Phase I and Pharmacokinetic Study of Farnesyl Protein Transferase Inhibitor R115777 in Advanced Cancer
ZUJEWSKI, J, HORAK, I. D, KOPP, W. C, KOHLER, D. R, CHOW, C, NOONE, M, HAKIM, F. T, LARKIN, G, GRESS, R. E, NUSSENBLATT, R. B, KREMER, A. B, COWAN, K. H, BOL, C. J, WOESTENBORGHS, R, BOWDEN, C, END, D. W, PIOTROVSKY, V. K, CHIAO, J, BELLY, R. T, TODD, A
Published in Journal of clinical oncology (14.02.2000)
Published in Journal of clinical oncology (14.02.2000)
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Journal Article
Characterization of the antitumor effects of the selective farnesyl protein transferase inhibitor R115777 in vivo and in vitro
END, David W, SMETS, Gerda, DEVINE, Ann, WOUTERS, Walter, BOWDEN, Charles, TODD, Alison V, APPLEGATE, Tanya L, FUERY, Caroline J, ANGIBAUD, Patrick, VENET, Marc, SANZ, Gerard, POIGNET, Herve, SKRZAT, Stacy
Published in Cancer research (Chicago, Ill.) (2001)
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Published in Cancer research (Chicago, Ill.) (2001)
Journal Article
Pharmacodynamics and pharmacokinetics of the novel thrombopoietin mimetic peptide RWJ-800088 in humans
Liem-Moolenaar, M, Cerneus, D, Molloy, C J, End, D, Brown, K H, de Kam, M L, Cohen, A F, van Hensbergen, Y, Burggraaf, J
Published in Clinical pharmacology and therapeutics (01.10.2008)
Published in Clinical pharmacology and therapeutics (01.10.2008)
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Journal Article
Clinical and biologic activity of the farnesyltransferase inhibitor R115777 in adults with refractory and relapsed acute leukemias: a phase 1 clinical-laboratory correlative trial
Karp, Judith E., Lancet, Jeffrey E., Kaufmann, Scott H., End, David W., Wright, John J., Bol, Kees, Horak, Ivan, Tidwell, Michael L., Liesveld, Jane, Kottke, Timothy J., Ange, Dawn, Buddharaju, Laxmi, Gojo, Ivana, Highsmith, W. Edward, Belly, Robert T., Hohl, Raymond J., Rybak, Mary Ellen, Thibault, Alain, Rosenblatt, Joseph
Published in Blood (01.06.2001)
Published in Blood (01.06.2001)
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Current status of clinical trials of farnesyltransferase inhibitors
Karp, J E, Kaufmann, S H, Adjei, A A, Lancet, J E, Wright, J J, End, D W
Published in Current opinion in oncology (01.11.2001)
Published in Current opinion in oncology (01.11.2001)
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Journal Article
Experimental studies with liarozole (R 75 251): An antitumoral agent which inhibits retinoic acid breakdown
De Coster, R., Wouters, W., Van Ginckel, R., End, D., Krekels, M., Coene, M.-C., Bowden, C.
Published in Journal of steroid biochemistry and molecular biology (01.09.1992)
Published in Journal of steroid biochemistry and molecular biology (01.09.1992)
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Conference Proceeding
Nerve growth factor-induced decrease in the cell-free phosphorylation of a soluble protein in PC12 cells
End, D, Tolson, N, Hashimoto, S, Guroff, G
Published in The Journal of biological chemistry (25.05.1983)
Published in The Journal of biological chemistry (25.05.1983)
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Phase I Trial and Pharmacokinetic Study of the Farnesyltransferase Inhibitor Tipifarnib in Children With Refractory Solid Tumors or Neurofibromatosis Type I and Plexiform Neurofibromas
WIDEMANN, Brigitte C, SALZER, Wanda L, JAYAPRAKASH, Nalini, ZANNIKOS, Peter, BALIS, Frank M, ARCECI, Robert J, BLANEY, Susan M, FOX, Elizabeth, END, David, GILLESPIE, Andrea, WHITCOMB, Patricia, PALUMBO, Joseph S, PITNEY, Aaron
Published in Journal of clinical oncology (20.01.2006)
Published in Journal of clinical oncology (20.01.2006)
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Journal Article
Farnesyl protein transferase inhibitor ZARNESTRA R115777 - history of a discovery
Venet, Marc, End, David, Angibaud, Patrick
Published in Current topics in medicinal chemistry (01.01.2003)
Published in Current topics in medicinal chemistry (01.01.2003)
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Journal Article
The Farnesyltransferase Inhibitor R115777 Reduces Hypoxia and Matrix Metalloproteinase 2 Expression in Human Glioma Xenograft
DELMAS, Caroline, END, Dave, ROCHAIX, Philippe, FAVRE, Gilles, TOULAS, Christine, COHEN-JONATHAN, Elizabeth
Published in Clinical cancer research (01.12.2003)
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Published in Clinical cancer research (01.12.2003)
Journal Article
Farnesyltransferase inhibitor, R115777, reverses the resistance of human glioma cell lines to ionizing radiation
Delmas, Caroline, Heliez, Christophe, Cohen‐Jonathan, Elizabeth, End, Dave, Bonnet, Jacques, Favre, Gilles, Toulas, Christine
Published in International journal of cancer (01.07.2002)
Published in International journal of cancer (01.07.2002)
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Journal Article
Preclinical Antitumor Activity and Pharmacodynamic Studies with the Farnesyl Protein Transferase Inhibitor R115777 in Human Breast Cancer
KELLAND, Lloyd R, SMITH, Vicki, JOHNSTON, Stephen R. D, VALENTI, Melanie, PATTERSON, Lisa, CLARKE, Paul A, DETRE, Simone, END, Dave, HOWES, Angela J, DOWSETT, Mitch, WORKMAN, Paul
Published in Clinical cancer research (01.11.2001)
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Published in Clinical cancer research (01.11.2001)
Journal Article
A rapid assay for measuring the metabolism of [ 3H]-retinoic acid in cell cultures
Garrabrant, Thomas A., End, David W.
Published in Journal of pharmacological and toxicological methods (01.12.1995)
Published in Journal of pharmacological and toxicological methods (01.12.1995)
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Journal Article
Stimulation of Platelet Production in Healthy Volunteers by a Novel Pegylated Peptide-Based Thrombopoietin (TPO) Receptor Agonist
Cerneus, Dirk, Brown, K., Harris, R., End, D., Molloy, C., Yurkow, E., Koblish, H., Franks, C., Moolenaar, M., Burggraaf, K.
Published in Blood (16.11.2005)
Published in Blood (16.11.2005)
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