New Quinoline-Based Heterocycles as Anticancer Agents Targeting Bcl-2
Hamdy, Rania, Elseginy, Samia A, Ziedan, Noha I, Jones, Arwyn T, Westwell, Andrew D
Published in Molecules (Basel, Switzerland) (02.04.2019)
Published in Molecules (Basel, Switzerland) (02.04.2019)
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Journal Article
New 4-phenylcoumarin derivatives as potent 3C protease inhibitors: Design, synthesis, anti-HAV effect and molecular modeling
Kassem, Asmaa F., Batran, Rasha Z., Abbas, Eman M.H., Elseginy, Samia A., Shaheen, Mohamed N.F., Elmahdy, Elmahdy M.
Published in European journal of medicinal chemistry (15.04.2019)
Published in European journal of medicinal chemistry (15.04.2019)
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Journal Article
Design, Synthesis and Evaluation of New Bioactive Oxadiazole Derivatives as Anticancer Agents Targeting Bcl-2
Hamdy, Rania, Elseginy, Samia A, Ziedan, Noha I, El-Sadek, Mohamed, Lashin, Elsaid, Jones, Arwyn T, Westwell, Andrew D
Published in International journal of molecular sciences (26.11.2020)
Published in International journal of molecular sciences (26.11.2020)
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Journal Article
Design, Synthesis and Biological Evaluation of Spiro Cyclohexane-1,2- Quinazoline Derivatives as Potent Dipeptidyl Peptidase IV Inhibitors
Syam, Yasmin M, El-Karim, Somaia S Abd, Nasr, Tamer, Elseginy, Samia A, Anwar, Manal M, Kamel, Mohsen M, Ali, Hanan F
Published in Mini reviews in medicinal chemistry (01.01.2019)
Published in Mini reviews in medicinal chemistry (01.01.2019)
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Journal Article
Synthesis, anticancer effect and molecular modeling of new thiazolylpyrazolyl coumarin derivatives targeting VEGFR-2 kinase and inducing cell cycle arrest and apoptosis
Mohamed, Tahia K., Batran, Rasha Z., Elseginy, Samia A., Ali, Mamdouh M., Mahmoud, Abeer E.
Published in Bioorganic chemistry (01.04.2019)
Published in Bioorganic chemistry (01.04.2019)
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Journal Article
Promising anti-SARS-CoV-2 drugs by effective dual targeting against the viral and host proteases
Elseginy, Samia A., Fayed, Bahgat, Hamdy, Rania, Mahrous, Noura, Mostafa, Ahmed, Almehdi, Ahmed M., S. M. Soliman, Sameh
Published in Bioorganic & medicinal chemistry letters (01.07.2021)
Published in Bioorganic & medicinal chemistry letters (01.07.2021)
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Journal Article
Design, synthesis and molecular modeling of new 4-phenylcoumarin derivatives as tubulin polymerization inhibitors targeting MCF-7 breast cancer cells
Batran, Rasha Z., Kassem, Asmaa F., Abbas, Eman M.H., Elseginy, Samia A., Mounier, Marwa M.
Published in Bioorganic & medicinal chemistry (23.07.2018)
Published in Bioorganic & medicinal chemistry (23.07.2018)
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Journal Article
Critical discovery and synthesis of novel antibacterial and resistance-modifying agents inspired by plant phytochemical defense mechanisms
Soliman, Sameh S.M., Saeed, Balsam Qubais, Elseginy, Samia A., Al-Marzooq, Farah, Ahmady, Islam M., El-Keblawy, Ali A., Hamdy, Rania
Published in Chemico-biological interactions (05.01.2021)
Published in Chemico-biological interactions (05.01.2021)
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Journal Article
Anti-Alzheimer activity of new coumarin-based derivatives targeting acetylcholinesterase inhibition
Kamel, Nahla N, Aly, Hanan F, Fouad, Ghadha I, Abd El-Karim, Somaia S, Anwar, Manal M, Syam, Yasmin M, Elseginy, Samia A, Ahmed, Kawkab A, Booles, Hoda F, Shalaby, Mohamed B, Khalil, Wagdy K. B, Sandhir, Rajat, Deshwal, Sonam, Rizk, Maha Z
Published in RSC advances (15.06.2023)
Published in RSC advances (15.06.2023)
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Journal Article
Design, synthesis, and computational validation of novel compounds selectively targeting HER2-expressing breast cancer
Elseginy, Samia A., Hamdy, Rania, Menon, Varsha, Almehdi, Ahmed M., El-Awady, Raafat, Soliman, Sameh S.M.
Published in Bioorganic & medicinal chemistry letters (15.12.2020)
Published in Bioorganic & medicinal chemistry letters (15.12.2020)
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Journal Article
Discovery of novel benzofuran-based derivatives as acetylcholinesterase inhibitors for the treatment of Alzheimer's disease: Design, synthesis, biological evaluation, molecular docking and 3D-QSAR investigation
Abd El-Karim, Somaia S., Anwar, Manal M., Ahmed, Nesreen S., Syam, Yasmin M., Elseginy, Samia A., Aly, Hanan F., Younis, Eman A., Khalil, Wagdy K.B., Ahmed, Kawkab A., Mohammed, Faten F., Rizk, Maha
Published in European journal of medicinal chemistry (15.11.2023)
Published in European journal of medicinal chemistry (15.11.2023)
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Journal Article
Selective inhibition of Rhizopus eumelanin biosynthesis by novel natural product scaffold-based designs caused significant inhibition of fungal pathogenesis
Soliman, Sameh S M, Hamdy, Rania, Elseginy, Samia A, Gebremariam, Teclegiorgis, Hamoda, Alshaimaa M, Madkour, Mohamed, Venkatachalam, Thenmozhi, Ershaid, Mai N, Mohammad, Mohammad G, Chamilos, Georgios, Ibrahim, Ashraf S
Published in Biochemical journal (17.07.2020)
Published in Biochemical journal (17.07.2020)
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