Abstract 812: New c-KIT mutations in GISTs: Bad for good
Laurini, Erik, Aulic, Suzana, Marson, Domenico, Fermeglia, Maurizio, Riboni, Roberta, Lucioni, Marco, Dellera, Elena, Alessiani, Mario, Perfetti, Vittorio, Pricl, Sabrina
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Quinolizidine-Derived Lucanthone and Amitriptyline Analogues Endowed with Potent Antileishmanial Activity
Tonelli, Michele, Sparatore, Anna, Basilico, Nicoletta, Cavicchini, Loredana, Parapini, Silvia, Tasso, Bruno, Laurini, Erik, Pricl, Sabrina, Boido, Vito, Sparatore, Fabio
Published in Pharmaceuticals (Basel, Switzerland) (25.10.2020)
Published in Pharmaceuticals (Basel, Switzerland) (25.10.2020)
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Journal Article
Chemoenzymatic synthesis of 2,6-disubstituted tetrahydropyrans with high σ1 receptor affinity, antitumor and analgesic activity
Kopp, Nicole, Civenni, Gianluca, Marson, Domenico, Laurini, Erik, Pricl, Sabrina, Catapano, Carlo V., Humpf, Hans-Ulrich, Almansa, Carmen, Nieto, Francisco Rafael, Schepmann, Dirk, Wünsch, Bernhard
Published in European journal of medicinal chemistry (05.07.2021)
Published in European journal of medicinal chemistry (05.07.2021)
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Synthesis and biological evaluation of new aryl-alkyl(alkenyl)-4-benzylpiperidines, novel Sigma Receptor (SR) modulators, as potential anticancer-agents
Rui, Marta, Rossi, Daniela, Marra, Annamaria, Paolillo, Mayra, Schinelli, Sergio, Curti, Daniela, Tesei, Anna, Cortesi, Michela, Zamagni, Alice, Laurini, Erik, Pricl, Sabrina, Schepmann, Dirk, Wűnsch, Bernhard, Urban, Ernst, Pace, Vittorio, Collina, Simona
Published in European journal of medicinal chemistry (29.11.2016)
Published in European journal of medicinal chemistry (29.11.2016)
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Journal Article
Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives
Briguglio, Irene, Loddo, Roberta, Laurini, Erik, Fermeglia, Maurizio, Piras, Sandra, Corona, Paola, Giunchedi, Paolo, Gavini, Elisabetta, Sanna, Giuseppina, Giliberti, Gabriele, Ibba, Cristina, Farci, Pamela, La Colla, Paolo, Pricl, Sabrina, Carta, Antonio
Published in European journal of medicinal chemistry (13.11.2015)
Published in European journal of medicinal chemistry (13.11.2015)
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Bioimaging: Surface Charge of Supramolecular Nanosystems for In Vivo Biodistribution: A MicroSPECT/CT Imaging Study (Small 37/2020)
Ding, Ling, Lyu, Zhenbin, Louis, Beatrice, Tintaru, Aura, Laurini, Erik, Marson, Domenico, Zhang, Mengjie, Shao, Wanxuan, Jiang, Yifan, Bouhlel, Ahlem, Balasse, Laure, Garrigue, Philippe, Mas, Eric, Giorgio, Suzanne, Iovanna, Juan, Huang, Yuanyu, Pricl, Sabrina, Guillet, Benjamin, Peng, Ling
Published in Small (Weinheim an der Bergstrasse, Germany) (01.09.2020)
Published in Small (Weinheim an der Bergstrasse, Germany) (01.09.2020)
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Journal Article
Antifungal and antimycobacterial activity of 1-(3,5-diaryl-4,5-dihydro-1H-pyrazol-4-yl)-1H-imidazole derivatives
ZAMPIERI, Daniele, GRAZIAMAMOLO, Maria, LAURINI, Erik, SCIALINO, Giuditta, BANFI, Elena, VIO, Luciano
Published in Bioorganic & medicinal chemistry (15.04.2008)
Published in Bioorganic & medicinal chemistry (15.04.2008)
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Journal Article
Chiral recognition at self-assembled multivalent (SAMul) nanoscale interfaces - enantioselectivity in polyanion bindingElectronic supplementary information (ESI) available: Full synthesis and characterisation data, assay methods, additional assay data and imaging. See DOI: 10.1039/c6cc04470k
Chan, Ching W, Laurini, Erik, Posocco, Paola, Pricl, Sabrina, Smith, David K
Year of Publication 18.08.2016
Year of Publication 18.08.2016
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Journal Article
Pd-Catalyzed Direct C–H Bond Functionalization of Spirocyclic σ1 Ligands: Generation of a Pharmacophore Model and Analysis of the Reverse Binding Mode by Docking into a 3D Homology Model of the σ1 Receptor
Meyer, Christina, Schepmann, Dirk, Yanagisawa, Shuichi, Yamaguchi, Junichiro, Dal Col, Valentina, Laurini, Erik, Itami, Kenichiro, Pricl, Sabrina, Wünsch, Bernhard
Published in Journal of medicinal chemistry (27.09.2012)
Published in Journal of medicinal chemistry (27.09.2012)
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Journal Article
Electrostatic binding of polyanions using self-assembled multivalent (SAMul) ligand displays - structure-activity effects on DNA/heparin binding
Fechner, Loryn E., Albanyan, Buthaina, Vieira, Vania M. P., Laurini, Erik, Posocco, Paola, Pricl, Sabrina, Smith, David K.
Published in Chemical science (Cambridge) (01.01.2016)
Published in Chemical science (Cambridge) (01.01.2016)
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Journal Article
Self-Assembled Nanomicelles as Curcumin Drug Delivery Vehicles: Impact on Solitary Fibrous Tumor Cell Protein Expression and Viability
Dagrada, Gianpaolo, Rupel, Katia, Zacchigna, Serena, Tamborini, Elena, Pilotti, Silvana, Cavalleri, Adalberto, Fechner, Loryn E, Laurini, Erik, Smith, David K, Brich, Silvia, Pricl, Sabrina
Published in Molecular pharmaceutics (01.10.2018)
Published in Molecular pharmaceutics (01.10.2018)
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Journal Article
Homology Model and Docking-Based Virtual Screening for Ligands of the σ 1 Receptor
Laurini, Erik, Col, Valentina Dal, Mamolo, Maria Grazia, Zampieri, Daniele, Posocco, Paola, Fermeglia, Maurizio, Vio, Luciano, Pricl, Sabrina
Published in ACS medicinal chemistry letters (10.11.2011)
Published in ACS medicinal chemistry letters (10.11.2011)
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Journal Article
Synthesis, Biological Evaluation, and Three-Dimensional in Silico Pharmacophore Model for sigma(1) Receptor Ligands Based on a Series of Substituted Benzo[d]oxazol-2(3H)-one Derivatives
Zampieri, Daniele, Mamolo, Maria Grazia, Laurini, Erik, Florio, Chiara, Zanette, Caterina, Fermeglia, Maurizio, Posocco, Paola, Paneni, Maria Silvia, Pricl, Sabrina, Vio, Luciano
Published in Journal of medicinal chemistry (10.09.2009)
Published in Journal of medicinal chemistry (10.09.2009)
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Journal Article
Synthesis, Pharmacological Evaluation, and sigma(1) Receptor Interaction Analysis of Hydroxyethyl Substituted Piperazines
Weber, Frauke, Brune, Stefanie, Korpis, Katharina, Bednarski, Patrick J., Laurini, Erik, Dal Col, Valentina, Pricl, Sabrina, Schepmann, Dirk, Wuensch, Bernhard
Published in Journal of medicinal chemistry (10.04.2014)
Published in Journal of medicinal chemistry (10.04.2014)
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Journal Article
β‐Catenin in desmoid‐type fibromatosis: deep insights into the role of T41A and S45F mutations on protein structure and gene expression
Colombo, Chiara, Belfiore, Antonino, Paielli, Nicholas, De Cecco, Loris, Canevari, Silvana, Laurini, Erik, Fermeglia, Maurizio, Pricl, Sabrina, Verderio, Paolo, Bottelli, Stefano, Fiore, Marco, Stacchiotti, Silvia, Palassini, Elena, Gronchi, Alessandro, Pilotti, Silvana, Perrone, Federica
Published in Molecular oncology (01.11.2017)
Published in Molecular oncology (01.11.2017)
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