Dual EGFR/ErbB-2 inhibitors from novel pyrrolidinyl-acetylenic thieno[3,2- d]pyrimidines
Hubbard, Robert D., Dickerson, Scott H., Emerson, Holly K., Griffin, Robert J., Reno, Michael J., Hornberger, Keith R., Rusnak, David W., Wood, Edgar R., Uehling, David E., Waterson, Alex G.
Published in Bioorganic & medicinal chemistry (01.11.2008)
Published in Bioorganic & medicinal chemistry (01.11.2008)
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Journal Article
Synthesis and stereochemical effects of pyrrolidinyl-acetylenic thieno[3,2- d]pyrimidines as EGFR and ErbB-2 inhibitors
Stevens, Kirk L., Alligood, Krystal J., Alberti, Jennifer G. Badiang, Caferro, Thomas R., Chamberlain, Stanley D., Dickerson, Scott H., Dickson, Hamilton D., Emerson, Holly K., Griffin, Robert J., Hubbard, Robert D., Keith, Barry R., Mullin, Robert J., Petrov, Kimberly G., Gerding, Roseanne M., Reno, Michael J., Rheault, Tara R., Rusnak, David W., Sammond, Douglas M., Smith, Stephon C., Uehling, David E., Waterson, Alex G., Wood, Edgar R.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Discovery and optimization of imidazo[1,2- a]pyridine inhibitors of insulin-like growth factor-1 receptor (IGF-1R)
Emmitte, Kyle A., Wilson, Brian J., Baum, Erich W., Emerson, Holly K., Kuntz, Kevin W., Nailor, Kristen E., Salovich, James M., Smith, Stephon C., Cheung, Mui, Gerding, Roseanne M., Stevens, Kirk L., Uehling, David E., Mook, Robert A., Moorthy, Ganesh S., Dickerson, Scott H., Hassell, Anne M., Anthony Leesnitzer, M., Shewchuk, Lisa M., Groy, Arthur, Rowand, Jason L., Anderson, Kelly, Atkins, Charity L., Yang, Jingsong, Sabbatini, Peter, Kumar, Rakesh
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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Journal Article
2-Pyrimidinyl Pyrazolopyridine Erbb Kinase Inhibitors
UEHLING DAVID E, DICKERSON SCOTT H, WATERSON ALEX G, EMERSON HOLLY K, SAMMOND DOUGLAS M, HARRIS PHILIP A, HUBBARD ROBERT D, STEVENS KIRK L, WILSON JOSEPH W
Year of Publication 28.02.2008
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Year of Publication 28.02.2008
Patent
Diamino-pyrimidines and their use as angiogenesis inhibitors
EMERSON HOLLY K, SAMMOND DOUGLAS M, CHEUNG MUI, CHAMBERLAIN STANLEY D, SEMONES MARCUS, JOHNSON NEIL W, NAILOR KRISTEN E
Year of Publication 20.10.2005
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Year of Publication 20.10.2005
Patent
Crystal structure of liganded cFMS kinase domain
MUSSO DAVID L, SHEWCHUK LISA M, EMERSON HOLLY K, PECKHAM GREGORY E, HOLMES WILLIAM D, CHAMBERLAIN STANLEY D, VEAL JAMES M, HASSELL ANNE M
Year of Publication 11.01.2007
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Year of Publication 11.01.2007
Patent