Liver-specific drug targeting by coupling to bile acids
KRAMER, W, WESS, G, MÜLLNER, S, NECKERMANN, G, SCHULZ, S, PETZINGER, E, SCHUBERT, G, BICKEL, M, GIRBIG, F, GUTJAHR, U, KOWALEWSKI, S, BARINGHAUS, K.-H, ENHSEN, A, GLOMBIK, H
Published in The Journal of biological chemistry (15.09.1992)
Published in The Journal of biological chemistry (15.09.1992)
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Journal Article
Synthesis of bile acid - drug conjugates: Potential drug - shuttles for liver specific targeting
Wess, G., Kramer, W., Schubert, G., Enhsen, A., Baringhaus, K.-H., Glombik, H., Müllner, S., Bock, K., Kleine, H., John, M., Neckermann, O., Hoffmann, A.
Published in Tetrahedron letters (29.01.1993)
Published in Tetrahedron letters (29.01.1993)
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Journal Article
Substrate specificity of the ileal and the hepatic Na(+)/bile acid cotransporters of the rabbit. I. Transport studies with membrane vesicles and cell lines expressing the cloned transporters
Kramer, W, Stengelin, S, Baringhaus, K H, Enhsen, A, Heuer, H, Becker, W, Corsiero, D, Girbig, F, Noll, R, Weyland, C
Published in Journal of lipid research (01.09.1999)
Published in Journal of lipid research (01.09.1999)
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Journal Article
Modified bile acids as carriers for peptides and drugs
Kramer, Werner, Wess, Günther, Enhsen, Alfons, Falk, Eugen, Hoffmann, Axel, Neckermann, Georg, Schubert, Gerrit, Urmann, Matthias
Published in Journal of controlled release (05.05.1997)
Published in Journal of controlled release (05.05.1997)
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Journal Article
Conference Proceeding
Intestinal absorption of peptides by coupling to bile acids
KRAMER, W, WESS, G, ENHSEN, A, FALK, E, FRIEDRICH, M, GLOMBIK, H, HOFFMANN, A, PITTIUS, C, URMANN, M, NECKERMANN, G, SCHUBERT, G, FINK, J, GIRBIG, F, GUTJAHR, U, KOWALEWSKI, S, BARINGHAUS, K.-H, BÖGER, G
Published in The Journal of biological chemistry (08.04.1994)
Published in The Journal of biological chemistry (08.04.1994)
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Journal Article
Bile acid derived HMG-CoA reductase inhibitors
Kramer, W, Wess, G, Enhsen, A, Bock, K, Falk, E, Hoffmann, A, Neckermann, G, Gantz, D, Schulz, S, Nickau, L
Published in Biochimica et biophysica acta (29.11.1994)
Published in Biochimica et biophysica acta (29.11.1994)
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Journal Article
PREPARATION OF 3-ALPHA-(OMEGA-AMINOALKOXY) AND 3-BETA-(OMEGA-AMINOALKOXY)-7-ALPHA,12-ALPHA-AMINOALKOXY-DIHYDROXY-5-BETA-CHOLANOIC ACID-ESTERS - VERSATILE SHUTTLES FOR DRUG TARGETING
WESS, G, KRAMER, W, ENHSEN, A, GLOMBIK, H, BARINGHAUS, KH, BOCK, K, KLEINE, H, SCHMITT, W
Published in Tetrahedron letters (29.01.1993)
Published in Tetrahedron letters (29.01.1993)
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Journal Article
Specific Inhibitors of Ileal Bile Acid Transport
Wess, Guenther, Kramer, Werner, Enhsen, Alfons, Glombik, Heiner, Baringhaus, Karl-Heinz, Boeger, Georg, Urmann, Matthias, Bock, Klaus, Kleine, Horst
Published in Journal of medicinal chemistry (01.04.1994)
Published in Journal of medicinal chemistry (01.04.1994)
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Journal Article
Synthesis and Biological Activity of Bile Acid-Derived HMG-CoA Reductase Inhibitors. The Role of 21-Methyl in Recognition of HMG-CoA Reductase and the Ileal Bile Acid Transport System
Wess, Guenther, Kramer, Werner, Han, Xiao Bing, Bock, Klaus, Enhsen, Alfons, Glombik, Heiner, Baringhaus, Karl-Heinz, Boeger, Georg, Urmann, Matthias
Published in Journal of medicinal chemistry (30.09.1994)
Published in Journal of medicinal chemistry (30.09.1994)
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Journal Article
Hepatobiliary transport of hepatic 3-hydroxy-3-methylglutaryl coenzyme A reductase inhibitors conjugated with bile acids
Petzinger, E, Nickau, L, Horz, J A, Schulz, S, Wess, G, Enhsen, A, Falk, E, Baringhaus, K H, Glombik, H, Hoffmann, A
Published in Hepatology (Baltimore, Md.) (01.12.1995)
Published in Hepatology (Baltimore, Md.) (01.12.1995)
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Journal Article
Topological Photoaffinity Labeling of the Rabbit Ileal Na+/Bile‐Salt‐Cotransport System
Kramer, Werner, Wess, Günther, Bewersdorf, Ulrike, Corsiero, Daniel, Girbig, Frank, Weyland, Claudia, Stengelin, Siegfried, Enhsen, Alfons, Bock, Klaus, Kleine, Horst, Dreau, Marie‐Anne, Schäfer, Hans‐Ludwig
Published in European journal of biochemistry (15.10.1997)
Published in European journal of biochemistry (15.10.1997)
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Journal Article
The design and synthesis of a scaffold for combinatorial chemistry based on bile acid
Wess, G, Bock, K, Kleine, H, Kurz, M, Guba, W, Hemmerle, H, LopezCalle, E, Baringhaus, KH, Glombik, H, Enhsen, A, Kramer, W
Published in Angewandte Chemie International Edition (18.10.1996)
Published in Angewandte Chemie International Edition (18.10.1996)
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