Design, synthesis, molecular docking and anticancer evaluations of 5-benzylidenethiazolidine-2,4-dione derivatives targeting VEGFR-2 enzyme
El-Adl, Khaled, El-Helby, Abdel-Ghany A., Sakr, Helmy, Eissa, Ibrahim H., El-Hddad, Sanadelaslam S.A., M.I.A. Shoman, Fatma
Published in Bioorganic chemistry (01.09.2020)
Published in Bioorganic chemistry (01.09.2020)
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Design, synthesis, molecular docking, and anticancer evaluations of 1‐benzylquinazoline‐2,4(1H,3H)‐dione bearing different moieties as VEGFR‐2 inhibitors
El‐Adl, Khaled, El‐Helby, Abdel‐Ghany A., Sakr, Helmy, El‐Hddad, Sanadelaslam S. A.
Published in Archiv der Pharmazie (Weinheim) (01.08.2020)
Published in Archiv der Pharmazie (Weinheim) (01.08.2020)
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Design, synthesis, molecular docking, anticancer evaluations, and in silico pharmacokinetic studies of novel 5‐[(4‐chloro/2,4‐dichloro)benzylidene]thiazolidine‐2,4‐dione derivatives as VEGFR‐2 inhibitors
El‐Adl, Khaled, El‐Helby, Abdel‐Ghany A., Sakr, Helmy, Ayyad, Rezk R., Mahdy, Hazem A., Nasser, Mohamed, Abulkhair, Hamada S., El‐Hddad, Sanadelaslam S. A.
Published in Archiv der Pharmazie (Weinheim) (01.02.2021)
Published in Archiv der Pharmazie (Weinheim) (01.02.2021)
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Design, synthesis, docking, ADMET profile, and anticancer evaluations of novel thiazolidine‐2,4‐dione derivatives as VEGFR‐2 inhibitors
El‐Adl, Khaled, Sakr, Helmy, El‐Hddad, Sanadelaslam S. A., El‐Helby, Abdel‐Ghany A., Nasser, Mohamed, Abulkhair, Hamada S.
Published in Archiv der Pharmazie (Weinheim) (01.07.2021)
Published in Archiv der Pharmazie (Weinheim) (01.07.2021)
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Design, synthesis, and docking of novel thiazolidine‐2,4‐dione multitarget scaffold as new approach for cancer treatment
Hanafy, Noura S., Aziz, Nada A. A. M., El‐Hddad, Sanadelaslam S. A., Abdelgawad, Mohamed A., Ghoneim, Mohammed M., Dawood, Amal F., Mohamady, Samy, El‐Adl, Khaled, Ahmed, Sahar
Published in Archiv der Pharmazie (Weinheim) (01.07.2023)
Published in Archiv der Pharmazie (Weinheim) (01.07.2023)
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Iodoquinazoline-derived VEGFR-2 and EGFRT790M dual inhibitors: Design, synthesis, molecular docking and anticancer evaluations
Mohamed, Abeer A., El-Hddad, Sanadelaslam S.A., Aljohani, Ahmed K.B., Khedr, Fathalla, Alatawi, Omar M., Keshek, Doaa E., Ahmed, Sahar, Alsulaimany, Marwa, Almadani, Sara A., El‐Adl, Khaled, Hanafy, Noura S.
Published in Bioorganic chemistry (01.02.2024)
Published in Bioorganic chemistry (01.02.2024)
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Design, Molecular Docking, Synthesis, Anticancer and Anti-Hyperglycemic Assessments of Thiazolidine-2,4-diones Bearing Sulfonylthiourea Moieties as Potent VEGFR-2 Inhibitors and PPARγ Agonists
Abdelgawad, Mohamed A, El-Adl, Khaled, El-Hddad, Sanadelaslam S A, Elhady, Mostafa M, Saleh, Nashwa M, Khalifa, Mohamed M, Khedr, Fathalla, Alswah, Mohamed, Nayl, AbdElAziz A, Ghoneim, Mohammed M, Abd El-Sattar, Nour E A
Published in Pharmaceuticals (Basel, Switzerland) (14.02.2022)
Published in Pharmaceuticals (Basel, Switzerland) (14.02.2022)
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