Expanding control of the tumor cell cycle with a CDK2/4/6 inhibitor
Freeman-Cook, Kevin, Hoffman, Robert L., Miller, Nichol, Almaden, Jonathan, Chionis, John, Zhang, Qin, Eisele, Koleen, Liu, Chaoting, Zhang, Cathy, Huser, Nanni, Nguyen, Lisa, Costa-Jones, Cinthia, Niessen, Sherry, Carelli, Jordan, Lapek, John, Weinrich, Scott L., Wei, Ping, McMillan, Elizabeth, Wilson, Elizabeth, Wang, Tim S., McTigue, Michele, Ferre, Rose Ann, He, You-Ai, Ninkovic, Sacha, Behenna, Douglas, Tran, Khanh T., Sutton, Scott, Nagata, Asako, Ornelas, Martha A., Kephart, Susan E., Zehnder, Luke R., Murray, Brion, Xu, Meirong, Solowiej, James E., Visswanathan, Ravi, Boras, Britton, Looper, David, Lee, Nathan, Bienkowska, Jadwiga R., Zhu, Zhou, Kan, Zhengyan, Ding, Ying, Mu, Xinmeng Jasmine, Oderup, Cecilia, Salek-Ardakani, Shahram, White, Michael A., VanArsdale, Todd, Dann, Stephen G.
Published in Cancer cell (11.10.2021)
Published in Cancer cell (11.10.2021)
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Efficacy of SERD/SERM Hybrid-CDK4/6 Inhibitor Combinations in Models of Endocrine Therapy-Resistant Breast Cancer
Wardell, Suzanne E, Ellis, Matthew J, Alley, Holly M, Eisele, Koleen, VanArsdale, Todd, Dann, Stephen G, Arndt, Kim T, Primeau, Tina, Griffin, Elizabeth, Shao, Jieya, Crowder, Robert, Lai, Jin-Ping, Norris, John D, McDonnell, Donald P, Li, Shunqiang
Published in Clinical cancer research (15.11.2015)
Published in Clinical cancer research (15.11.2015)
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Discovery of Highly Selective Inhibitors of Microtubule-Associated Serine/Threonine Kinase-like (MASTL)
Gallego, Rebecca A., Scales, Stephanie, Toledo, Chad, Auth, Marin, Bernier, Louise, Berry, Madeline, Brun, Sonja, Chung, Loanne, Davis, Carl, Diehl, Wade, Dress, Klaus, Eisele, Koleen, Elleraas, Jeff, Ewanicki, Jason, Fobian, Yvette, Greasley, Samantha, Greenwald, Eric C., Johnson, Ted W., Khamphavong, Penney, Lafontaine, Jennifer, Li, Jian, Linton, Angelica, Maestre, Michael, Miller, Nichol, Murtaza, Anwar, Patman, Ryan L., Quinlan, Casey L., Ramms, Dana J., Richardson, Paul, Sach, Neal, Salomon-Ferrer, Romelia, Silva, Francisco, Timofeevski, Sergei, Tran, Phuong, Tran-Dubé, Michelle, Wang, Fen, Wang, Wei, Wythes, Martin, Yang, Shouliang, Zou, Aihua, VanArsdale, Todd, McAlpine, Indrawan
Published in Journal of medicinal chemistry (05.11.2024)
Published in Journal of medicinal chemistry (05.11.2024)
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Abstract 2960: A novel mouse model of pancreatic cancer reveals new insights into cell cycle deregulation
Adams, Christina, Wang, Lynn, Wang, Tim S., Miller, Nichol, McMillan, Elizabeth, Ramstetter, Monica, Chionis, John, Eisele, Koleen, Almaden, Jonathan, Affolter, Timothy, Pillai, Smitha, VanArsdale, Todd, Dillon, Chris, Dann, Stephen G.
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Abstract 5709: PF-07104091, a first-in-class CDK2-selective inhibitor for the treatment of HR+/HER2- breast cancer and CCNE1high ovarian cancer
Shen, Chen, Qiu, Ming, Huser, Nanni, Pascual, Bernadette, Zhang, Qin, VanArsdale, Todd, Murtaza, Anwar, Almaden, Jonathan, Kim, berly, Anders, Lars, Eisele, Koleen
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Abstract 330: Engineering electrophile-sensitive kinase mutants to accelerate oncology target validation
Oyer, Jon A., Johnson, Ted W., Wang, Andrew C., Maestre, Michael F., Flores-Bojorquez, Ana, Melnychuk, Roksolana, Timofeevski, Sergei, Niessen, Sherry, Wang, Zhenxiong, Li, Jian, Diehl, Wade C., Eisele, Koleen J., Lee, Nathan V., Zou, Aihua, Davis, Carl, Greenwald, Eric C., DeForest, Jacob, Ornelas, Martha, Li, Bryan, Scales, Stephanie, Khamphavong, Penney L., Ambler, Catherine M., Huang, Yun, Salomon-Ferrer, Romelia, Greasley, Samantha E., Bolanos, Ben, Grodsky, Neil, Lum, Lawrence, VanArsdale, Todd L., McAlpine, Indrawan J.
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Axitinib and crizotinib combination therapy inhibits bone loss in a mouse model of castration resistant prostate cancer
Eswaraka, Jeetendra, Giddabasappa, Anand, Han, Guangzhou, Lalwani, Kush, Eisele, Koleen, Feng, Zheng, Affolter, Timothy, Christensen, James, Li, Gang
Published in BMC cancer (02.10.2014)
Published in BMC cancer (02.10.2014)
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Abstract A08: Mechanistic basis of Palbociclib combinatorial activity in ER+ breast cancer and non-breast indications
Dann, Stephen, Chionis, John, Choating, Liu, Chen, Enhong, Wei, Ping, Eisele, Koleen, Shields, David J., Rejto, Paul A., VanArsdale, Todd
Published in Molecular cancer research (01.11.2016)
Published in Molecular cancer research (01.11.2016)
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Abstract 5903: MASTL small-molecule inhibition to target mitosis for cancer therapy
Toledo, Chad M., Eisele, Koleen J., Kim, Dong Hyun, Mu, Xinmeng, Brun, Sonja, Davis, Carl, Greenwald, Eric C., Hui, Fion, He, Meilan, Yang, Yanling, Flores-Bojorquez, Ana, Li, Yuxin, Khamphavong, Penney L., Lee, Joseph H., Li, Jian, Ramms, Dana J., Jones, Greg, Auth, Marin, Painter, Cory L., Nager, Andrew, Oyer, Jon, Timofeevski, Sergei L., Pierceall, William E., Murtaza, Anwar, Heyen, Jonathan R., Gallego, Rebecca, Quinlan, Casey, McAlpine, Indrawan, VanArsdale, Todd L.
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Abstract LB-136: Mechanistic exploration of combined CDK4/6 and ER inhibition in ER-positive breast cancer
Lee, Nathan V., Yuan, Jing, Eisele, Koleen, Cao, Joan Q., Painter, Cory L., Chionis, John, Liu, Chaoting, Shields, David J., Kan, Julie L.C., Arndt, Kim, VanArsdale, Todd
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Abstract 2817: Preclinical studies of the PI3K/mTOR dual inhibitors in endometrial cancer cell lines
Yuan, Jing, Garza, Scott J., Cao, Joan, Fisher, Timothy S., Lee, Nathan V., Eisele, Koleen, Pasis, Angela, Hook, Kenneth, Christensen, James G., Kan, Julie L.
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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COMBINATION THERAPIES AND USES FOR TREATING CANCER
SHARMA, Shikhar, WANG, Hui, DANN, Stephen George, KUNG, Pei-Pei, KRAUS, Manfred, EISELE, Koleen Jill, FAN, Conglin
Year of Publication 22.06.2023
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Year of Publication 22.06.2023
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