Development of a Continuous Photochemical Bromination/Alkylation Sequence En Route to AMG 423
Quasdorf, Kyle, Murray, James I, Nguyen, Hanh, Silva Elipe, Maria V, Ericson, Ari, Kircher, Eric, Guan, Lianxiu, Caille, Seb
Published in Organic process research & development (18.02.2022)
Published in Organic process research & development (18.02.2022)
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Journal Article
A Continuous Process for Manufacturing Apremilast. Part I: Process Development and Intensification by Utilizing Flow Chemistry Principles
Hsieh, Hsiao-Wu, Cohen, Carolyn M., Griffin, Daniel J., Ananthoji, Padmini, Avci, Nadide Hazal, Brown, Derek B., Ericson, Ari, Fostinis, James D., Irfan, Muhammad, Langille, Neil, Lovette, Michael A., Murray, James I., Spada, Simone, Thiel, Oliver R., Aiello, Frankie, Daou, Joseph, Goudas-Salomon, Nicole, Pan, Ende, Sarkar, Nandini, Wimalasinghe, Rasangi, Wu, Zufan Steven, Zeng, Alicia, Beaver, Matthew G.
Published in Organic process research & development (17.05.2024)
Published in Organic process research & development (17.05.2024)
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Journal Article
오메캄티브 메카빌의 합성
MURRAY JAMES, CAILLE SEBASTIEN, QUASDORF KYLE, NGUYEN HANNAH, SILVA ELIPE MARIA VICTORIA, ERICSON ARI ELIZABETH
Year of Publication 15.01.2024
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Year of Publication 15.01.2024
Patent
Implementing Continuous Manufacturing for the Final Methylation Step in the AMG 397 Process to Deliver Key Quality Attributes
Tom, Janine K, Achmatowicz, Michal M, Beaver, Matthew G, Colyer, John, Ericson, Ari, Hwang, Tsang-Lin, Jiao, Nancy, Langille, Neil F, Liu, Min, Lovette, Michael A, Sangodkar, Rahul P, Sharvan Kumar, Srividya, Spada, Simone, Perera, Damith, Sheeran, Jillian, Campbell, Kiersten, Doherty, Timothy, Ford, David D, Fang, Yuan-Qing, Rossi, Emiliano, Santoni, Gabriella, Cui, Sheng, Walker, Shawn D
Published in Organic process research & development (19.03.2021)
Published in Organic process research & development (19.03.2021)
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Journal Article
거대환식 MCL-1 저해제 중간체의 폐환 합성
CHERNEY ALAN H, SMITH AUSTIN G, TEDROW JASON S, ST PIERRE GABRIELLE, ERICSON ARI, BEAVER MATTHEW G, BAUCOM KYLE D, COLYER JOHN T, ROOSEN PHILIPP C, SANGODKAR RAHUL P, LOVETTE MICHAEL A, CUI SHENG, THIEL OLIVER RALF, HUANG LIANG, MILBURN ROBERT RONALD
Year of Publication 13.01.2023
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Year of Publication 13.01.2023
Patent
SYNTHESIS OF OMECAMTIV MECARBIL
MURRAY, James, NGUYEN, Hannah, CAILLE, Sebastien, QUASDORF, Kyle, SILVA ELIPE, Maria Victoria, ERICSON, Ari Elizabeth
Year of Publication 17.01.2024
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Year of Publication 17.01.2024
Patent
Synthesis of omecamtiv mecarbil
MURRAY James, CAILLE Sebastien, QUASDORF Kyle, NGUYEN Hannah, ERICSON Ari Elizabeth, SILVA ELIPE Maria Victoria
Year of Publication 01.11.2023
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Year of Publication 01.11.2023
Patent
SYNTHESIS OF OMECAMTIV MECARBIL
MURRAY, James, NGUYEN, Hannah, CAILLE, Sebastien, QUASDORF, Kyle, SILVA ELIPE, Maria Victoria, ERICSON, Ari Elizabeth
Year of Publication 19.10.2023
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Year of Publication 19.10.2023
Patent
Synthesis of omecamtiv mecarbil
Ericson, Ari Elizabeth, Quasdorf, Kyle, Silva Elipe, Maria Victoria, Murray, James, Caille, Sebastien, Nguyen, Hannah
Year of Publication 18.07.2023
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Year of Publication 18.07.2023
Patent
SYNTHESIS OF OMECAMTIV MECARBIL
MURRAY, James, NGUYEN, Hannah, CAILLE, Sebastien, QUASDORF, Kyle, SILVA ELIPE, Maria Victoria, ERICSON, Ari Elizabeth
Year of Publication 27.10.2022
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Year of Publication 27.10.2022
Patent
SYNTHESIS OF OMECAMTIV MECARBIL
MURRAY, James, NGUYEN, Hannah, CAILLE, Sebastien, QUASDORF, Kyle, SILVA ELIPE, Maria Victoria, ERICSON, Ari Elizabeth
Year of Publication 22.09.2022
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Year of Publication 22.09.2022
Patent
SYNTHESIS OF OMECAMTIV MECARBIL
MURRAY, JAMES, CAILLE, SEBASTIEN, SILVA ELIPE, MARIA VICTORIA, QUASDORF, KYLE, ERICSON, ARI ELIZABETH, NGUYEN, HANNAH
Year of Publication 15.09.2022
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Year of Publication 15.09.2022
Patent
SYNTHESIS OF OMECAMTIV MECARBIL
MURRAY, James, NGUYEN, Hannah, CAILLE, Sebastien, QUASDORF, Kyle, SILVA ELIPE, Maria Victoria, ERICSON, Ari Elizabeth
Year of Publication 15.09.2022
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Year of Publication 15.09.2022
Patent
Ring closing synthesis of macrocyclic Mcl-1 inhibitor intermediates
CHERNEY, Alan H, SANGODKAR, Rahul P, CUI, Sheng, THIEL, Oliver Ralf, ROOSEN, Philipp C, ST-PIERRE, Gabrielle, MILBURN, Robert Ronald, TEDROW, Jason S, COLYER, John T, ERICSON, Ari, SMITH, Austin G, HUANG, Liang, BEAVER, Matthew G, BAUCOM, Kyle D, LOVETTE, Michael A
Year of Publication 13.06.2024
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Year of Publication 13.06.2024
Patent
Ring Closing Synthesis of Macrocyclic MCL-1 Inhibitor Intermediates
CHERNEY, Alan H, SANGODKAR, Rahul P, CUI, Sheng, THIEL, Oliver Ralf, ROOSEN, Philipp C, ST-PIERRE, Gabrielle, MILBURN, Robert Ronald, TEDROW, Jason S, COLYER, John T, ERICSON, Ari, SMITH, Austin G, HUANG, Liang, BEAVER, Matthew G, BAUCOM, Kyle D, LOVETTE, Michael A
Year of Publication 01.06.2023
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Year of Publication 01.06.2023
Patent
RING CLOSING SYNTHESIS OF MACROCYCLIC MCL-1 INHIBITOR INTERMEDIATES
CHERNEY, Alan H, SANGODKAR, Rahul P, CUI, Sheng, THIEL, Oliver Ralf, ROOSEN, Philipp C, ST-PIERRE, Gabrielle, MILBURN, Robert Ronald, TEDROW, Jason S, COLYER, John T, ERICSON, Ari, SMITH, Austin G, HUANG, Liang, BEAVER, Matthew G, BAUCOM, Kyle D, LOVETTE, Michael A
Year of Publication 15.03.2023
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Year of Publication 15.03.2023
Patent
RING CLOSING SYNTHESIS OF MACROCYCLIC MCL-1 INHIBITOR INTERMEDIATES
CHERNEY, Alan H, SANGODKAR, Rahul P, CUI, Sheng, THIEL, Oliver Ralf, ROOSEN, Philipp C, ST-PIERRE, Gabrielle, MILBURN, Robert Ronald, TEDROW, Jason S, COLYER, John T, ERICSON, Ari, BEAVER, Matthew G, SMITH, Austin G, HUANG, Liang, BAUCOM, Kyle D, LOVETTE, Michael A
Year of Publication 23.01.2023
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Year of Publication 23.01.2023
Patent
Síntesis de omecamtiv mecarbil
MURRAY, James, NGUYEN, Hannah, CAILLE, Sebastien, QUASDORF, Kyle, SILVA ELIPE, Maria Victoria, ERICSON, Ari Elizabeth
Year of Publication 02.02.2024
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Year of Publication 02.02.2024
Patent
Ring closing synthesis of macrocyclic Mcl-1 inhibitor intermediates
CHERNEY, Alan H, SANGODKAR, Rahul P, CUI, Sheng, THIEL, Oliver Ralf, ROOSEN, Philipp C, ST-PIERRE, Gabrielle, MILBURN, Robert Ronald, TEDROW, Jason S, COLYER, John T, ERICSON, Ari, SMITH, Austin G, HUANG, Liang, BEAVER, Matthew G, BAUCOM, Kyle D, LOVETTE, Michael A
Year of Publication 15.12.2022
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Year of Publication 15.12.2022
Patent
SYNTHESIS OF OMECAMTIV MECARBIL
MURRAY James, CAILLE Sebastien, QUASDORF Kyle, NGUYEN Hannah, ERICSON Ari Elizabeth, SILVA ELIPE Maria Victoria
Year of Publication 24.11.2023
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Year of Publication 24.11.2023
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