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Published in Bioorganic & medicinal chemistry letters (15.07.2005)
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The Discovery of Setileuton, a Potent and Selective 5-Lipoxygenase Inhibitor
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Published in ACS medicinal chemistry letters (08.07.2010)
Published in ACS medicinal chemistry letters (08.07.2010)
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Substituted coumarins as potent 5-lipoxygenase inhibitors
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Published in Bioorganic & medicinal chemistry letters (01.05.2006)
Published in Bioorganic & medicinal chemistry letters (01.05.2006)
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Published in Bioorganic & medicinal chemistry letters (15.04.2011)
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
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Solid-phase analogue synthesis of caspase-3 inhibitors via palladium-catalyzed amination of 3-bromopyrazinones
Isabel, Elise, Aspiotis, Renee, Black, W. Cameron, Colucci, John, Fortin, Réjean, Giroux, André, Grimm, Erich L., Han, Yongxin, Mellon, Christophe, Nicholson, Donald W., Rasper, Dita M., Renaud, Johanne, Roy, Sophie, Tam, John, Tawa, Paul, Vaillancourt, John P., Xanthoudakis, Steven, Zamboni, Robert J.
Published in Bioorganic & medicinal chemistry letters (15.03.2007)
Published in Bioorganic & medicinal chemistry letters (15.03.2007)
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A straightforward approach to the synthesis of the tricyclic core of taxol
Wang, Zhaoyin, Warder, Scott E, Perrier, Helene, Grimm, Erich L, Bernstein, Michael A, Ball, Richard G
Published in Journal of organic chemistry (01.05.1993)
Published in Journal of organic chemistry (01.05.1993)
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Discovery of novel aspartyl ketone dipeptides as potent and selective caspase-3 inhibitors
Han, Yongxin, Giroux, André, Grimm, Erich L., Aspiotis, Renée, Francoeur, Sébastien, Bayly, Christopher I., Mckay, Daniel J., Roy, Sophie, Xanthoudakis, Steve, Vaillancourt, John P., Rasper, Dita M., Tam, John, Tawa, Paul, Thornberry, Nancy A., Paterson, Erin P., Garcia-Calvo, Margarita, Becker, Joseph W., Rotonda, Jennifer, Nicholson, Donald W., Zamboni, Robert J.
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
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3,4-Diaryl-5-hydroxyfuranones: highly selective inhibitors of cyclooxygenase-2 with aqueous solubility
Black, W.Cameron, Brideau, Christine, Chan, Chi-Chung, Charleson, Stella, Cromlish, Wanda, Gordon, Robert, Grimm, Erich L., Hughes, Gregory, Leger, Serge, Li, Chun-Sing, Riendeau, Denis, Thérien, Michel, Wang, Zhaoyin, Xu, Li-Jing, Prasit, Petpiboon
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
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Lipophilic versus hydrogen-bonding effect in P3 on potency and selectivity of valine aspartyl ketones as caspase 3 inhibitors
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Published in Bioorganic & medicinal chemistry letters (01.09.2005)
Published in Bioorganic & medicinal chemistry letters (01.09.2005)
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Nicotinyl aspartyl ketones as inhibitors of caspase-3
Isabel, Elise, Black, W.Cameron, Bayly, Christopher I, Grimm, Erich L, Janes, Marc K, McKay, Daniel J, Nicholson, Donald W, Rasper, Dita M, Renaud, Johanne, Roy, Sophie, Tam, John, Thornberry, Nancy A, Vaillancourt, John P, Xanthoudakis, Steven, Zamboni, Robert
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
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Solid phase synthesis of selective caspase-3 peptide inhibitors
GRIMM, Erich L, ROY, Bruno, VAILLANCOURT, John P, XANTHOUDAKIS, Steven, ZAMBONI, Robert J, ASPIOTIS, Renee, BAYLY, Christopher I, NICHOLSON, Donald W, RASPER, Dita M, RENAUD, Johanne, ROY, Sophie, TAM, John, TAWA, Paul
Published in Bioorganic & medicinal chemistry (01.03.2004)
Published in Bioorganic & medicinal chemistry (01.03.2004)
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Inhibitors of the inducible microsomal prostaglandin E 2 synthase (mPGES-1) derived from MK-886
Riendeau, Denis, Aspiotis, Renee, Ethier, Diane, Gareau, Yves, Grimm, Erich L., Guay, Jocelyne, Guiral, Sébastien, Juteau, Hélène, Mancini, Joseph A., Méthot, Nathalie, Rubin, Joel, Friesen, Richard W.
Published in Bioorganic & medicinal chemistry letters (15.07.2005)
Published in Bioorganic & medicinal chemistry letters (15.07.2005)
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THE UNSYMMETRICAL SILAKETAL AS A NEUTRAL, REMOVABLE TETHER FOR EFFECTING INTRAMOLECULAR DIELS-ALDER REACTIONS
GILLARD, JW, FORTIN, R, GRIMM, EL, MAILLARD, M, TJEPKEMA, M, BERNSTEIN, MA, GLASER, R
Published in Tetrahedron letters (25.02.1991)
Published in Tetrahedron letters (25.02.1991)
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Journal Article
Lipophilic versus hydrogen-bonding effect in P 3 on potency and selectivity of valine aspartyl ketones as caspase 3 inhibitors
Mellon, Christophe, Aspiotis, Reneé, Black, Cameron W., Bayly, Christopher I., Grimm, Erich L., Giroux, André, Han, Yongxin, Isabel, Elise, McKay, Daniel J., Nicholson, Donald W., Rasper, Dita M., Roy, Sophie, Tam, John, Thornberry, Nancy A., Vaillancourt, John P., Xanthoudakis, Steven, Zamboni, Robert
Published in Bioorganic & medicinal chemistry letters (01.09.2005)
Published in Bioorganic & medicinal chemistry letters (01.09.2005)
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