Cell-based optimization of novel benzamides as potential antimalarial leads
Wu, Tao, Nagle, Advait, Sakata, Tomoyo, Henson, Kerstin, Borboa, Rachel, Chen, Zhong, Kuhen, Kelli, Plouffe, David, Winzeler, Elizabeth, Adrian, Francisco, Tuntland, Tove, Chang, Jonathan, Simerson, Susan, Howard, Steven, Ek, Jared, Isbell, John, Deng, Xianming, Gray, Nathanael S., Tully, David C., Chatterjee, Arnab K.
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
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Imidazolopiperazines: Lead Optimization of the Second-Generation Antimalarial Agents
Nagle, Advait, Wu, Tao, Kuhen, Kelli, Gagaring, Kerstin, Borboa, Rachel, Francek, Caroline, Chen, Zhong, Plouffe, David, Lin, Xuena, Caldwell, Christopher, Ek, Jared, Skolnik, Suzanne, Liu, Fenghua, Wang, Jianling, Chang, Jonathan, Li, Chun, Liu, Bo, Hollenbeck, Thomas, Tuntland, Tove, Isbell, John, Chuan, Tiffany, Alper, Philip B, Fischli, Christoph, Brun, Reto, Lakshminarayana, Suresh B, Rottmann, Matthias, Diagana, Thierry T, Winzeler, Elizabeth A, Glynne, Richard, Tully, David C, Chatterjee, Arnab K
Published in Journal of medicinal chemistry (10.05.2012)
Published in Journal of medicinal chemistry (10.05.2012)
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Journal Article
Imidazolopiperazines: Hit to Lead Optimization of New Antimalarial Agents
Wu, Tao, Nagle, Advait, Kuhen, Kelli, Gagaring, Kerstin, Borboa, Rachel, Francek, Caroline, Chen, Zhong, Plouffe, David, Goh, Anne, Lakshminarayana, Suresh B, Wu, Jeanette, Ang, Hui Qing, Zeng, Peiting, Kang, Min Low, Tan, William, Tan, Maria, Ye, Nicole, Lin, Xuena, Caldwell, Christopher, Ek, Jared, Skolnik, Suzanne, Liu, Fenghua, Wang, Jianling, Chang, Jonathan, Li, Chun, Hollenbeck, Thomas, Tuntland, Tove, Isbell, John, Fischli, Christoph, Brun, Reto, Rottmann, Matthias, Dartois, Veronique, Keller, Thomas, Diagana, Thierry, Winzeler, Elizabeth, Glynne, Richard, Tully, David C, Chatterjee, Arnab K
Published in Journal of medicinal chemistry (28.07.2011)
Published in Journal of medicinal chemistry (28.07.2011)
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Discovery of novel 1H-imidazol-2-yl-pyrimidine-4,6-diamines as potential antimalarials
Deng, Xianming, Nagle, Advait, Wu, Tao, Sakata, Tomoyo, Henson, Kerstin, Chen, Zhong, Kuhen, Kelli, Plouffe, David, Winzeler, Elizabeth, Adrian, Francisco, Tuntland, Tove, Chang, Jonathan, Simerson, Susan, Howard, Steven, Ek, Jared, Isbell, John, Tully, David C., Chatterjee, Arnab K., Gray, Nathanael S.
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
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Journal Article
A strategy to profile prime and non-prime proteolytic substrate specificity
Petrassi, H. Michael, Williams, Jennifer A., Li, Jun, Tumanut, Christine, Ek, Jared, Nakai, Takashi, Masick, Brian, Backes, Bradley J., Harris, Jennifer L.
Published in Bioorganic & medicinal chemistry letters (15.06.2005)
Published in Bioorganic & medicinal chemistry letters (15.06.2005)
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Journal Article
Substrate Profiling of Deubiquitin Hydrolases with a Positional Scanning Library and Mass Spectrometry
Mason, Daniel E, Ek, Jared, Peters, Eric C, Harris, Jennifer L
Published in Biochemistry (Easton) (01.06.2004)
Published in Biochemistry (Easton) (01.06.2004)
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Purifying the Masses: Integrating Prepurification Quality Control, High-Throughput LC/MS Purification, and Compound Plating To Feed High-Throughput Screening
Isbell, John J, Zhou, Yingyao, Guintu, Christina, Rynd, Matthew, Jiang, Shumei, Petrov, Dimitri, Micklash, Ken, Mainquist, Jim, Ek, Jared, Chang, Jim, Weselak, Mark, Backes, Bradley J, Brailsford, Andrew, Shave, Darcy
Published in Journal of combinatorial chemistry (01.03.2005)
Published in Journal of combinatorial chemistry (01.03.2005)
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