New quinazolinone‐based derivatives as DHFR/EGFR‐TK inhibitors: Synthesis, molecular modeling simulations, and anticancer activity
El‐Gazzar, Yomna I., Ghaiad, Heba R., El Kerdawy, Ahmed M., George, Riham F., Georgey, Hanan H., Youssef, Khairia M., El‐Subbagh, Hussein I.
Published in Archiv der Pharmazie (Weinheim) (01.01.2023)
Published in Archiv der Pharmazie (Weinheim) (01.01.2023)
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Imidazo[2′,1′:2,3]thiazolo[4,5-d]pyridazinone as a new scaffold of DHFR inhibitors: Synthesis, biological evaluation and molecular modeling study
Ewida, Menna A., Abou El Ella, Dalal A., Lasheen, Deena S., Ewida, Heba A., El-Gazzar, Yomna I., El-Subbagh, Hussein I.
Published in Bioorganic chemistry (01.10.2018)
Published in Bioorganic chemistry (01.10.2018)
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Thiazolo[4,5-d]pyridazine analogues as a new class of dihydrofolate reductase (DHFR) inhibitors: Synthesis, biological evaluation and molecular modeling study
Ewida, Menna A., Abou El Ella, Dalal A., Lasheen, Deena S., Ewida, Heba A., El-Gazzar, Yomna I., El-Subbagh, Hussein I.
Published in Bioorganic chemistry (01.10.2017)
Published in Bioorganic chemistry (01.10.2017)
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