Discovery of a Novel Inhaled PI3Kδ Inhibitor for the Treatment of Respiratory Diseases
Erra, Montse, Taltavull, Joan, Bernal, Francisco Javier, Caturla, Juan Francisco, Carrascal, Marta, Pagès, Lluís, Mir, Marta, Espinosa, Sònia, Gràcia, Jordi, Domínguez, María, Sabaté, Mar, Paris, Stéphane, Maldonado, Mónica, Hernández, Begoña, Bravo, Mónica, Calama, Elena, Miralpeix, Montserrat, Lehner, Martin D, Calbet, Marta
Published in Journal of medicinal chemistry (08.11.2018)
Published in Journal of medicinal chemistry (08.11.2018)
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Journal Article
Discovery of novel quaternary ammonium derivatives of (3R)-quinuclidinyl amides as potent and long acting muscarinic antagonists
Prat, Maria, Antonia Buil, Maria, Dolors Fernandez, Maria, Tort, Laia, Manuel Monleon, Juan, Casals, Gaspar, Ferrer, Manuel, Castro, Jordi, Gavalda, Amadeu, Miralpeix, Montserrat, Ramos, Israel, Vilella, Dolors, Maria Huerta, Josep, Espinosa, Sonia, Hernandez, Begono, Segarra, Victor, Cordoba, Monica
Published in Bioorganic & medicinal chemistry letters (15.04.2015)
Published in Bioorganic & medicinal chemistry letters (15.04.2015)
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Journal Article
Discovery of novel quaternary ammonium derivatives of (3 R)-quinuclidinyl carbamates as potent and long acting muscarinic antagonists
Prat, Maria, Buil, María Antonia, Fernández, Maria Dolors, Castro, Jordi, Monleón, Juan Manuel, Tort, Laia, Casals, Gaspar, Ferrer, Manuel, Huerta, Josep Maria, Espinosa, Sònia, López, Manuel, Segarra, Victor, Gavaldà, Amadeu, Miralpeix, Montserrat, Ramos, Israel, Vilella, Dolors, González, Marisa, Córdoba, Mònica, Cárdenas, Alvaro, Antón, Francisca, Beleta, Jorge, Ryder, Hamish
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
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Journal Article
Ets-1 transcription is required in tissue factor driven microvessel formation and stabilization
Arderiu, Gemma, Peña, Esther, Aledo, Rosa, Espinosa, Sonia, Badimon, Lina
Published in Angiogenesis (London) (01.12.2012)
Published in Angiogenesis (London) (01.12.2012)
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Journal Article
Setup and validation of shake-flask procedures for the determination of partition coefficients (logD) from low drug amounts
Andrés, Axel, Rosés, Martí, Ràfols, Clara, Bosch, Elisabeth, Espinosa, Sonia, Segarra, Víctor, Huerta, Josep M.
Published in European journal of pharmaceutical sciences (30.08.2015)
Published in European journal of pharmaceutical sciences (30.08.2015)
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Journal Article
Retention of ionizable compounds in high-performance liquid chromatography
Espinosa, Sonia, Bosch, Elisabeth, Rosés, Martı́
Published in Journal of Chromatography A (01.07.2002)
Published in Journal of Chromatography A (01.07.2002)
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Journal Article
Effect of propylene glycol on the skin penetration of drugs
Carrer, Victor, Alonso, Cristina, Pont, Mercè, Zanuy, Miriam, Córdoba, Mònica, Espinosa, Sonia, Barba, Clara, Oliver, Marc A., Martí, Meritxell, Coderch, Luisa
Published in Archives of Dermatological Research (01.07.2020)
Published in Archives of Dermatological Research (01.07.2020)
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Journal Article
Prediction of the skin permeability of topical drugs using in silico and in vitro models
Alonso, Cristina, Carrer, Víctor, Espinosa, Sonia, Zanuy, Miriam, Córdoba, Mònica, Vidal, Bernat, Domínguez, María, Godessart, Núria, Coderch, Luisa, Pont, Mercè
Published in European journal of pharmaceutical sciences (01.08.2019)
Published in European journal of pharmaceutical sciences (01.08.2019)
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Journal Article
Abediterol (LAS100977), an inhaled long-acting β2-adrenoceptor agonist, has a fast association rate and long residence time at receptor
Ramos, Israel, Aparici, Mònica, Letosa, Maria, Puig, Carlos, Gavaldà, Amadeu, Huerta, Josep Maria, Espinosa, Sonia, Vilella, Dolors, Miralpeix, Montserrat
Published in European journal of pharmacology (15.01.2018)
Published in European journal of pharmacology (15.01.2018)
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Journal Article
Retention of ionizable compounds on high-performance liquid chromatography
Bosch, Elisabeth, Espinosa, Sonia, Rosés, Martı́
Published in Journal of Chromatography A (01.10.1998)
Published in Journal of Chromatography A (01.10.1998)
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Journal Article
Abediterol (LAS100977), an inhaled long-acting β 2 -adrenoceptor agonist, has a fast association rate and long residence time at receptor
Ramos, Israel, Aparici, Mònica, Letosa, Maria, Puig, Carlos, Gavaldà, Amadeu, Huerta, Josep Maria, Espinosa, Sonia, Vilella, Dolors, Miralpeix, Montserrat
Published in European journal of pharmacology (15.01.2018)
Published in European journal of pharmacology (15.01.2018)
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Journal Article
Discovery of Novel Quaternary Ammonium Derivatives of (3R)-Quinuclidinol Esters as Potent and Long-Acting Muscarinic Antagonists with Potential for Minimal Systemic Exposure after Inhaled Administration: Identification of (3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane Bromide (Aclidinium Bromide)
Prat, María, Fernández, Dolors, Buil, M. Antonia, Crespo, María I, Casals, Gaspar, Ferrer, Manuel, Tort, Laia, Castro, Jordi, Monleón, Juan M, Gavaldà, Amadeu, Miralpeix, Montserrat, Ramos, Israel, Doménech, Teresa, Vilella, Dolors, Antón, Francisca, Huerta, Josep M, Espinosa, Sonia, López, Manuel, Sentellas, Sonia, González, Marisa, Albertí, Joan, Segarra, Victor, Cárdenas, Alvaro, Beleta, Jorge, Ryder, Hamish
Published in Journal of medicinal chemistry (27.08.2009)
Published in Journal of medicinal chemistry (27.08.2009)
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Journal Article
Retention of ionizable compounds in high-performance liquid chromatography: IX. Modelling retention in reversed-phase liquid chromatography as a function of pH and solvent composition with acetonitrile–water mobile phases
Espinosa, Sonia, Bosch, Elisabeth, Rosés, Martı́
Published in Journal of Chromatography A (15.02.2002)
Published in Journal of Chromatography A (15.02.2002)
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Journal Article