Synthesis, antimicrobial evaluation, DNA gyrase inhibition, and in silico pharmacokinetic studies of novel quinoline derivatives
El‐Shershaby, Mohamed H., El‐Gamal, Kamal M., Bayoumi, Ashraf H., El‐Adl, Khaled, Ahmed, Hany E. A., Abulkhair, Hamada S.
Published in Archiv der Pharmazie (Weinheim) (01.02.2021)
Published in Archiv der Pharmazie (Weinheim) (01.02.2021)
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Journal Article
From triazolophthalazines to triazoloquinazolines: A bioisosterism-guided approach toward the identification of novel PCAF inhibitors with potential anticancer activity
El-Shershaby, Mohamed H., Ghiaty, Adel, Bayoumi, Ashraf H., Al-Karmalawy, Ahmed A., Husseiny, Ebtehal M., El-Zoghbi, Mona S., Abulkhair, Hamada S.
Published in Bioorganic & medicinal chemistry (15.07.2021)
Published in Bioorganic & medicinal chemistry (15.07.2021)
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Journal Article
The antimicrobial potential and pharmacokinetic profiles of novel quinoline-based scaffolds: synthesis and in silico mechanistic studies as dual DNA gyrase and DHFR inhibitors
El-Shershaby, Mohamed H., El-Gamal, Kamal M., Bayoumi, Ashraf H., El-Adl, Khaled, Alswah, Mohamed, Ahmed, Hany E. A., Al-Karmalamy, Ahmed A., Abulkhair, Hamada S.
Published in New journal of chemistry (21.08.2021)
Published in New journal of chemistry (21.08.2021)
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Journal Article
1,2,4-Triazolo[4,3-]quinazolines: a bioisosterism-guided approach towards the development of novel PCAF inhibitors with potential anticancer activity
El-Shershaby, Mohamed H, Ghiaty, Adel, Bayoumi, Ashraf H, Ahmed, Hany E. A, El-Zoghbi, Mona S, El-Adl, Khaled, Abulkhair, Hamada S
Published in New journal of chemistry (07.07.2021)
Published in New journal of chemistry (07.07.2021)
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Journal Article
The antimicrobial potential and pharmacokinetic profiles of novel quinoline-based scaffolds: synthesis and mechanistic studies as dual DNA gyrase and DHFR inhibitors
El-Shershaby, Mohamed H, El-Gamal, Kamal M, Bayoumi, Ashraf H, El-Adl, Khaled, Alswah, Mohamed, Ahmed, Hany E. A, Al-Karmalamy, Ahmed A, Abulkhair, Hamada S
Published in New journal of chemistry (09.08.2021)
Published in New journal of chemistry (09.08.2021)
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Journal Article