Search Results - "Erik Laurini" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Identification of RC-33 as a potent and selective sigma 1 receptor agonist potentiating NGF-induced neurite outgrowth in PC12 cells. Part 2: g-Scale synthesis, physicochemical characterization and in vitro metabolic stability

Identification of RC-33 as a potent and selective sigma 1 receptor agonist potentiating NGF-induced neurite outgrowth in PC12 cells. Part 2: g-Scale synthesis, physicochemical characterization and in vitro metabolic stability

by Rossi, Daniela, Marra, Annamaria, Picconi, Pietro, Serra, Massimo, Catenacci, Laura, Sorrenti, Milena, Laurini, Erik, Fermeglia, Maurizio, Pricl, Sabrina, Brambilla, Stefania, Almirante, Nicoletta, Peviani, Marco, Curti, Daniela, Collina, Simona
Published in Bioorganic & medicinal chemistry (01.05.2013)

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Journal Article

Rigidity versus Flexibility: Is This an Issue in σ1 Receptor Ligand Affinity and Activity?

Rigidity versus Flexibility: Is This an Issue in σ1 Receptor Ligand Affinity and Activity?

by Weber, Frauke, Brune, Stefanie, Börgel, Frederik, Lange, Carsten, Korpis, Katharina, Bednarski, Patrick J, Laurini, Erik, Fermeglia, Maurizio, Pricl, Sabrina, Schepmann, Dirk, Wünsch, Bernhard
Published in Journal of medicinal chemistry (09.06.2016)

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Journal Article

Impact of siRNA Overhangs for Dendrimer-Mediated siRNA Delivery and Gene Silencing

Impact of siRNA Overhangs for Dendrimer-Mediated siRNA Delivery and Gene Silencing

by Posocco, Paola, Liu, Xiaoxuan, Laurini, Erik, Marson, Domenico, Chen, Chao, Liu, Cheng, Fermeglia, Maurizio, Rocchi, Palma, Pricl, Sabrina, Peng, Ling
Published in Molecular pharmaceutics (05.08.2013)

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Journal Article

Thiazole-Based sigma(1) Receptor Ligands: Diversity by Late-Stage C-H Arylation of Thiazoles, Structure-Affinity and Selectivity Relationships, and Molecular Interactions

Thiazole-Based sigma(1) Receptor Ligands: Diversity by Late-Stage C-H Arylation of Thiazoles, Structure-Affinity and Selectivity Relationships, and Molecular Interactions

by Kokornaczyk, Artur K., Schepmann, Dirk, Yamaguchi, Junichiro, Itami, Kenichiro, Laurini, Erik, Fermeglia, Maurizio, Pricl, Sabrina, Wuensch, Bernhard
Published in ChemMedChem (06.07.2017)

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Journal Article

Improving selectivity preserving affinity: New piperidine-4-carboxamide derivatives as effective sigma-1-ligands

Improving selectivity preserving affinity: New piperidine-4-carboxamide derivatives as effective sigma-1-ligands

by Zampieri, Daniele, Laurini, Erik, Vio, Luciano, Fermeglia, Maurizio, Pricl, Sabrina, Wünsch, Bernhard, Schepmann, Dirk, Mamolo, Maria Grazia
Published in European journal of medicinal chemistry (27.01.2015)

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Journal Article

Copper(II) binding to flexible triethanolamine-core PAMAM dendrimers: a combined experimental/in silico approach

Copper(II) binding to flexible triethanolamine-core PAMAM dendrimers: a combined experimental/in silico approach

by Ottaviani, Maria Francesca, Cangiotti, Michela, Fattori, Alberto, Coppola, Concetta, Posocco, Paola, Laurini, Erik, Liu, Xiaoxuan, Liu, Cheng, Fermeglia, Maurizio, Peng, Ling, Pricl, Sabrina
Published in Physical chemistry chemical physics : PCCP (14.01.2014)

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Journal Article

Molecular and functional characterization of a new 3' end KIT juxtamembrane deletion in a duodenal GIST treated with neoadjuvant Imatinib

Molecular and functional characterization of a new 3' end KIT juxtamembrane deletion in a duodenal GIST treated with neoadjuvant Imatinib

by Perfetti, Vittorio, Laurini, Erik, Aulić, Suzana, Fermeglia, Maurizio, Riboni, Roberta, Lucioni, Marco, Dallera, Elena, Delfanti, Sara, Pugliese, Luigi, Latteri, Francesco Saverio, Pietrabissa, Andrea, Pricl, Sabrina
Published in Oncotarget (22.08.2017)

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Journal Article

Structure–activity relationship study of dendritic polyglycerolamines for efficient siRNA transfection

Structure–activity relationship study of dendritic polyglycerolamines for efficient siRNA transfection

by Mehrabadi, Fatemeh Sheikhi, Hirsch, Ole, Zeisig, Reiner, Posocco, Paola, Laurini, Erik, Pricl, Sabrina, Haag, Rainer, Kemmner, Wolfgang, Calderon, Marcelo
Published in RSC advances (01.09.2015)

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Journal Article

Electrostatic binding of polyanions using self-assembled multivalent (SAMul) ligand displays - structure-activity effects on DNA/heparin bindingElectronic supplementary information (ESI) available: Full synthetic methods and characterisation data, assay and modelling methodologies, further experimental data from binding assays, DLS and TEM. See DOI: 10.1039/c5sc04801j

Electrostatic binding of polyanions using self-assembled multivalent (SAMul) ligand displays - structure-activity effects on DNA/heparin bindingElectronic supplementary information (ESI) available: Full synthetic methods and characterisation data, assay and modelling methodologies, further experimental data from binding assays, DLS and TEM. See DOI: 10.1039/c5sc04801j

by Fechner, Loryn E, Albanyan, Buthaina, Vieira, Vânia M. P, Laurini, Erik, Posocco, Paola, Pricl, Sabrina, Smith, David K
Year of Publication 21.06.2016

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Journal Article

Emergence of highly-ordered hierarchical nanoscale aggregates on electrostatic binding of self-assembled multivalent (SAMul) cationic micelles with polyanionic heparin

Emergence of highly-ordered hierarchical nanoscale aggregates on electrostatic binding of self-assembled multivalent (SAMul) cationic micelles with polyanionic heparin

by Vieira, Vania M P, Liljeström, Ville, Posocco, Paola, Laurini, Erik, Pricl, Sabrina, Kostiainen, Mauri A, Smith, David K
Published in Journal of materials chemistry. B, Materials for biology and medicine (2017)

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Journal Article

Through the open door: Preferential binding of dasatinib to the active form of BCR-ABL unveiled by in silico experiments

Through the open door: Preferential binding of dasatinib to the active form of BCR-ABL unveiled by in silico experiments

by Laurini, Erik, Posocco, Paola, Fermeglia, Maurizio, Gibbons, Don L., Quintás-Cardama, Alfonso, Pricl, Sabrina
Published in Molecular oncology (01.10.2013)

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Journal Article

Rigidity versus Flexibility: Is This an Issue in σ 1 Receptor Ligand Affinity and Activity?

Rigidity versus Flexibility: Is This an Issue in σ 1 Receptor Ligand Affinity and Activity?

by Weber, Frauke, Brune, Stefanie, Börgel, Frederik, Lange, Carsten, Korpis, Katharina, Bednarski, Patrick J., Laurini, Erik, Fermeglia, Maurizio, Pricl, Sabrina, Schepmann, Dirk, Wünsch, Bernhard
Published in Journal of medicinal chemistry (09.06.2016)

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Journal Article

Synthesis, Pharmacological Evaluation, and σ1 Receptor Interaction Analysis of Hydroxyethyl Substituted Piperazines

Synthesis, Pharmacological Evaluation, and σ1 Receptor Interaction Analysis of Hydroxyethyl Substituted Piperazines

by Weber, Frauke, Brune, Stefanie, Korpis, Katharina, Bednarski, Patrick J, Laurini, Erik, Dal Col, Valentina, Pricl, Sabrina, Schepmann, Dirk, Wünsch, Bernhard
Published in Journal of medicinal chemistry (10.04.2014)

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Journal Article

Abstract 2900: Sigma-1 receptor control tumorigenic and stem cell-like phenotype in human cancers

Abstract 2900: Sigma-1 receptor control tumorigenic and stem cell-like phenotype in human cancers

by Civenni, Gianluca, Marchetti, Martina, Pandit, Shusil, Monte, Celeste De, Sereni, Federica, Merulla, Jessica, Zadic, Sabrina, Losa, Marco, Allegrini, Sara, Albino, Domenico, Mapelli, Sarah, Laurini, Erik, Wunsch, Bernhard, Pricl, Sabrina, Carbone, Giuseppina M., Catapano, Carlo V.
Published in Cancer research (Chicago, Ill.) (01.07.2017)

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Journal Article

Thiazole-Based σ 1 Receptor Ligands: Diversity by Late-Stage C-H Arylation of Thiazoles, Structure-Affinity and Selectivity Relationships, and Molecular Interactions

Thiazole-Based σ 1 Receptor Ligands: Diversity by Late-Stage C-H Arylation of Thiazoles, Structure-Affinity and Selectivity Relationships, and Molecular Interactions

by Kokornaczyk, Artur K, Schepmann, Dirk, Yamaguchi, Junichiro, Itami, Kenichiro, Laurini, Erik, Fermeglia, Maurizio, Pricl, Sabrina, Wünsch, Bernhard
Published in ChemMedChem (06.07.2017)

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Journal Article

Fluorinated PET Tracers for Molecular Imaging of σ1 Receptors in the Central Nervous System

Fluorinated PET Tracers for Molecular Imaging of σ1 Receptors in the Central Nervous System

by Weber, Frauke, Brust, Peter, Laurini, Erik, Pricl, Sabrina, Wünsch, Bernhard
Published in Sigma Receptors: Their Role in Disease and As Therapeutic Targets (2017)

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Book Chapter

Thiazole-Based [sigma]1 Receptor Ligands: Diversity by Late-Stage C-H Arylation of Thiazoles, Structure-Affinity and Selectivity Relationships, and Molecular Interactions

Thiazole-Based [sigma]1 Receptor Ligands: Diversity by Late-Stage C-H Arylation of Thiazoles, Structure-Affinity and Selectivity Relationships, and Molecular Interactions

by Kokornaczyk, Artur K, Schepmann, Dirk, Yamaguchi, Junichiro, Itami, Kenichiro, Laurini, Erik, Fermeglia, Maurizio, Pricl, Sabrina, Wunsch, Bernhard
Published in ChemMedChem (01.07.2017)

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Journal Article

Electrostatic binding of polyanions using self-assembled multivalent (SAMul) ligand displays – structure–activity effects on DNA/heparin binding† †Electronic supplementary information (ESI) available: Full synthetic methods and characterisation data, assay and modelling methodologies, further experimental data from binding assays, DLS and TEM. See DOI: 10.1039/c5sc04801j

Electrostatic binding of polyanions using self-assembled multivalent (SAMul) ligand displays – structure–activity effects on DNA/heparin binding† †Electronic supplementary information (ESI) available: Full synthetic methods and characterisation data, assay and modelling methodologies, further experimental data from binding assays, DLS and TEM. See DOI: 10.1039/c5sc04801j

by Fechner, Loryn E., Albanyan, Buthaina, Vieira, Vânia M. P., Laurini, Erik, Posocco, Paola, Pricl, Sabrina, Smith, David K.
Published in Chemical science (Cambridge) (18.04.2016)

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Journal Article

Synthesis and receptor binding studies of some new arylcarboxamide derivatives as sigma-1 ligands

Synthesis and receptor binding studies of some new arylcarboxamide derivatives as sigma-1 ligands

by Zampieri, Daniele, Laurini, Erik, Vio, Luciano, Golob, Samuel, Fermeglia, Maurizio, Pricl, Sabrina, Mamolo, Maria Grazia
Published in Bioorganic & medicinal chemistry letters (15.02.2014)

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Journal Article

Correction: Targeting Hsp27/eIF4E interaction with phenazine compound: a promising alternative for castration-resistant prostate cancer treatment

Correction: Targeting Hsp27/eIF4E interaction with phenazine compound: a promising alternative for castration-resistant prostate cancer treatment

by Ziouziou, Hajer, Andrieu, Claudia, Laurini, Erik, Karaki, Sara, Fermeglia, Maurizio, Oueslati, Ridha, Taieb, David, Camplo, Michel, Siri, Olivier, Pricl, Sabrina, Katsogiannou, Maria, Rocchi, Palma
Published in Oncotarget (19.06.2018)

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Journal Article

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