A Chemoproteomic Approach to Query the Degradable Kinome Using a Multi-kinase Degrader
Huang, Hai-Tsang, Dobrovolsky, Dennis, Paulk, Joshiawa, Yang, Guang, Weisberg, Ellen L., Doctor, Zainab M., Buckley, Dennis L., Cho, Joong-Heui, Ko, Eunhwa, Jang, Jaebong, Shi, Kun, Choi, Hwan Geun, Griffin, James D., Li, Ying, Treon, Steven P., Fischer, Eric S., Bradner, James E., Tan, Li, Gray, Nathanael S.
Published in Cell chemical biology (18.01.2018)
Published in Cell chemical biology (18.01.2018)
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Structure-Guided Development of a Potent and Selective Non-covalent Active-Site Inhibitor of USP7
Lamberto, Ilaria, Liu, Xiaoxi, Seo, Hyuk-Soo, Schauer, Nathan J., Iacob, Roxana E., Hu, Wanyi, Das, Deepika, Mikhailova, Tatiana, Weisberg, Ellen L., Engen, John R., Anderson, Kenneth C., Chauhan, Dharminder, Dhe-Paganon, Sirano, Buhrlage, Sara J.
Published in Cell chemical biology (21.12.2017)
Published in Cell chemical biology (21.12.2017)
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Inhibition of USP10 induces degradation of oncogenic FLT3
Weisberg, Ellen L, Schauer, Nathan J, Yang, Jing, Lamberto, Ilaria, Doherty, Laura, Bhatt, Shruti, Nonami, Atsushi, Meng, Chengcheng, Letai, Anthony, Wright, Renee, Tiv, Hong, Gokhale, Prafulla C, Ritorto, Maria Stella, De Cesare, Virginia, Trost, Matthias, Christodoulou, Alexandra, Christie, Amanda, Weinstock, David M, Adamia, Sophia, Stone, Richard, Chauhan, Dharminder, Anderson, Kenneth C, Seo, Hyuk-Soo, Dhe-Paganon, Sirano, Sattler, Martin, Gray, Nathanael S, Griffin, James D, Buhrlage, Sara J
Published in Nature chemical biology (01.12.2017)
Published in Nature chemical biology (01.12.2017)
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Selective USP7 inhibition elicits cancer cell killing through a p53-dependent mechanism
Schauer, Nathan J, Liu, Xiaoxi, Magin, Robert S, Doherty, Laura M, Chan, Wai Cheung, Ficarro, Scott B, Hu, Wanyi, Roberts, Rebekka M, Iacob, Roxana E, Stolte, Björn, Giacomelli, Andrew O, Perera, Sumner, McKay, Kyle, Boswell, Sarah A, Weisberg, Ellen L, Ray, Arghya, Chauhan, Dharminder, Dhe-Paganon, Sirano, Anderson, Ken C, Griffin, James D, Li, Jianing, Hahn, William C, Sorger, Peter K, Engen, John R, Stegmaier, Kimberly, Marto, Jarrod A, Buhrlage, Sara J
Published in Scientific reports (24.03.2020)
Published in Scientific reports (24.03.2020)
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Discovery of a Potent and Selective DDR1 Receptor Tyrosine Kinase Inhibitor
Kim, Hyung-Gu, Tan, Li, Weisberg, Ellen L, Liu, Feiyang, Canning, Peter, Choi, Hwan Geun, Ezell, Scott A, Wu, Hong, Zhao, Zheng, Wang, Jinhua, Mandinova, Anna, Griffin, James D, Bullock, Alex N, Liu, Qingsong, Lee, Sam W, Gray, Nathanael S
Published in ACS chemical biology (18.10.2013)
Published in ACS chemical biology (18.10.2013)
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The STAT5 inhibitor pimozide decreases survival of chronic myelogenous leukemia cells resistant to kinase inhibitors
Nelson, Erik A., Walker, Sarah R., Weisberg, Ellen, Bar-Natan, Michal, Barrett, Rosemary, Gashin, Laurie B., Terrell, Shariya, Klitgaard, Josephine L., Santo, Loredana, Addorio, Martha R., Ebert, Benjamin L., Griffin, James D., Frank, David A.
Published in Blood (24.03.2011)
Published in Blood (24.03.2011)
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Small molecule inhibition of deubiquitinating enzyme JOSD1 as a novel targeted therapy for leukemias with mutant JAK2
Yang, Jing, Weisberg, Ellen L, Liu, Xiaoxi, Magin, Robert S, Chan, Wai Cheung, Hu, Bin, Schauer, Nathan J, Zhang, Shengzhe, Lamberto, Ilaria, Doherty, Laura, Meng, Chengcheng, Sattler, Martin, Cabal-Hierro, Lucia, Winer, Eric, Stone, Richard, Marto, Jarrod A, Griffin, James D, Buhrlage, Sara J
Published in Leukemia (01.01.2022)
Published in Leukemia (01.01.2022)
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Anti‐SARS‐CoV‐2 activity of targeted kinase inhibitors: Repurposing clinically available drugs for COVID‐19 therapy
Boytz, RuthMabel, Słabicki, Mikołaj, Ramaswamy, Sita, Patten, J. J., Zou, Charles, Meng, Chengcheng, Hurst, Brett L., Wang, Jinhua, Nowak, Radosław P., Yang, Priscilla L., Sattler, Martin, Stone, Richard M., Griffin, James D., Gray, Nathanael S., Gummuluru, Suryaram, Davey, Robert A., Weisberg, Ellen
Published in Journal of medical virology (01.01.2023)
Published in Journal of medical virology (01.01.2023)
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Discovery of N‑(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia
Liang, Xiaofei, Wang, Beilei, Chen, Cheng, Wang, Aoli, Hu, Chen, Zou, Fengming, Yu, Kailin, Liu, Qingwang, Li, Feng, Hu, Zhenquan, Lu, Tingting, Wang, Junjie, Wang, Li, Weisberg, Ellen L, Li, Lili, Xia, Ruixiang, Wang, Wenchao, Ren, Tao, Ge, Jian, Liu, Jing, Liu, Qingsong
Published in Journal of medicinal chemistry (24.01.2019)
Published in Journal of medicinal chemistry (24.01.2019)
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Inhibition of the deubiquitinating enzyme USP47 as a novel targeted therapy for hematologic malignancies expressing mutant EZH2
Yang, Jing, Weisberg, Ellen L, Qi, Shuang, Ni, Wei, Mei, Husheng, Wang, Zuowei, Meng, Chengcheng, Zhang, Shengzhe, Hou, Mingqi, Qi, Ziping, Wang, Aoli, Jiang, Yunyun, Jiang, Zongru, Huang, Tao, Liu, Qingwang, Magin, Robert S, Doherty, Laura, Wang, Wenchao, Liu, Jing, Buhrlage, Sara J, Liu, Qingsong, Griffin, James D
Published in Leukemia (01.04.2022)
Published in Leukemia (01.04.2022)
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Selectively targeting FLT3-ITD mutants over FLT3-wt by a novel inhibitor for acute myeloid leukemia
Wang, Aoli, Hu, Chen, Chen, Cheng, Liang, Xiaofei, Wang, Beilei, Zou, Fengming, Yu, Kailin, Li, Feng, Liu, Qingwang, Qi, Ziping, Wang, Junjie, Wang, Wenliang, Wang, Li, Weisberg, Ellen L, Wang, Wenchao, Li, Lili, Ge, Jian, Xia, Ruixiang, Liu, Jing, Liu, Qingsong
Published in Haematologica (Roma) (01.02.2021)
Published in Haematologica (Roma) (01.02.2021)
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Essential role of the histone lysine demethylase KDM4A in the biology of malignant pleural mesothelioma (MPM)
Lapidot, Moshe, Case, Abigail E, Weisberg, Ellen L, Meng, Chengcheng, Walker, Sarah R, Garg, Swati, Ni, Wei, Podar, Klaus, Hung, Yin P, Carrasco, Ruben D, Knott, Aine, Gokhale, Prafulla C, Sharma, Sunil, Pozhitkov, Alex, Kulkarni, Prakash, Frank, David A, Salgia, Ravi, Griffin, James D, Saladi, Srinivas V, Bueno, Raphael, Sattler, Martin
Published in British journal of cancer (17.08.2021)
Published in British journal of cancer (17.08.2021)
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3D tissue engineered plasma cultures support leukemic proliferation and induces drug resistance
Alhallak, Kinan, de la Puente, Pilar, Jeske, Amanda, Sun, Jennifer, Muz, Barbara, Rettig, Michael P., Sahin, Ilyas, Weisberg, Ellen L., Griffin, James D., Reagan, John L., DiPersio, John F., Azab, Abdel Kareem
Published in Leukemia & lymphoma (24.08.2021)
Published in Leukemia & lymphoma (24.08.2021)
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Synergy between BRD9- and IKZF3-Targeting as a Therapeutic Strategy for Multiple Myeloma
Chowdhury, Basudev, Garg, Swati, Ni, Wei, Sattler, Martin, Sanchez, Dana, Meng, Chengcheng, Akatsu, Taisei, Stone, Richard, Forrester, William, Harrington, Edmund, Buhrlage, Sara J, Griffin, James D, Weisberg, Ellen
Published in Cancers (01.04.2024)
Published in Cancers (01.04.2024)
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Characterization of AMN107, a selective inhibitor of native and mutant Bcr-Abl
Weisberg, Ellen, Manley, Paul W., Breitenstein, Werner, Brüggen, Josef, Cowan-Jacob, Sandra W., Ray, Arghya, Huntly, Brian, Fabbro, Doriano, Fendrich, Gabriele, Hall-Meyers, Elizabeth, Kung, Andrew L., Mestan, Jürgen, Daley, George Q., Callahan, Linda, Catley, Laurie, Cavazza, Cara, Mohammed, Azam, Neuberg, Donna, Wright, Renee D., Gilliland, D. Gary, Griffin, James D.
Published in Cancer cell (01.02.2005)
Published in Cancer cell (01.02.2005)
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Acute myeloid leukemia cells require 6-phosphogluconate dehydrogenase for cell growth and NADPH-dependent metabolic reprogramming
Bhanot, Haymanti, Weisberg, Ellen L, Reddy, Mamatha M, Nonami, Atsushi, Neuberg, Donna, Stone, Richard M, Podar, Klaus, Salgia, Ravi, Griffin, James D, Sattler, Martin
Published in Oncotarget (15.09.2017)
Published in Oncotarget (15.09.2017)
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Inhibition of SDF-1-induced migration of oncogene-driven myeloid leukemia by the L-RNA aptamer (Spiegelmer), NOX-A12, and potentiation of tyrosine kinase inhibition
Weisberg, Ellen L, Sattler, Martin, Azab, Abdel Kareem, Eulberg, Dirk, Kruschinski, Anna, Manley, Paul W, Stone, Richard, Griffin, James D
Published in Oncotarget (15.12.2017)
Published in Oncotarget (15.12.2017)
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Inhibitors of the Transcription Factor STAT3 Decrease Growth and Induce Immune Response Genes in Models of Malignant Pleural Mesothelioma (MPM)
Lapidot, Moshe, Case, Abigail E, Larios, Dalia, Gandler, Helen I, Meng, Chengcheng, Tošić, Isidora, Weisberg, Ellen L, Poitras, Michael J, Gokhale, Prafulla C, Paweletz, Cloud P, Podar, Klaus, Salgia, Ravi, Saladi, Srinivas V, Griffin, James D, Frank, David A, Bueno, Raphael, Sattler, Martin
Published in Cancers (22.12.2020)
Published in Cancers (22.12.2020)
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Inhibition of Wild-Type p53-Expressing AML by the Novel Small Molecule HDM2 Inhibitor CGM097
Weisberg, Ellen, Halilovic, Ensar, Cooke, Vesselina G, Nonami, Atsushi, Ren, Tao, Sanda, Takaomi, Simkin, Irene, Yuan, Jing, Antonakos, Brandon, Barys, Louise, Ito, Moriko, Stone, Richard, Galinsky, Ilene, Cowens, Kristen, Nelson, Erik, Sattler, Martin, Jeay, Sebastien, Wuerthner, Jens U, McDonough, Sean M, Wiesmann, Marion, Griffin, James D
Published in Molecular cancer therapeutics (01.10.2015)
Published in Molecular cancer therapeutics (01.10.2015)
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