Analysis of the crystal structure of an active MCM hexamer
Miller, Justin M, Arachea, Buenafe T, Epling, Leslie B, Enemark, Eric J
Published in eLife (29.09.2014)
Published in eLife (29.09.2014)
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A conserved MCM single-stranded DNA binding element is essential for replication initiation
Froelich, Clifford A, Kang, Sukhyun, Epling, Leslie B, Bell, Stephen P, Enemark, Eric J
Published in eLife (01.04.2014)
Published in eLife (01.04.2014)
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Journal Article
Discovery of (4-Pyrazolyl)-2-aminopyrimidines as Potent and Selective Inhibitors of Cyclin-Dependent Kinase 2
Hummel, Joshua R., Xiao, Kai-Jiong, Yang, Jeffrey C., Epling, Leslie B., Mukai, Ken, Ye, Qinda, Xu, Meizhong, Qian, Dingquan, Huo, Lu, Weber, Michael, Roman, Valerie, Lo, Yvonne, Drake, Katherine, Stump, Kristine, Covington, Maryanne, Kapilashrami, Kanishk, Zhang, Guofeng, Ye, Min, Diamond, Sharon, Yeleswaram, Swamy, Macarron, Ricardo, Deller, Marc C., Wee, Susan, Kim, Sunkyu, Wang, Xiaozhao, Wu, Liangxing, Yao, Wenqing
Published in Journal of medicinal chemistry (22.02.2024)
Published in Journal of medicinal chemistry (22.02.2024)
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Discovery of Potent and Selective Inhibitors of Wild-Type and Gatekeeper Mutant Fibroblast Growth Factor Receptor (FGFR) 2/3
Shvartsbart, Artem, Roach, Jeremy J., Witten, Michael R., Koblish, Holly, Harris, Jennifer J., Covington, Maryanne, Hess, Rodrigo, Lin, Luping, Frascella, Michelle, Truong, Lisa, Leffet, Lynn, Conlen, Patricia, Beshad, Elham, Klabe, Ron, Katiyar, Kamna, Kaldon, Laura, Young-Sciame, Ruth, He, Xin, Petusky, Susan, Chen, Kwang-Jong, Horsey, April, Lei, Hsiang-Ting, Epling, Leslie B., Deller, Marc C., Vechorkin, Oleg, Yao, Wenqing
Published in Journal of medicinal chemistry (24.11.2022)
Published in Journal of medicinal chemistry (24.11.2022)
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Abstract 5900: INCB161734: A novel, potent, and orally bioavailable KRAS G12D selective inhibitor demonstrates antitumor activity in KRAS G12D mutant tumors
Farren, Matthew R., Roman, Valerie, Gallion, Alexandra, Allali-Hassani, Abdellah, Sokolsky, Alexander, Kong, Weixi, Smith, Amanda, Wang, Hui, Correa, Gina, Deller, Marc, Epling, Leslie B., Procak, Jessica, Zhang, Guofeng, Pecko, Katherine, Kennedy, Keith, Boer, Jason, Kurzeja-Lipinski, Kerri, Covington, Maryanne, Chen, Kwang-Jong, Wallower, Renee, Rocha, Jennifer, Pan, Rina, Perry, Anthony, Yuska, Brad, Wang, Xiaozhao, Macarron, Ricardo, Kim, Sunkyu
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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