Kilogram-Scale Synthesis of the CXCR4 Antagonist GSK812397
Boggs, Sharon, Elitzin, Vassil I, Gudmundsson, Kristjan, Martin, Michael T, Sharp, Matthew J
Published in Organic process research & development (17.07.2009)
Published in Organic process research & development (17.07.2009)
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Journal Article
An Enyne Cycloisomerization Approach to the Triple Reuptake Inhibitor GSK1360707F
Deschamps, Nicole M, Elitzin, Vassil I, Liu, Bing, Mitchell, Mark B, Sharp, Matthew J, Tabet, Elie A
Published in Journal of organic chemistry (21.01.2011)
Published in Journal of organic chemistry (21.01.2011)
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Journal Article
Development of a New Synthesis for the Large-Scale Preparation of Triple Reuptake Inhibitor (−)-GSK1360707
Elitzin, Vassil I, Harvey, Kimberly A, Kim, Hyunjung, Salmons, Matthew, Sharp, Matthew J, Tabet, Elie A, Toczko, Matthew A
Published in Organic process research & development (16.07.2010)
Published in Organic process research & development (16.07.2010)
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Journal Article
Development of Large-Scale Routes to Potent GPR119 Receptor Agonists
Matsuoka, Richard T, Boros, Eric E, Brown, Andrew D, Bullock, Kae M, Canoy, Will L, Carpenter, Andrew J, Cobb, Jeremy D, Condon, Shannon E, Deschamps, Nicole M, Elitzin, Vassil I, Erickson, Greg, Fang, Jing M, Igo, David H, Joshi, Biren K, Kaldor, Istvan W, Mitchell, Mark B, Peckham, Gregory E, Reynolds, Daniel W, Salmon, Matthew C, Sharp, Matthew J, Tabet, Elie A, Toczko, Jennifer F, Wu, Lianming Michael, Zhou, Xiao-ming M
Published in Organic process research & development (19.08.2016)
Published in Organic process research & development (19.08.2016)
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Journal Article
Function-Oriented Synthesis: Studies Aimed at the Synthesis and Mode of Action of 1α-Alkyldaphnane Analogues
Wender, Paul A, D'Angelo, Noel, Elitzin, Vassil I, Ernst, Martin, Jackson-Ugueto, Eileen E, Kowalski, John A, McKendry, Sharon, Rehfeuter, Markus, Sun, Robert, Voigtlaender, David
Published in Organic letters (26.04.2007)
Published in Organic letters (26.04.2007)
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Journal Article
Synthesis of 7-trifluoromethylpyrazolo[1,5-a]pyridinedicarboxylate
Chong, Pek, Davis, Roman, Elitzin, Vassil, Hatcher, Mark, Liu, Bing, Salmons, Matthew, Tabet, Elie
Published in Tetrahedron letters (12.12.2012)
Published in Tetrahedron letters (12.12.2012)
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Journal Article
Abstract ND12: TNG260: A novel, orally active, CoREST-selective deacetylase inhibitor for the treatment of STK11-mutant cancers
Ahronian, Leanne G., Zhang, Minjie, Min, Chengyin, Tsai, Alice W., Ermolieff, Jacques, McCarren, Patrick, Wyman, Margaret, Guerin, David, Wang, Ye, Bejnood, Alborz, Amemiya, Kenjie, McMillan, Brian, Das, Nikitha, Shahagadkar, Preksha, Doyon, Brian, Mignault, Andre, Liang, Colin, Elitzin, Vassil, Meier, Samuel R., Choi, Ashley, Yu, Yi, Maxwell, John P., Haines, Brian B., Andersen, Jannik N., DiBenedetto, Heather, Weitzman, Aaron, Huang, Alan, Wu, Xinyuan
Published in Cancer research (Chicago, Ill.) (29.05.2023)
Published in Cancer research (Chicago, Ill.) (29.05.2023)
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Journal Article
Effects of nitrogen and alkene substitution on the PtCl sub(2 catalyzed cycloisomerization of N-tethered 1,6-enyne precursors to the triple reuptake inhibitor GSK1360707)
Elitzin, Vassil, Liu, Bing, Sharp, Matthew, Tabet, Elie
Published in Tetrahedron letters (06.07.2011)
Published in Tetrahedron letters (06.07.2011)
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Journal Article
444 TNG260, a CoREST-selective deacetylase inhibitor, reverses anti-PD1 resistance driven by loss of STK11
Ahronian, Leanne, Wu, Xinyuan, Zhang, Minjie, Min, Chengyin, Tsai, Alice, Ermolieff, Jacques, McCarren, Patrick, Wyman, Margaret, Wang, Ye, Bejnood, Alborz, Amemiya, Kenjie, McMillan, Brian, Das, Nikitha, Doyon, Brian, Mignault, Andre, Liang, Colin, Elitzin, Vassil, Yu, Yi, Meier, Samuel, Choi, Ashley, Maxwell, John, Huang, Alan
Published in Journal for immunotherapy of cancer (01.11.2022)
Published in Journal for immunotherapy of cancer (01.11.2022)
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Journal Article
Biological and Structural Characterization of Rotamers of C–C Chemokine Receptor Type 5 (CCR5) Inhibitor GSK214096
Kazmierski, Wieslaw M, Danehower, Susan, Duan, Maosheng, Ferris, Robert G, Elitzin, Vassil, Minick, Douglas, Sharp, Matthew, Stewart, Eugene, Villeneuve, Manon
Published in ACS medicinal chemistry letters (11.12.2014)
Published in ACS medicinal chemistry letters (11.12.2014)
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Journal Article
Function-oriented synthesis: studies aimed at the synthesis and mode of action of 1alpha-alkyldaphnane analogues
Wender, Paul A, D'Angelo, Noel, Elitzin, Vassil I, Ernst, Martin, Jackson-Ugueto, Eileen E, Kowalski, John A, McKendry, Sharon, Rehfeuter, Markus, Sun, Robert, Voigtlaender, David
Published in Organic letters (26.04.2007)
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Published in Organic letters (26.04.2007)
Journal Article