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Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atom
Zyk, Nikolai Y., Ber, Anton P., Nimenko, Ekaterina A., Shafikov, Radik R., Evteev, Sergei A., Petrov, Stanislav A., Uspenskaya, Anastasia A., Dashkova, Natalia S., Ivanenkov, Yan A., Skvortsov, Dmitry A., Beloglazkina, Elena K., Majouga, Alexander G., Machulkin, Aleksei E.
Published in Bioorganic & medicinal chemistry letters (01.09.2022)
Published in Bioorganic & medicinal chemistry letters (01.09.2022)
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New Small-Molecule Glycoconjugates of Docetaxel and GalNAc for Targeted Delivery to Hepatocellular Carcinoma
Petrov, Rostislav A, Mefedova, Sofiia R, Yamansarov, Emil Yu, Maklakova, Svetlana Yu, Grishin, Dmitrii A, Lopatukhina, Elena V, Burenina, Olga Y, Lopukhov, Anton V, Kovalev, Sergey V, Timchenko, Yury V, Ondar, Evgenia E, Ivanenkov, Yan A, Evteev, Sergei A, Vaneev, Alexander N, Timoshenko, Roman V, Klyachko, Natalia L, Erofeev, Alexander S, Gorelkin, Petr V, Beloglazkina, Elena K, Majouga, Alexander G
Published in Molecular pharmaceutics (04.01.2021)
Published in Molecular pharmaceutics (04.01.2021)
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Discovery of Bivalent GalNAc-Conjugated Betulin as a Potent ASGPR-Directed Agent against Hepatocellular Carcinoma
Yamansarov, Emil Yu, Lopatukhina, Elena V, Evteev, Sergei A, Skvortsov, Dmitry A, Lopukhov, Anton V, Kovalev, Sergey V, Vaneev, Alexander N, Shkil’, Dmitry O, Akasov, Roman A, Lobov, Alexander N, Naumenko, Victor A, Pavlova, Ekaterina N, Ryabaya, Oxana O, Burenina, Olga Yu, Ivanenkov, Yan A, Klyachko, Natalia L, Erofeev, Alexander S, Gorelkin, Petr V, Beloglazkina, Elena K, Majouga, Alexander G
Published in Bioconjugate chemistry (21.04.2021)
Published in Bioconjugate chemistry (21.04.2021)
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Synthesis and Evaluation of New Trivalent Ligands for Hepatocyte Targeting via the Asialoglycoprotein Receptor
Reshitko, Galina S, Yamansarov, Emil Yu, Evteev, Sergei A, Lopatukhina, Elena V, Shkil’, Dmitry O, Saltykova, Irina V, Lopukhov, Anton V, Kovalev, Sergey V, Lobov, Alexander N, Kislyakov, Ivan V, Burenina, Olga Yu, Klyachko, Natalia L, Garanina, Anastasiia S, Dontsova, Olga A, Ivanenkov, Yan A, Erofeev, Alexander S, Gorelkin, Peter V, Beloglazkina, Elena K, Majouga, Alexander G
Published in Bioconjugate chemistry (20.05.2020)
Published in Bioconjugate chemistry (20.05.2020)
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AlphaFold for a medicinal chemist: tool or toy?
Ivanenkov, Ya. A., Evteev, S. A., Malyshev, A. S., Terentiev, V. A., Bezrukov, D. S., Ereshchenko, A. V., Korzhenevskaya, A. A., Zagribelnyy, B. A., Shegai, P. V., Kaprin, A. D.
Published in Russian chemical reviews (01.01.2024)
Published in Russian chemical reviews (01.01.2024)
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Synthesis of allobetulin-based asialoglycoprotein receptor-targeted glycoconjugates
Seleznev, Egor I., Yamansarov, Emil Yu, Lopatukhina, Elena V., Lopuhov, Anton V., Skvortsov, Dmitry A., Evteev, Sergei A., Yamansarova, Elvira T., Adelgareeva, Amina Yu, Klyachko, Natalia L., Beloglazkina, Elena K., Ivanenkov, Yan A., Majouga, Alexander G.
Published in Mendeleev communications (01.09.2019)
Published in Mendeleev communications (01.09.2019)
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